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http://www.dcchemicals.com

D&C Chemicals provides a wide range of research chemicals and biochemicals including novel life-science reagents, reference compounds, APIs and Natural compounds for laboratory and scientific use. D&C Chem has established a global network of thousands of customers from many research centers, Pharmaceutical companies and Reagent companies in the USA, Europe and Japan. The Pharmaceutical companies include: Johnson & Johnson, Pfizer, Novartis,Merk-EMD, Eli Lilly, Sanofi-Aventis and so on.

We are also the official vendor of more than 100 universities and institutes including:Harvard University,Yale University,NIH/NCI,City of Hope ORG, PARTNERS ORG,John Hopkins University, Universittsklinikum,Oxford University,Newcastle University,UNC,UCSF and many other universities and institutes. Our bioactive compounds received good feedback from our customers.


Product List: 5,720

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Product List

(+)-ARGLABIN
CAS:84692-91-1
Trade Name: Arglabin
Formula: C15H18O3
DC9645
>98%
Arglabin is a sesquiterpene gamma-lactone is isolated from Artemisia glabella; anticancer natural compound.
(+)-BICUCULLINE
CAS:485-49-4
Formula: C20H17NO6
DC10625
>98%
(+)-Bicuculline is a competitive antagonist of GABAA receptors with IC50 of 2 M, also blocks Ca(2+)-activated potassium channels.
(+)-CORYNOLINE
CAS:18797-79-0
Formula: C21H21NO5
DCZ-007
>98%,Standard References Grade
>98%,Standard References
(+)-ETOMOXIR (SODIUM SALT)
CAS:828934-41-4
Formula: C15H18ClNaO4
DC7412
>98%
A PPARa agonist and an irreversible CPT-1 inhibitor.
(+)-JQ1
CAS:1268524-70-4
Trade Name: JQ-1,JQ 1,JQ1,+JQ 1,+JQ-1,+JQ1
Formula: C23H25ClN4O2S
DC5019
HPLC Purity>99%,ee purity>99%
(+)-JQ1 is a BET bromodomain inhibitor, binding to all bromodomains of the BET family, but not to bromodomains outside the BET family.
(+)-NARWEDINE
CAS:7318-5-0
Trade Name: D-Narwedine,(+)Narwedine,+Narwedine
Formula: C17H19NO3
DC9976
>98%
(+)-Narwedine. Galantamine(Narwedin) is a competitive and reversible cholinesterase(AChE) inhibitor.
(+)-USNIACIN
CAS:7562-61-0
Formula: C18H16O7
DCS-001
>98%,Standard References Grade
>98%,Standard References
(+)MK-801 MALEATE
CAS:77086-22-7
Trade Name: MK 801 ,MK801
Formula: C20H19NO4
DC7960
>98%
Dizocilpine maleate(MK 801) is a potent N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 30.5 nM
(+)PD 128907
CAS:300576-59-4
Formula: C14H19NO3.HCl
DC5060
>98%
(+)PD 128907 is a potent D3 dopamine receptor agonist (Ki = 2.3 nM). Displays 18 - 200-fold selectivity over other dopamine receptor subtypes.
(+,-)-OCTOPAMINE HCL
CAS:770-05-8,4502-14-1,104-14-3(freebase)
Trade Name: N/A
Formula: C8H11NO2.HCl
DCAPI1338
>99%
Octopamine (OA), a biogenic monoamine structurally related to noradrenaline, acts as a neurohormone, a neuromodulator and a neurotransmitter in invertebrates.
(+/-)-SULFINPYRAZONE
CAS:57-96-5
Trade Name: (+/-)-Sulfinpyrazone
Formula: C23H20N2O3S
DC10268
>98%
Sulfinpyrazone is one of the most studied platelet COX inhibitors, also a uricosuric agent that competitively inhibits uric acid reabsorption in kidney proximal tubules.
(-)-ASARININ
CAS:133-04-0
Formula: C20H18O6
DCX-016
>98%,Standard References Grade
>98%,Standard References
(-)-EPICATECHIN GALLATE
CAS:1257-08-5
Formula: C22H18O10
DCB-022
>98%,Standard References Grade
>98%,Standard References
(-)-EPIGALLOCATECHIN
CAS:970-74-1
Formula: C15H14O7
DCB-021
>98%,Standard References Grade
>98%,Standard References
(-)-EPIGALLOCATECHIN GALLATE
CAS:989-51-5
Formula: C22H18O11
DCB-023
>98%,Standard References Grade
>98%,Standard References
(-)-GALLOCATECHIN
CAS:3371-27-5
Formula: C15H14O7
DCZ-267
>98%
>98%,Standard References
(-)-GALLOCATECHIN GALLATE
CAS:4233-96-9
Formula: C22H18O11
DCM-059
>98%,Standard References Grade
>98%,Standard References
(-)-HUPERZINE A
CAS:102518-79-6
Formula: C15H18N2O
DCS-019
>98%,Standard References Grade
>98%,Standard References
(-)-JQ-1
CAS:1268524-71-5
Trade Name: JQ-1,JQ1,-JQ1,JQ 1
Formula: C23H25ClN4O2S
DC8261
>98%,ee>99%
The (-)-JQ1 stereoisomer has no appreciable affinity to BET bromodomains,it is the negative control of +JQ-1.
(-)-LICARIN B
CAS:51020-87-2
Formula: C20H20O4
DCL-044
>98%,Standard References Grade
>98%,Standard References
(-)-NARWEDINE
CAS:510-77-0
Trade Name: L-Narwedine
Formula: C17H19NO3
DC7861
>98%
Galantamine(Narwedin) is a competitive and reversible cholinesterase(AChE) inhibitor.
(-)-SPARTEINE (SULFATE PENTAHYDRATE)
CAS:6160-12-9
Trade Name: (-)-Sparteine sulfate salt;Lupinidine sulfate pentahydrate
Formula: C15H28N2O4S
DC9624
>98%
(-)-Sparteine sulfate pentahydrate is a class 1a antiarrhythmic agent and a sodium channel blocker.
(-)-STYLOPINE
CAS:4312-32-7
Formula: C19H17NO4
DCZ-103
>98%
>98%,Standard References
(-)-SYRINGARESNOL-4-O-SS-D-APIOFURANOSYL-(1 2)-SS-D-GLUCOPYRANOSIDE
CAS:136997-64-3
Formula: C33H44O17
DCD-050
>98%,Standard References Grade
>98%,Standard References
(-)BLEBBISTATIN
CAS:856925-71-8
Formula: C18H16N2O2
DC7818
>98%
(-)-Blebbistatin is a cell-permeable inhibitor for non muscle myosin II ATPase with IC50 of ~2 M, does not inhibit myosin light chain kinase, inhibits contraction of the cleavage furrow without disrupting mitosis or contractile ring assembly.
(-)MK-801 MALEATE
CAS:121917-57-5
Trade Name: MK 801 ,MK801
Formula: C20H19NO4
DC7961
>98%
(-)-MK 801 Maleate is the enantiomer of (+)-MK-801; (+)-MK-801 is a highly potent and selective non-competitive NMDA glutamate receptor antagonist .
()-HUPERZINE A
CAS:120786-18-7
Trade Name: Huperzine a
Formula: C15H18N2O
DC9329
>98%
Huperzine A, an active Lycopodium alkaloid extracted from traditional Chinese herb, is a potent, selective and reversible acetylcholinesterase (AChE) inhibitor and has been widely used in China for the treatment of Alzheimer's disease (AD).
()-PIRMENOL
CAS:68252-19-7
Formula: C22H30N2O
DC10364
>98%
Pirmenol inhibits IK.ACh by blocking muscarinic receptors. The IC50 of Pirmenol for inhibition of Carbachol-induced IK.ACh is 0.1 M.
()-SLV319(IBIPINABANT)
CAS:362519-49-1
Trade Name: SLV 319,SLV-319
Formula: C23H20Cl2N4O2S
DC10094
>98%
()-SLV 319 is a potent and selective CB1 receptor antagonist (Ki = 7.8 nM). Exhibits 1000-fold selectivity for CB1 over CB2 receptors.
(1R,2S)-VU0155041
CAS:1263273-14-8
Formula: C14H15Cl2NO3
DC10160
>98%
(1R,2S)-VU0155041, Cis regioisomer of VU0155041, is a partial mGluR4 agonist with an EC50 of 2.35 M.
(1S,3R,5R)-PIM447 DIHYDROCHLORIDE
Trade Name: (1S,3R,5R)-LGH447 dihydrochloride
Formula: C24H25Cl2F3N4O
DC10428
>98%
(1S,3R,5R)-PIM447 (dihydrochloride) an PIM inhibitor extracted from patent US 20100056576 A1, compound example 72, has IC50 values of 0.095 M for Pim1, 0.522 M for Pim2 and 0.369 M for Pim3.
(20S)-PROTOPANAXADIOL
CAS:30636-90-9
Formula: C30H52O3
DC9833
>98%
(20S)-Protopanaxadiol (20-Epiprotopanaxadiol) is an aglycon metabolic derivative of the protopanaxadiol-type ginseng saponin; apoptosis inducer.
(2R,3S)-3-PHENYLISOSERINE HYDROCHLORIDE
CAS:132201-32-2
Formula: C9H12ClNO3
DCZ-166
>98%
>98%,Standard References
(E)-[6]-DEHYDROPARADOL
CAS:878006-06-5
Formula: C17H24O3
DC10426
>98%
(E)-[6]-Dehydroparadol, extracted from patent US 9272994, compound M15, shows growth inhibition and induction of apoptosis against human cancer cells with IC50 values of 43.02 M in HCT-116 cell and 41.59 M in H-1299 cell, respectively.
(R)-(+)-CORYPALMINE
CAS:13063-54-2
Formula: C20H23NO4
DCS-067
>98%,Standard References Grade
>98%,Standard References
(R)-(-)-MODAFINIC ACID
CAS:112111-45-2
Trade Name: Armodafinic acid
Formula: C15H14O3S
DC9558
>98%
(R)-(-)-Modafinic acid(Armodafinic acid) is the major metabolite of Modafinil(HY-10521A), which is a central nervous system vigilance promoting agent, which posseses neuroprotective properties._x000D_IC50 value:_x000D_Target: neuroprotective agent_x000D_
(R)-(-)-ROLIPRAM
CAS:85416-75-7
Trade Name: (R)-Rolipram;(-)-Rolipram
Formula: C16H21NO3
DC9584
>98%
(R)-(-)-Rolipram is a potent and cAMP-specific PDE4 inhibitor with IC50 of 0.22 uM; 2.5-fold more potent than (+)-rolipram (IC50= 2.58 uM) in inhibiting membrane-bound PDE 4._x000D_
(R)-1,2,3,4-TETRAHYDRO-3-ISOQUINOLINECARBOXYLIC ACID
CAS:103733-65-9
Trade Name: D-phenylalanine analogue
Formula: C10H11NO2
DC9533
>98%
(R)-1,2,3,4-Tetrahydro-3-isoquinolinecarboxylic acid is a constrained Phe analogue which can fold into a beta-bend and a helical structure, and to adopt a preferred side-chain disposition in the peptide._x000D_
(R)-BACLOFEN
CAS:69308-37-8
Trade Name: STX 209;STX-209;STX209
Formula: C10H12ClNO2
DC9450
>98%
(R)-Baclofen(STX209) is a selective GABAB receptor agonist.
(R)-BPO-27
CAS:1415390-47-4
Trade Name: (R)-BPO 27; (R)-BPO27
Formula: C26H18BrN3O6
DC10388
>98%
(R)-BPO-27 is a potent CFTR inhibitor with an IC50 of 4 nM
(R)-EQUOL
CAS:221054-79-1
Trade Name: Isoequol
Formula: C15H14O3
DC8450
>98%
In contrast to the estrogen receptor (ER) selectivity of (S)-equol , (R)-equol is a weaker ER agonist that binds to ERa and ER with Ki values of 27.4 and 15.4 nM, respectively.
(R)-IMPP
CAS:N/A
Trade Name: R-IMPP
Formula: C24H27N3O2
DC10521
>98%
(R)-IMPP is a cell-permeable inhibitor of the secretion of proprotein convertase subtilisin/kexin type 9 (PCSK9; IC50 = 4.8 M).
(R)-LANSOPRAZOLE
CAS:138530-94-6
Formula: C16H14F3N3O2S
DC9092
>98%
(R)-Lansoprazole is a proton pump inhibitor which prevents the stomach from producing acid.
(R)-MECLIZINE
CAS:189298-48-4
Formula: C25H27Cl2N2
DC7757
>98%
Meclizine is a histamine H1 receptor antagonist used to treat nausea and motion sickness.
(R)PFI-2 HCL
CAS:1627607-87-7
Trade Name: PFI-2, PFI2,PFI 2,R PFI-2,R-PFI2
Formula: C23H25F4N3O3S
DC7679
>98%
PFI-2 is a novel potent and selective SETD7 histone lysine methyltransferase inhibitor with IC50 ~2 nM. It has > 100-fold selectivity over other methyltransferases and other non-epigenetic targets.
(S)-(+)-KETOPROFEN
CAS:22161-81-5
Formula: C16H14O3
DC9005
>98%
(S)-(+)-MODAFINIC ACID
CAS:112111-44-1
Formula: C15H14O3S
DC9559
>98%
(S)-(+)-Modafinic acid is the major metabolite of Modafinil(HY-10521A), which is a central nervous system vigilance promoting agent, which posseses neuroprotective properties._x000D_IC50 value:_x000D_Target: neuroprotective agent_x000D_
(S)-(+)-ROLIPRAM
CAS:85416-73-5
Trade Name: (+)-Rolipram;(S)-Rolipram
Formula: C16H21NO3
DC9581
>98%
(S)-(+)-Rolipram is a PDE4-inhibitor and an anti-inflammatory agent, less potent than its R enantiomer._x000D_
(S)-AMLODIPINE
CAS:103129-82-4
Formula: C20H25N2O5Cl
DC9122
>98%
(S)-CARBIDOPA
CAS:38821-49-7
Formula: C10H16N2O5
DC8992
>98%
(S)-EQUOL
CAS:531-95-3
Formula: C15H14O3
DC8451
>98%
(S)-Equol preferentially binds ER (Ki = 0.73 nM) and demonstrates approximately 9-fold lower affinity for ERa (Ki = 6.41 nM).
(S)-GOSSYPOL (ACETIC ACID)
CAS:1189561-66-7
Trade Name: (S)-(+)-Gossypol acetic acid
Formula: C32H34O10
DC9368
>98%
(S)-Gossypol acetic acid is a inhibitor of Bcl-2, potently induce cell death in Jurkat cells overexpressing Bcl-2 (IC50, 18.1M) or Bcl-xL (IC50, 22.9M)._x000D_
(S)-KETOPROFEN TROMETAMOL
CAS:156604-79-4
Formula: C16H14O3.C4H11NO3
DC9099
>98%
(S)-PFI-2 HCL
CAS:1627607-88-8
Trade Name: PFI2,PFI-2,SPFI2,SPFI-2,PFI 2,SPFI 2,S-PFI-2
Formula: C23H25F4N3O3S.HCl
DC8290
>97%
Negative control of (R)-PFI 2 hydrochloride. Exhibits 500-fold lower activity in a SETD7 enzymatic assay (IC50 = 1 M) compared to the active enantiomer.
(S)-TEDIZOLID
CAS:1431699-67-0
Trade Name: (S)-3-(3-fluoro-4-(6-(2-methyl-2H-tetrazol-5-yl)pyridin-3-yl)phenyl)-5-(hydroxymethyl)oxazolidin-2-o
Formula: C17H15FN6O3
DC9352
>98%
Tedizolid is the active moiety of the prodrug tedizolid phosphate, with high potency against Gram-positive species._x000D_
(S)GINSENOSIDE RG2
CAS:80952-72-3
Formula: C42H72O13
DCR-038
>98%,Standard References Grade
>98%,Standard References
(Z)-MUTAGENIC IMPURITY OF TENOFOVIR DISOPROXIL
CAS:1464851-21-5
Formula: C8H9N5
DC10396
>98%
(Z)-Mutagenic Impurity of Tenofovir Disoproxil is a mutagenic impurity in tenofovir disoproxil fumarate. Tenofovir is an antiretroviral drug known as nucleotide analogue reverse transcriptase (NtART) inhibitor, which blocks reverse transcriptase, a crucia
1,3,5,8-TETRAHYDROXYLXANTHONE
DCS-097
>98%,Standard References Grade
>98%,Standard References
1,4-DIAMINOBUTANE
CAS:110-60-1
Formula: C4H12N2
DCF-015
>98%,Standard References Grade
>98%,Standard References
1,4-NAPHTHOQUINONE
CAS:130-15-4
Formula: C10H6O2
DCZ-270
>98%
>98%,Standard References
1,7-DIHYDROXY-2,3,8-TRIMETHOXY-6-METHYLANTHRACENE-9,10-DIONE;OBTUSIN
CAS:70588-05-5
Formula: C18H16O7
DCH-071
>98%,Standard References Grade
>98%,Standard References
1,8-DIACETOXY-3-CARBOXYANTHRAQUINONE
CAS:13739-02-1
Formula: C19H12O8
DCS-087
>98%,Standard References Grade
>98%,Standard References
1,8-DIHYDROXYANTHRAQUINONE
CAS:117-10-2
Formula: C14H8O4
DCE-005
>98%,Standard References Grade
>98%,Standard References
1-AZAKENPAULLONE
CAS:676596-65-9
Trade Name: 9-Bromo-7,12-dihydropyrido[3',2':2,3]azepino[4,5-b]indol-6(5H)-one; 1-AKP; kenpaullone;
Formula: C15H10BrN3O
DC5144
>98%
1-Azakenpaullone is a potent and ATP-competitive GSK-3 (glycogen synthase kinase-3) inhibitor (IC50 = 18 nM).
1-DEOXYNOJIRIMYCIN
CAS:19130-96-2
Formula: C6H13NO4
DCT-003
>98%,Standard References Grade
>98%,Standard References
1-HYDROXY-2,3,4,7-TETRAMETHOXYXANTHONE
CAS:14103-09-4
Formula: C17H16O7
DCQ-076
>98%,Standard References Grade
>98%,Standard References
1-KESTOSE
CAS:470-69-9
Formula: C19H34O16
DC9220
>98%
1-METHOXY PMS
CAS:65162-13-2
Trade Name: 1-Methoxy-5-methylphenazinium methylsulfate
Formula: C15H16N2O5S
DC8835
>98%
1-Methoxy PMS is an electron mediator for NAD(P)H-tetrazolium salt.
1-METHYL-7-NITROISATOIC ANHYDRIDE
CAS:73043-80-8
Formula: C9H6N2O5
DC8649
>98%
1-methyl-7-nitroisatoic anhydride is a reagent that detects local nucleotide flexibility, for probing 2'-hydroxyl reactivity.
1-METHYL-L-TRYPTOPHAN
CAS:21339-55-9
Formula: C12H14N2O2
DCX-039
>98%,Standard References Grade
>98%,Standard References
1-NA-PP1
CAS:221243-82-9
Trade Name: 1-Naphthyl PP1
Formula: C19H19N5
DC9281
>98%
1-Naphthyl PP1(1-NA-PP 1) is a selective inhibitor of src family kinases v-Src and c-Fyn as well as the tyrosine kinase c-Abl (IC50 values are 1.0, 0.6, 0.6, 18 and 22 M for v-Src, c-Fyn, c-Abl, CDK2 and CAMK II respectively).
1-NM-PP1
CAS:221244-14-0
Formula: C20H21N5
DC8640
>98%
1-NM-PP1 is a cell permeable inhibitor of kinases that have been mutated, by a single base substitution, to become analog sensitive (as), as compared to the wild-type kinase.
1-O-ACETYL BRITANNILACTONE
CAS:681457-46-5
Formula: C17H24O5
DCZ-155
>98%
>98%,Standard References
1-TRIACONTANOL
CAS:593-50-0
Formula: C30H62O
DCS-050
>98%,Standard References Grade
>98%,Standard References
10-DEACETYLBACCATIN III
CAS:32981-86-5
Formula: C29H36O10
DCT-001
>98%,Standard References Grade
>98%,Standard References
10-GINGEROL
CAS:23513-15-7
Formula: C21H34O4
DCJ-037
>98%,Standard References Grade
>98%,Standard References
10-HYDROXY-2-DECENOIC ACID
CAS:14113-05-4
Formula: C10H18O3
DCQ-026
>98%,Standard References Grade
>98%,Standard References
10-HYDROXYCAMPTOTHECIN
CAS:19685-09-7
Formula: C20H16N2O5
DCQ-011
>98%,Standard References Grade
>98%,Standard References
10-HYDROXYSCANDINE
CAS:119188-47-5
Formula: C21H22N2O4
DCQ-056
>98%,Standard References Grade
>98%,Standard References
10-METHOXYCAMPTOTHECINE
DCJ-063
>98%,Standard References Grade
>98%,Standard References
10058-F4
CAS:403811-55-2
Formula: C12H11NOS2
DC7575
>98%
10058-F4 is a c-Myc inhibitor that specificallly inhibits the c-Myc-Max interaction and prevents transactivation of c-Myc target gene expression.
10074-G5
CAS:413611-93-5
Trade Name: 10074G5,10074 G5
Formula: C18H12N4O3
DC10075
>98%
10074-G5 is a c-Myc Max interaction inhibitor.
13-DEHYDROXYINDACONINTINE
Formula: C34H47NO9
DCQ-066
>98%,Standard References Grade
>98%,Standard References
1400W DIHYDROCHLORIDE
CAS:214358-33-5
Formula: C10H15N3.2HCl
DC9998
>98%
1400W dihydrochloride is a slow, tight binding, potent and highly selective inhibitor of inducible nitric oxide synthase (Kd = 7 nM).
17-AAG
CAS:75747-14-7
Trade Name: Tanespimycin;NSC 330507;CP 127374;17AAG;17 AAG
Formula: C31H43N3O8
DC9482
>98%
17-AAG(NSC 330507; CP 127374) is a potent HSP90 inhibitor with IC50 of 5 nM, having a 100-fold higher binding affinity for HSP90 derived from tumour cells than HSP90 from normal cells._x000D_
18 SS-GLYCYRRHETINTIC ACID
CAS:471-53-4
Formula: C30H46O4
DCG-032
>98%,Standard References Grade
>98%,Standard References
1A,25-DIHYDROXY VITAMIN D2
CAS:60133-18-8
Trade Name: N/A
Formula: C28H44O3
DCAPI1554
>99%
1a,25-Dihydroxyvitamin D2 is an active metabolite of vitamin D. It is known that 1a,25-Dihydroxyvitamin D2 can be detected in human serum using high-performance liquid chromatography and ultraviolet detection. Vitamin D2, known as ergocalciferol, is a fat
2,2'-DIHYDROXY-4-METHOXYBENZOPHENONE
CAS:131-53-3
Trade Name: 2,2'-Dihydroxy-4-methoxybenzophenone
Formula: C14H12O4
DC10243
>98%
Dioxybenzone (benzophenone-8) is an organic compound used in sunscreen to block UVB and short-wave UVA (ultraviolet) rays
2,3,5,4'-TETRAHYDROXY STILBENE-2- -SS-D-GLUCOSIDE
CAS:82373-94-2
Formula: C20H22O9
DCS-029
>98%,Standard References Grade
>98%,Standard References
2,4,5-TRIMETHOXYBENZALDEHYDE
CAS:4460-86-0
Formula: C10H12O4
DCX-067
>98%,Standard References Grade
>98%,Standard References
2,4-PYRIMIDINEDIAMINE WITH LINKER
CAS:1430089-64-7
Trade Name: 2,4-Pyrimidinediamine with linker
Formula: C19H24N8
DC7972
>98%
2,4-Pyrimidinediamine with linker is a patent compound in WO2013055780A1, Page 71; multikinase inhibitor and has a -NH2 terminal linker for further synthesis.
2,5-DIHYDROXYBENZOIC ACID
CAS:490-79-9
Formula: C7H6O4
DCZ-259
>98%
>98%,Standard References
2,6-DIHYDROXYPURINE
CAS:69-89-6
Formula: C5H4N4O2
DCH-069
>98%,Standard References Grade
>98%,Standard References
2-(1-ETHOXYETHOXY) ETHYL)BENZENE
CAS:2556-10-7
Formula: C12H18O2
DCF-023
>98%,Standard References Grade
>98%,Standard References
2-(PYRIDYLDITHIO)ETHYLAMINE HYDROCHLORIDE
CAS:106139-15-5
Trade Name: (S)-2-Pyridylthio cysteamine hydrochloride
Formula: C7H11ClN2S2
DC10184
>98%
2-(Pyridyldithio)ethylamine hydrochloride is a novel disulfideintercalating cross-linking reagent.
2-ADAMANTANOL
CAS:700-57-2
Formula: C10H16O
DCJ-018
>98%,Standard References Grade
>98%,Standard References
2-ADAMANTANONE
CAS:700-58-3
Formula: C10H14O
DCJ-021
>98%,Standard References Grade
>98%,Standard References
2-HYDROXY-1,4-NAPHOQUINONE
CAS:83-72-7
Formula: C10H6O3
DCZ-278
>98%
>98%,Standard References
2-HYDROXY-4-METHOXYBENZALDEHYDE
CAS:673-22-3
Formula: C8H8O3
DCJ-042
>98%,Standard References Grade
>98%,Standard References
2-HYDROXY-N-(4-HYDROXYPHENYL) -BENZAMIDE
CAS:526-18-1
Formula: C13H11NO3
DC8981
>98%
2-HYDROXYADENOSINE
CAS:1818-71-9
Formula: C10H13N5O5
DCB-003
>98%,Standard References Grade
>98%,Standard References
2-METHOXYCINNAMIC ACID
CAS:6099-03-2
Formula: C10H10O3
DCL-018
>98%,Standard References Grade
>98%,Standard References
2-METHOXYESTRADIOL
CAS:362-07-2
Formula: C19H26O3
DC9044
>98%
2-methoxyestradiol (2ME2; NSC-659853) is a natural metabolite of estrogen that is known to inhibit HIF-1 alpha with an IC50 of 0.71 0.11 M for the inhibition of BPAEC migration.
2-METHYLVALERIC ACID
CAS:97-61-0
Formula: C6H12O2
DCE-036
>98%,Standard References Grade
>98%,Standard References
2-PHENYL-2-(1-PIPERIDINYL)PROPANE
CAS:92321-29-4
Trade Name: 1-(1-Methyl-1-phenylethyl)piperidine; 1-(a,a-Dimethylbenzyl)piperidine;
Formula: C14H21N
DC8572
>98%
2-Phenyl-2-(1-piperidinyl)propane is an analog of phencyclidine that acts as a mechanism-based inactivator of human cytochrome P450 (CYP) 2B6 (Ki = 5.6 M; IC50 = 5.1 M).
2-PMPA(NAALADASEINHIBITOR)
CAS:173039-10-6
Formula: C6H11O7P
DC10014
>98%
2-PMPA is a potent and selective inhibitor of glutamate carboxypeptidase II (GCPII) with an IC50 of 300 pM.
2-PYRROLIDINECARBOXYLIC ACID
CAS:147-85-3
Formula: C5H9NO2
DCP-006
>98%,Standard References Grade
>98%,Standard References
2-UNDECANONE
CAS:112-12-9
Formula: C11H22O
DCJ-058
>98%,Standard References Grade
>98%,Standard References
2-O-GALLOYLHYPERIN
CAS:53209-27-1
Formula: C28H24O16
DCM-005
>98%,Standard References Grade
>98%,Standard References
20(R)-NOTOGINSENOSIDE R2
CAS:948046-15-9
Formula: C41H70O13
DCZ-102
>98%
>98%,Standard References
20(R)GINSENOSIDE RG3
CAS:38243-03-7
Formula: C42H72O13
DCR-037
>98%,Standard References Grade
>98%,Standard References
20(R)PROTOPANAXDIOL
Formula: C30H52O3
DCY-121
>98%,Standard References Grade
>98%,Standard References
20(S)-GINSENOSIDE CK
CAS:39262-14-1
Formula: C36H62O8
DCR-028
>98%,Standard References Grade
>98%,Standard References
20(S)-GINSENOSIDE RH2
CAS:67400-17-3
Formula: C36H62O8
DCR-036
>98%,Standard References Grade
>98%,Standard References
20-DEOXYINGENOL
CAS:54706-99-9
Trade Name: N/A
Formula: C20H28O4
DC9647
>98%
20-Deoxyingenol is a natural compound.
20-O-ACETYLINGENOL-3-ANGELATE
CAS:82425-35-2
Formula: C27H36O7
DC9655
>98%
20-O-Acetylingenol-3-angelate is a natural compound.
21-EPISERRATENEDIOL
CAS:1449-06-5
Formula: C30H50O2
DCB-054
>98%,Standard References Grade
>98%,Standard References
23-HYDROXY BUTULINIC ACID (23-HBA)
CAS:85999-40-2
Formula: C30H48O4
DC9802
>98%
23-hydroxy butulinic acid (23-HBA) is a potent angiogenesis inhibitor.
25-OCH3-PROTOPANAXTIOL
DCJ-047
>98%,Standard References Grade
>98%,Standard References
25-OH-PPD
Formula: C30H54O4
DCQ-082
>98%,Standard References Grade
>98%,Standard References
25-OH-VD2
CAS:21343-40-8
Trade Name: N/A
Formula: C28H44O2
DCAPI1508
>99%
25-Hydroxyvitamin D2 is used in serum to measure the concentration of vitamin D produced by the skin. It is known that 25-Hydroxyvitamin D2 can be detected in human serum using high-performance liquid chromatography and ultraviolet detection. Vitamin D2,
2A,5A-EPOXY-1,2-DIHYDROAKUAMMILAN-17-OIC ACID METHYL ESTER
CAS:4684-32-6
Formula: C20H22N2O3
DCY-081
>98%,Standard References Grade
>98%,Standard References
3',6-DISINAPOYLSUCROSE
CAS:139891-98-8
Formula: C34H42O19
DCZ-233
>98%
>98%,Standard References
3'-HYDROXY PUERARIN
CAS:117076-54-5
Formula: C21H20O10
DCQ-017
>98%,Standard References Grade
>98%,Standard References
3,'6-D ISINAPOYL SUCROSE
Formula: C36H46O17
DCF-013
>98%,Standard References Grade
>98%,Standard References
3,29-DIBENZOYL RAROUNITRIOL
CAS:873001-54-8
Formula: C44H58O5
DCE-025
>98%,Standard References Grade
>98%,Standard References
3,3'-DIINDOLYLMETHANE
CAS:1968-05-4
Formula: C17H14N2
DC9892
>98%
3,3'-Diindolylmethane(DIM) is a major digestive product of indole-3-carbinol, a potential anticancer component of cruciferous vegetables.
3,3-DI-O-METHYLELLAGIC ACID
CAS:2239-88-5
Formula: C16H10O8
DCE-030
>98%,Standard References Grade
>98%,Standard References
3,4,5-TRICAFFEOYLQUINIC ACID
CAS:86632-03-3
Formula: C34H30O15
DCS-122
>98%,Standard References Grade
>98%,Standard References
3,4,5-TRIMETHOXYCINNAMIC ACID
CAS:90-50-6
Formula: C12H14O5
DCZ-106
>98%
>98%,Standard References
3,4-DIHYDROXYBENZOIC ACID
CAS:99-50-3
Formula: C7H6O4
DCY-031
>98%,Standard References Grade
>98%,Standard References
3,4-DIHYDROXYPHENYLETHANOL
CAS:10597-60-1
Formula: C8H10O3
DCQ-079
>98%,Standard References Grade
>98%,Standard References
3,4-DIMETHOXYBENZOIC ACID
CAS:93-07-2
Formula: C9H10O4
DCL-062
>98%,Standard References Grade
>98%,Standard References
3,4-DIMETHOXYBENZYL ALCOHOL
CAS:93-03-8
Formula: C9H12O3
DCL-076
>98%,Standard References Grade
>98%,Standard References
3,5,6,7,8,3,4-HEPTEMTHOXYFLAVONE
Formula: C22H24O9
DCQ-083
>98%,Standard References Grade
>98%,Standard References
3,5,7-TRIHYDROXYFLAVONE
CAS:548-83-4
Formula: C15H10O5
DCG-013
>98%,Standard References Grade
>98%,Standard References
3,5-DIMETHOXY-4-HYDROXYBENZALDEHYDE
CAS:134-96-3
Formula: C9H10O4
DCD-044
>98%,Standard References Grade
>98%,Standard References
3-(4-PYRIDYL)
CAS:7272-84-6
Trade Name: Rho Kinase Inhibitor III; ROCK Inhibitor III; Rockout
Formula: C13H10N2
DC8567
>98%
3-(4-Pyridyl)indole is a ROCK-I inhibitor (IC50 = 25 M) that promotes cell spreading, inhibits membrane blebbing, and induces dissolution of actin stress fibers in a wound healing assay
3-CYANO-7-ETHOXYCOUMARIN
CAS:117620-77-6
Formula: C12H9NO3
DC9249
>98%
3-Cyano-7-ethoxycoumarin is a fluorescent P450 substrate (excitation/emission wavelengths = 408/455 nm); metabolized to cyano-hydroxycoumarin.
3-DEAZANEPLANOCIN A (DZNEP)
CAS:102052-95-9
Formula: C12H14N4O3
DC5190
>98%
3-deazaneplanocin A (DZNeP), an analog of adenosine, is a competitive inhibitor of S-adenosylhomocysteine hydrolase with Ki of 50 pM.
3-EPIWILSONINE
CAS:39024-15-2
Formula: C20H25NO4
DCB-058
>98%,Standard References Grade
>98%,Standard References
3-HYDROXY-4-METHOXYBENZOIC ACID
CAS:645-08-9
Formula: C8H8O4
DCZ-141
>98%
>98%,Standard References
3-HYDROXY-4-METHOXYCINNAMIC ACID
CAS:537-73-5
Formula: C10H10O4
DCY-044
>98%,Standard References Grade
>98%,Standard References
3-HYDROXY-4H-PYRAN-4-ONE
CAS:496-63-9
Formula: C5H4O3
DCJ-055
>98%,Standard References Grade
>98%,Standard References
3-INDOLEBUTYRIC ACID (IBA)
CAS:133-32-4
Trade Name: IBA
Formula: C12H13NO2
DCAPI1054
>99%
3-Indolebutyric acid (IBA)
3-ISOMANGOSTIN
CAS:19275-46-8
Formula: C24H26O6
DCY-180
>98%,Standard References Grade
>98%,Standard References
3-METHYLADENINE
CAS:5142-23-4
Trade Name: 3-MA
Formula: C6H7N5
DC7348
>98%
3-Methyladenine (3-MA) is a selective PI3K inhibitor for Vps34 and PI3K? with IC50 of 25 M and 60 M.
3-METHYLCYCLOPENTADECANONE
CAS:541-91-3
Formula: C16H30O
DCS-031
>98%,Standard References Grade
>98%,Standard References
3-N-BUTYLPHATHLIDE
CAS:6066-49-5
Formula: C12H14O2
DCZ-037
>98%,Standard References Grade
>98%,Standard References
3-O-ALPHA-L-ARABINOPYRANOSYLPOMOLIC ACID BETA-D-GLUCOPYRANOSYL ESTER
CAS:35286-58-9
Formula: C41H66O13
DCK-016
>98%,Standard References Grade
>98%,Standard References
3-O-CAFFEOYLQUINIC ACID
CAS:327-97-9
DCL-068
>98%,Standard References Grade
>98%,Standard References
3-O-GALLOYLMUCIC ACID
Formula: C13H14O12
DCM-065
>98%,Standard References Grade
>98%,Standard References
3-O-METHYLGALLIC ACID
CAS:3934-84-7
Formula: C8H8O5
DCJ-046
>98%,Standard References Grade
>98%,Standard References
3-TYP
CAS:120241-79-4
Trade Name: 3-TYP,3 TYP,3TYP
Formula: C7H6N4
DC10616
>98%
3-TYP is a selective SIRT3 inhibitor.
3- METHOXY PUERARIN
CAS:117047-07-1
Formula: C22H22O10
DCJ-017
>98%,Standard References Grade
>98%,Standard References
3-METHOXY APIIN;CHRYSOEIOL-7-(2-O-APIOSYLGLUCOSIDE)
DCJ-060
>98%,Standard References Grade
>98%,Standard References
3-METHOXY-5-HYDROXYISOFLAVONE-7-O-SS-D-GLUCOSIDE
DCJ-054
>98%,Standard References Grade
>98%,Standard References
3PO
CAS:18550-98-6
Trade Name: 3 PO,3-PO
Formula: C13H10N2O
DC10452
>98%
3PO is a PFKFB3 (6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase) inhibitor; reduces glycolytic flux and suppresses glucose uptake.
4 8C
CAS:14003-96-4
Formula: C11H8O4
DC10037
>98%
48C is a potent and selective IRE1 Rnase inhibitor with IC50 of 76 nM.
4'-DEMETHYLEPIPODOPHYLLOTOXIN
CAS:6559-91-7
Formula: C21H20O8
DCQ-004
>98%,Standard References Grade
>98%,Standard References
4'-O-METHYLPUERARIN
CAS:92117-94-7
Formula: C22H22O9
DCJ-049
>98%,Standard References Grade
>98%,Standard References
4-(4-HYDROXYPHENYL) -2-BUTANONE
CAS:5471-51-2
Formula: C10H12O2
DCF-022
>98%,Standard References Grade
>98%,Standard References
4-AMINO-4-METHYLPENTAN-2-ONEHYDROGENOXALATE
CAS:625-04-7
Formula: C6H13NO
DCS-077
>98%,Standard References Grade
>98%,Standard References
4-HYDROXY-3-METHOXYBENZYLALCOHOL(VANILLICALCOHOL)
CAS:498-00-0
Formula: C8H10O3
DCX-055
>98%,Standard References Grade
>98%,Standard References
4-HYDROXY-3-METHOXYCINNAMALDEHYDE
CAS:458-36-6
Formula: C10H10O3
DCZ-104
>98%
>98%,Standard References
4-HYDROXYCINNAMIC ACID
CAS:501-98-4
Formula: C9H8O3
DCD-032
>98%,Standard References Grade
>98%,Standard References
4-HYDROXYISOLEUCINE
CAS:55399-93-4
Formula: C6H13NO3
DCZ-279
>98%
>98%,Standard References
4-HYDROXYPHENETHYL ALCOHOL
CAS:501-94-0
Formula: C8H10O2
DCL-042
>98%,Standard References Grade
>98%,Standard References
4-ISOPROPYLTOLUENE
CAS:99-87-6
Formula: C10H14
DCD-037
>98%,Standard References Grade
>98%,Standard References
4-METHOXYPHENYLACETIC ACID
CAS:104-01-8
Formula: C9H10O3
DCZ-249
>98%
>98%,Standard References
4-METHOXYSALICYLIC ACID
CAS:2237-36-7
Formula: C8H8O4
DCJ-057
>98%,Standard References Grade
>98%,Standard References
4-METHYLUMBELLIFERONE
CAS:90-33-5
Formula: C10H8O3
DCQ-012
>98%,Standard References Grade
>98%,Standard References
4-NITROCATECHOL
CAS:3316-09-4
Formula: C6H5NO4
DC8951
>98%
4-OXO-4-HPR
CAS:865536-65-8
Trade Name: 4-oxo-4-fenretinide
Formula: C26H31NO3
DC9978
>98%
4-oxo-4-HPR is a recently identified fenretinide metabolite, induces marked G2-M cell cycle arrest and apoptosis in fenretinide-sensitive and fenretinide-resistant cell lines.
4-P-PDOT
CAS:620170-78-7
Formula: C19H21NO
DC10090
>98%
4-P-PDOT is a slelctive MT2 melatonin receptor antagonist 300 fold selective for MT2 (MEL-1B-R) vs MT1 (MEL-1A-R) melatonin receptor subtype.
4-SULFONAMIDE-PHENYLHYDRAZINE HYDROCHLORIDE
CAS:27918-19-0
Formula: C6H10ClN3O2S
DCH-028
>98%,Standard References Grade
>98%,Standard References
4E1RCAT
CAS:328998-25-0
Formula: C28H18N2O6
DC8245
>98%
4E1RCat is an inhibitor of protein translation that has been shown to prevent eIF4E:eIF4G and eIF4E:4E-BP1 interaction.
4E2RCAT
CAS:432499-63-3
Formula: C22H14ClNO4S2
DC10415
>98%
4E2RCat is an inhibitor of eIF4E-eIF4G interaction with an IC50 of 13.5 M.
4EGI-1
CAS:315706-13-9
Formula: C18H12Cl2N4O4S
DC7349
>98%
4EGI-1 is a competitive eIF4E/eIF4G interaction inhibitor by binding to eIF4E with KD of 25 M.
4SC-202
CAS:1186222-89-8
Trade Name: 4SC-202,4SC202,4SC 202
Formula: C30H29N5O6S2
DC7592
>98%
4SC-202 is an orally bioavailable benzamide and inhibitor of human class I histone deacetylases (HDACs) isoenzymes 1, 2 and 3, with potential antineoplastic activity. HDAC inhibitor 4SC-202 selectively binds to and inhibits class I HDACs leading to an acc
4SC-202 FREE BASE
CAS:910462-43-0
Trade Name: 4SC-202,4SC 202,4SC202
Formula: C23H21N5O3S
DC8423
>98%
4SC-202 is a selective class I HDAC inhibitor with IC50 of 1.20 M, 1.12 M, and 0.57 M for HDAC1, HDAC2, and HDAC3, respectively. Also displays inhibitory activity against Lysine specific demethylase 1 (LSD1). Phase 1.
5,15-DIACETYL-3-BENZOYLLATHYROL
CAS:218916-52-0
Formula: C31H38O7
DCQ-045
>98%,Standard References Grade
>98%,Standard References
5,5-DIMETHYLOXAZOLIDINE-2,4-DIONE
CAS:3166-62-9
Trade Name: 5,5-Dimethyloxazolidine-2,4-dione
Formula: C21H28NO3.Br
DC10262
>98%
Dimethadione is an anticonvulsant that is the active metabolite of trimethadione.
5,6-DIHYDRO-5-AZACYTIDINE
CAS:62488-57-7
Trade Name: DHAC; Dihydro-5-azacytidine; NSC 264-880; NSC 26480; NSC 265483
Formula: C8H14N4O5
DC9997
>98%
5,6-Dihydro-5-azacytidine|cas 62488-57-7
5,6-DIMETHOXY-2H-FURO[2,3-H]CHROMEN-2-ONE
CAS:131-12-4
Formula: C13H10O5
DCZ-245
>98%
>98%,Standard References
5,7-DIHYDROXYCHROMONE
CAS:31721-94-5
Formula: C9H6O4
DCE-032
>98%,Standard References Grade
>98%,Standard References
5-AMINOLEVULINIC ACID HCL
CAS:5451-09-2
Trade Name: Levulan, ALA
Formula: C5H9NO3.HCl
DCAPI1240
>99%
5-Aminolevulinic acid HCl
5-AZACYTIDINE
CAS:320-67-2
Trade Name: N/A
Formula: C8H12N4O5
DCAPI1525
>99%
5-Azacytidine is a potent growth inhibitor and a cytotoxic agent. 5-Azacytidine acts as a demethylating agent by inhibiting DNA methyltransferase (Dnmt), forming covalent adducts with cellular DNMT1 depleting enzyme activity. 5-Azacytidine also improves t
5-CHLORO-8-HYDROXY-7-IODOQUINOLINE
CAS:130-26-7
Trade Name: 5-Chloro-8-hydroxy-7-iodoquinoline
Formula: C9H5ClINO
DC10242
>98%
Clioquinol is an orally bioavailable, lipophilic, copper-binding, halogenated 8-hydroxyquinoline with antifungal, antiparasitic and potential antitumor activities.
5-ETHOXYCHELERTHRINE
CAS:79559-55-0
Formula: C23H23NO5
DCY-154
>98%,Standard References Grade
>98%,Standard References
5-FAM SE
CAS:92557-80-7
Formula: C25H15NO9
DC9371
>98%
5-FAM SE is a single isomer, it is one of the most popular green fluorescent reagents used for labeling peptides, proteins and nucleotides.
5-FLUOROURACIL
CAS:51-21-8
Formula: C4H3FN2O2
DC8944
>98%
5-Fluorouracil is a potent antitumor agent that affects pyrimidine synthesis by inhibiting thymidylate synthetase thus depleting intracellular dTTP pools.
5-HYDROXY-1,4-NAPHTHALENEDIONE
CAS:481-39-0
Formula: C10H6O3
DCZ-244
>98%
>98%,Standard References
5-HYDROXY-1-TETRALONE
CAS:28315-93-7
Formula: C10H10O2
DCZ-276
>98%
>98%,Standard References
5-HYDROXY-6,7-DIMETHOXYLFLAVONE
CAS:740-33-0
Formula: C17H14O5
DCQ-071
>98%,Standard References Grade
>98%,Standard References
5-HYDROXY-7,8-DIMETHOXYFLAVONE
CAS:3570-62-5
Formula: C17H14O5
DCQ-070
>98%,Standard References Grade
>98%,Standard References
5-HYDROXYMETHYLFURFURAL
CAS:67-47-0
Formula: C6H6O3
DCQ-042
>98%,Standard References Grade
>98%,Standard References
5-HYDROXYTRYPTOPHAN
CAS:56-69-9
Formula: C11H12N2O3
DCQ-032
>98%,Standard References Grade
>98%,Standard References
5-IODOTUBERCIDIN
CAS:24386-93-4
Trade Name: 5-Iodo-7--D-ribofuranosyl-7H-pyrrolo[2,3-d]pyrimidin-4- amine
Formula: C11H13IN4O4
DC5179
>98%
5-Iodotubercidin (Itu) has been shown to inhibit mitogen-activated protein kinase (ERK2) (Ki = 525 nM), adenosine kinase (ADK) (Ki = 30 nM), casein kinases 1 & 2 (CSNK1A1 & CSNK2A1), protein kinase A (PKA) and insulin receptor kinase (IC50 ranging from 0.
5-ISOPROPYL-2-METHYLPHENOL
CAS:499-75-2
Formula: C10H14O
DCX-048
>98%,Standard References Grade
>98%,Standard References
5-METHYL FURFURAL
CAS:620-02-0
Formula: C6H6O2
DCJ-044
>98%,Standard References Grade
>98%,Standard References
5-METHYL-7-METHOXYISOFLAVONE
CAS:82517-12-2
Formula: C17H14O3
DCJ-045
>98%,Standard References Grade
>98%,Standard References
5-O-METHYLVISAMMIOSIDE
CAS:84272-85-5
Formula: C22H28O10
DCJ-002
>98%,Standard References Grade
>98%,Standard References
5-R-RIVAROXABAN
CAS:865479-71-6
Trade Name: Xarelto; BAY 59-7939
Formula: C19H18ClN3O5S
DC9444
>98%
5-R-Rivaroxaban is (R) enantiomer of Rivaroxaban.
5-TAMRA
CAS:91809-66-4
Trade Name: 5-Carboxytetramethylrhodamine
Formula: C25H22N2O5
DC9373
>98%
The amine-reactive 5-TAMRA, SE and its conjugates yield bright, pH-insensitive orange-red fluorescence (approximate excitation/emission maxima ~546/579) with good photostability.
5IA (A5IA)
CAS:215874-86-5
Trade Name: ?5ia
Formula: C17H14N8O2
DC7642
>98%
a5IA is a selective inverse agonist for ?5 subtype of GABAA receptor with a higher intrinsic activity at the A5 subtype than other drugs.
6-FAM
CAS:3301-79-9
Trade Name: 6-Carboxyfluorescein
Formula: C21H12O7
DC9377
>98%
The single isomer, 6-FAM, contains a carboxylic acid that can be used to react with primary amines via carbodiimide activation of the carboxylic acid.
6-FAM SE
CAS:92557-81-8
Formula: C25H15NO9
DC9372
>98%
6-FAM SE is another isomer of carboxyfluorescein.
6-FITC
CAS:3326-31-6
Trade Name: 6-Fluorescein Isothiocyanate
Formula: C21H11NO5S
DC9376
>98%
6-Fluorescein isothiocyanate(6-FITC) is a derivative of fluorescein used in wide-ranging applications including flow cytometry.
6-GINGEROL
CAS:23513-14-6
Formula: C17H26O4
DCJ-019
>98%,Standard References Grade
>98%,Standard References
6-HYDROXYINDOLE
CAS:2380-86-1
Formula: C8H7NO
DCY-168
>98%,Standard References Grade
>98%,Standard References
6-HYDROXYPURINE
CAS:68-94-0
Formula: C5H4N4O
DCC-069
>98%,Standard References Grade
>98%,Standard References
6-MERCAPTOPURINE (6-MP) MONOHYDRATE
CAS:6112-76-1
Formula: C5H6N4OS
DC8864
>98%
6-Mercaptopurine Monohydrate is a widely used antileukemic agent and immunosuppressive drug that inhibits de novo purine synthesis through incorporation of thiopurine methyltransferase metabolites into DNA and RNA.
6-O-CAFFEOYLERIGEROSIDE
Formula: C20H20O11
DCD-075
>98%,Standard References Grade
>98%,Standard References
6-SHOGAOL
CAS:555-66-8
Formula: C17H24O3
DCJ-038
>98%,Standard References Grade
>98%,Standard References
6-TAMRA
CAS:91809-67-5
Trade Name: 6-Carboxytetramethylrhodamine
Formula: C25H22N2O5
DC9374
>98%
Tetramethylrhodamine (TMR, TRITC) has been a widely used fluorophore for preparing bioconjugates, especially fluorescent antibody and avidin derivatives used in immunochemistry.
6-TG/THIOGUANINE
CAS:154-42-7
Formula: C5H5N5S
DC8953
>98%
6-Thioguanine(6-TG) belongs to the thiopurine family of drugs that also include mercaptopurine and azathioprine, which are examples of antimetabolites; it is a purine analogue of the nucleobase guanine.
6-THIO-DG
CAS:789-61-7
Formula: C10H13N5O3S
DC8861
>98%
6-thio-dG is a nucleoside analog and telomerase substrate.
666-15
CAS:1433286-70-4
Formula: C33H31Cl2N3O5
DC10187
>98%
666-15 is a potent and selective CREB inhibitor with an IC50 of 81 nM.
6H05
CAS:1469338-01-9
Formula: C20H30ClN3O2S3.CF3COOH
DC7736
>98%
6H05 is a selective, and allosteric inhibitor of oncogenic K-Ras(G12C).
7,8-BENZOFLAVONE
CAS:604-59-1
Formula: C19H12O2
DCZ-162
>98%
>98%,Standard References
7,8-DIHYDROXYCOUMARIN
CAS:486-35-1
Formula: C9H6O4
DCR-007
>98%,Standard References Grade
>98%,Standard References
7,8-DIHYDROXYFLAVONE
CAS:38183-03-8
Trade Name: 7,8-Dihydroxyflavone
Formula: C15H10O4
DC10215
>98%
7,8-Dihydroxyflavone acts as a potent and selective small-molecule agonist of the TrkB receptor (Kd 320 nM), the main signaling receptor of brain-derived neurotrophic factor (BDNF).
7-AMINO-4-METHYLCOUMARIN
CAS:26093-31-2
Formula: C10H9NO2
DCA-020
>98%,Standard References Grade
>98%,Standard References
7-AMINOCEPHALOSPORANIC ACID
CAS:957-68-6
Trade Name: 7-ACA
Formula: C10H12N2O5S
DCAPI1394
>99%
7-Aminocephalosporanic acid is used for synthesis of cephalosporin antibiotics and intermediates.
7-EPITAXOL
CAS:105454-04-4
Formula: C47H51NO14
DCB-077
>98%,Standard References Grade
>98%,Standard References
7-ETHYL-10-HYDROXY-CAMPTOTHECIN
CAS:119577-28-5
Formula: C22H20N2O5
DCS-016
>98%,Standard References Grade
>98%,Standard References
7-ETHYLCAMPTOTHECIN
CAS:78287-27-1
Formula: C22H20N2O4
DCZ-143
>98%
>98%,Standard References
7-HYDROXY ARISTOLOCHIC ACID A
CAS:79185-75-4
Formula: C17H11NO8
DCQ-050
>98%,Standard References Grade
>98%,Standard References
7-HYDROXY-5,8-DIMETHOXYFLAVANONE
CAS:54377-24-1
DCQ-057
>98%,Standard References Grade
>98%,Standard References
7-HYDROXYCOUMARIN
CAS:93-35-6
Formula: C9H6O3
DCS-025
>98%,Standard References Grade
>98%,Standard References
7-METHOXYCOUMARIN
CAS:531-59-9
Formula: C10H8O3
DCJ-070
>98%,Standard References Grade
>98%,Standard References
7-O-METHYLCHRYSIN
Formula: C16H12O4
DCJ-052
>98%,Standard References Grade
>98%,Standard References
7-TACA
CAS:37539-03-0
Formula: C10H11N5O3S2
DC8874
>98%
Impurity D of Cefoperazone
7ACC2
CAS:1472624-85-3
Trade Name: 7ACC 2; 7ACC-2, 7ACC 2; 7ACC-2
Formula: C18H15NO4
DC7876
>98%
7ACC2 is a new potent MCT inhibitor with IC50 of 11 nM for inhibition of [14C]-lactate influx; new antitumor treatment targeting lactate transport in cancer cells.
7BETA-HYDROXYLATHYROL
CAS:34208-98-5
Formula: C20H30O5
DCAP003
>98%,Standard References Grade
>98%,Standard References
8-BROMO-CAMP
CAS:76939-46-3
Formula: C10H10BrN5NaO6P
DC8388
>98%
8-Bromo-cAMP is a cell perbeable cyclic AMP (cAMP) analog and a PKA activator.
8-DEACETYLYUNACONITINE
Formula: C33H47O10
DCQ-089
>98%,Standard References Grade
>98%,Standard References
8-GERANOPSORALEN
CAS:7437-55-0
Formula: C21H22O4
DCZ-286
>98%
purity >98%,Standard References
8-GINGEROL
CAS:30462-35-2
Formula: C43H32O20
DCJ-020
>98%,Standard References Grade
>98%,Standard References
8-METHOXYPSORALEN
CAS:298-81-7
Formula: C12H8O4
DCH-035
>98%,Standard References Grade
>98%,Standard References
8-O-ACETYL SHANZHISIDE METHYL ESTER
CAS:57420-46-9
Formula: C19H28O12
DC10186
>98%
8-O-Acetyl shanzhiside methyl ester (ND01) is an iridoid glucoside isolated from the leaves of Lamiophlomis rotata Kudo, a Chinese folk medicinal plant in Xi-zang.
8-O-ACETYLHARPAGIDE
CAS:6926-14-3
Formula: C17H26O11
DCY-112
>98%,Standard References Grade
>98%,Standard References
8-OH-DPAT
CAS:78950-78-4
Formula: C16H25NO
DC10537
>98%
8-OH-DPAT is a research chemical of the aminotetralin chemical class and has been widely used to study the function of the 5-HT1A receptor.
8DM
CAS:24916-90-3
Formula: C22H28O5
DC9097
>98%
9-AMINO-MINOCYCLINE HCL
CAS:149934-21-4
Formula: C23H28N4O7.ClH
DC9165
>98%
9-AMINOCAMPTOTHECIN
CAS:91421-43-1
Formula: C20H17N3O4
DCA-019
>98%,Standard References Grade
>98%,Standard References
9-DIHYDRO-13-ACETYLBACCATIN III
CAS:142203-65-4
Trade Name: 9-DHAB III; 13-Acetyl-9-dihydrobaccatin III
Formula: C33H42O12
DC9557
>98%
9-Dihydro-13-acetylbaccatin III (9-DHAB III) is an intermediate for taxol analog preparations.
9-METHOXYCAMPTOTHECIN
CAS:39026-92-1(19685-10-0)
Formula: C21H18N2O5
DCZ-250
>98%
>98%,Standard References
9-METHYLADENINE
CAS:700-00-5
Trade Name: N9-Methyladenine, 9-METHYL-9H-PURIN-6-AMINE, 9-Methyl-9H-adenine, 6-Amino-9-methylpurine, 700-00-5,
Formula: C6H7N5
DC7350
>98%
9-NITROCAMPTOTHECIN
CAS:86639-62-5
Formula: C20H15N3O6
DCX-058
>98%,Standard References Grade
>98%,Standard References
A 419259 (TRIHYDROCHLORIDE)
CAS:1435934-25-0
Trade Name: A419259 trihydrochloride;A-419259 trihydrochloride;RK 20449 trihydrochloride;RK20449 trihydrochlorid
Formula: C29H37Cl3N6O
DC9628
>98%
A 419259 3Hcl is an apoptosis inducing agent that inhibits Src family kinases (c-Src).
A 804598
CAS:1125758-85-1
Trade Name: A 804598; A804598
Formula: C19H12N6
DC9954
>98%
A-804598 is a novel, competitive, and selective P2X7 receptor antagonist with IC50 of 10 nM, 9 nM and 11 nM in rat, mouse and human P2X7 receptors respectively.
A 922500
CAS:959122-11-3
Trade Name: DGAT-1 Inhibitor 4a; A-922500; A922500
Formula: C26H24N2O4
DC7038
>98%
A 922500 is a potent, selective, and orally bioavailable DGAT-1 inhibitor with IC50 values of 7 nM and 24 nM for human and mouse DGAT-1 respectively.
A-1210477
CAS:1668553-26-1
Trade Name: A-1210477,A 1210477,A1210477
Formula: C46H55N7O7S
DC8475
>98%
A-1210477 is a potent and selective MCL-1 inhibitor.
A-1331852
CAS:1430844-80-6
Trade Name: A 1331852,A1331852
Formula: C38H38N6O3S
DC9296
>98%
A-1331852 is a high affinity BH3 mimetic Ligand of BCL protein BCL-XL.
A-196
CAS:N/A
Trade Name: A-196,A 196,A196
Formula: C18H16Cl2N4
DC10509
>98%
A-196 is a potent and selective chemical inhibitor of SUV420H1 and SUV420H2 that inhibits the di- and trimethylation of H4K20me in multiple cell lines.
A-205804
CAS:251992-66-2
Trade Name: A205804,A 205804,A-205804
Formula: C15H12N2OS2
DC7044
>98%
A-205804 is a potent and selective inhibitor of E-selectin and ICAM-1 expression with IC50 of 20 nM and 25 nM respectively.
A-317491
CAS:475205-49-3
Formula: C33H27NO8
DC10643
>98%
A-317491 is a novel potent and selective non-nucleotide antagonist of P2X3 and P2X2/3 receptors with Ki values of 22 nM and 9 nM for human P2X3 and P2X2/3 receptors.
A-317491 (SODIUM SALT HYDRATE)
Trade Name: A 317491;A317491;(S)-5-((3-phenoxybenzyl)(1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl)benzene-1,2,4-
Formula: C33H29NNaO9+
DC9574
>98%
A-317491 is a non-nucleotide P2X3 and P2X2/3 receptor antagonist, which inhibits calcium flux mediated by the receptors._x000D_
A-366
CAS:1527503-11-2
Trade Name: A-366, A366,A 366
Formula: C19H27N3O2
DC7855
>98%
A-366 is a potent and selective G9a/GLP histone lysine methyltransferase inhibitor (IC50 = 3.3 nM).
A-438079 HCL
CAS:899431-18-6
Trade Name: A-438079,A438079,A 438079
Formula: C13H10Cl3N5
DC8406
>98%
A-438079 HCl is a potent, and selective P2X7 receptor antagonist with pIC50 of 6.9.
A-674563
CAS:552325-73-2
Trade Name: A-674563; A 674563; A674563
Formula: C22H22N4O
DC5163
>98%
A-674563 is a potent, orally available Akt1 inhibitor with an IC50 value of 11nM. Also displays activity against PKA and CDK2 with IC50 values of 16nM and 46nM respectively.
A-740003
CAS:861393-28-4
Trade Name: A 740003; A740003
Formula: C26H30N6O3
DC7351
>98%
A-740003 is potent, selective and competitive P2X7 receptor antagonist (IC50 values are 18 and 40 nM for rat and human receptors respectively).
A-769662
CAS:844499-71-4
Trade Name: A 769662; A769662
Formula: C20H12N2O3S
DC7045
>98%
A-769662 is a potent, reversible AMPK activator with EC50 of 0.8 M, little effect on GPPase/FBPase activity.
A-790742
CAS:854755-48-9
Trade Name: CHEMBL470508, A-790742,A790742,A 790742
Formula: C49H65N7O7
DC7785
>98%
A-790742 is a potent human immunodeficiency virus type 1 (HIV-1) protease inhibitor, with 50% effective concentrations ranging from 2 to 7 nM against wild-type HIV-1.
A-803467
CAS:944261-79-4
Trade Name: A803467
Formula: C19H16ClNO4
DC2061
>98%
A-803467 is a selective NaV1.8 channel blocker with IC50 of 8 nM.
A-867744
CAS:1000279-69-5
Trade Name: A 867744;A867744
Formula: C20H19ClN2O3S
DC9516
>98%
A-867744 is a positive allosteric modulator of a7 nAChRs (IC50 values are 0.98 and 1.12 M for human and rat a7 receptor ACh-evoked currents respectively, in X.
A-966492
CAS:934162-61-5
Trade Name: A966492,A 966492,A-966492
Formula: C18H17FN4O
DC7046
>98%
A-966492 is a novel and potent inhibitor of PARP1 and PARP2 with Ki of 1 nM and 1.5 nM, respectively.
A-AMYLOID PRECURSOR PROTEIN MODULATOR
CAS:497259-23-1
Trade Name: (2S,5S)-(E,E)-8-(5-(4-(Trifluoromethyl)phenyl)-2,4-pentadienoylamino)benzolactam; PKC Activator V
Formula: C27H30F3N3O3
DC8534
>98%
a-Amyloid Precursor Protein Modulator is a cell-permeable benzolactam derived PKC activator (Ki = 11.9 nM for PKCa) that efficiently enhances non-amyloidogenic a-processing of amyloid precursor protein (APP) even at 100 nM in human fibroblast AG06848.
A-AMYRENONE
CAS:20248-08-2
Formula: C30H48O
DCX-041
>98%,Standard References Grade
>98%,Standard References
A-ASARONE
CAS:2883-98-9
Formula: C12H16O3
DCX-063
>98%,Standard References Grade
>98%,Standard References
A-CHCA
CAS:28166-41-8
Formula: C10H7NO3
DC10644
>98%
4-Chloro-a-cyanocinnamic acid (a-CHCA) is a classic monocarboxylate transporters (MCT) inhibitor. a-cyano-4-hydroxycinnamate (CHC) has a 10-fold selectivity for MCT1 compared to other MCTs.
A-CYPERONE
CAS:473-08-5
Formula: C15H22O
DCX-038
>98%,Standard References Grade
>98%,Standard References
A-HEDERIN
CAS:35790-95-5
Formula: C41H66O12
DCC-030
>98%,Standard References Grade
>98%,Standard References
A-LINOLEIC ACID
CAS:60-33-3
Formula: C18H32O2
DCY-096
>98%,Standard References Grade
>98%,Standard References
A-MANGOSTIN
CAS:6147-11-1
Formula: C24H26O6
DCD-034
>98%,Standard References Grade
>98%,Standard References
A-PINENE
CAS:2437-95-8
Formula: C10H16
DCP-011
>98%,Standard References Grade
>98%,Standard References
A-SPINASTEROL
CAS:481-18-5
Formula: C29H48O
DCB-055
>98%,Standard References Grade
>98%,Standard References
A-SPINASTERYL-3-O-SS-D-GLUCOSIDE
DCB-066
>98%,Standard References Grade
>98%,Standard References
A-TERPINEOL
CAS:10482-56-1
Formula: C10H18O
DCS-110
>98%,Standard References Grade
>98%,Standard References
A-TERTHIOPHENE
CAS:1081-34-1
Formula: C12H8S3
DCS-075
>98%,Standard References Grade
>98%,Standard References
A1155463
CAS:1235034-55-5
Trade Name: A-1155463; A 1155463; A1155463.
Formula: C35H32FN5O4S2
DC9768
>98%
A-1155463 is a highly potent and selective BCL-XL inhibitor.
A395
CAS:N/A
Trade Name: A-395,A 395
Formula: C26H33N4SO2F
DC10129
>98%
A-395 potently inhibited the formation of H3K27me3 (via antagonizing EED in the trimeric PRC2 complex (EZH2:EED:SUZ12)) with IC50 = 34 2 nM (Hill Slope = 0.7)
A66
CAS:1166227-08-2
Formula: C17H23N5O2S2
DC7538
>98%
A66 is a potent and specific p110a inhibitor with IC50 of 32 nM, >100 fold selectivity for p110a over other class-I PI3K isoforms.
A77-01
CAS:607737-87-1
Trade Name: A7701,A 7701, A-7701
Formula: C18H14N4
DC8020
>98%
A 77-01 is a potent inhibitor of TGF- type I receptor superfamily activin-like kinase ALK5 with IC50 of 25 nM.
A83-01
CAS:909910-43-6
Trade Name: A83-01; A-83-01,A8301,A-8301,A 8301
Formula: C25H19N5S
DC7286
>98%
A83-01 is a selective inhibitor of TGF- type I receptor ALK5 kinase, type I activin/nodal receptor ALK4 and type I nodal receptor ALK7 (IC50 values are 12, 45 and 7.5 nM respectively).
A967079
CAS:1170613-55-4
Formula: C12H14FNO
DC9222
>98%
AA26-9
CAS:1312782-34-5
Formula: C7H10N4O
DC10165
>98%
AA26-9 is a potent and broad spectrum serine hydrolase inhibitor.
AB-MECA
CAS:152918-26-8
Formula: C18H21N7O4
DC8667
>98%
AB-MECA is a high affinity A3 adenosine receptor agonist, has high affinity for recombinant A1 and A3 receptors.
ABACAVIR
CAS:136470-78-5
Formula: C14H18N6O
DC9029
>98%
Abacavir is a powerful nucleoside analog reverse transcriptase inhibitor (NRTI) used to treat HIV and AIDS.
ABC294640
CAS:915385-81-8
Trade Name: ABC294640; ABC-294640; ABC 294640; 3-(4-chlorophenyl)-adamantane-1-carboxylic acid (pyridin-4-ylmeth
Formula: C23H25ClN2O
DC5027
>98%
ABC294640 is an orally available, aryladamantane compound and selective inhibitor of sphingosine kinase-2 (SK2) with potential antineoplastic activity.
ABIRATERONE (CB-7598)
CAS:154229-19-3,154229-18-2
Trade Name: CB7598
Formula: C24H31NO
DC2710
99%
Abiraterone (CB-7598) is a potent CYP17 inhibitor with IC50 of 2 nM.
ABR-215062 (LAQUINIMOD)
CAS:248281-84-7
Trade Name: ABR215062, ABR 215062 (Laquinimod)
Formula: C19H17ClN2O3
DC2071
99%
Laquinimod (ABR-215062) is a potent immunomodulator.
ABSCISIC ACID
CAS:14375-45-2
Formula: C15H20O4
DCZ-114
>98%
>98%,Standard References
ABSINTHIN
CAS:1362-42-1
Formula: C30H40O6
DCY-110
>98%,Standard References Grade
>98%,Standard References
ABT-263(NAVITOCLAX)
CAS:923564-51-6
Trade Name: ABT263,ABT-263
Formula: C47H55ClF3N5O6S3
DC4127
99%
ABT-263 (Navitoclax) is a potent inhibitor of Bcl-xL, Bcl-2 and Bcl-w with Ki of = 0.5 nM, =1 nM and = 1 nM, respectively.
ABT-333
CAS:1132935-63-7
Trade Name: ABT333; ABT 333
Formula: C26H27N3O5S
DC7352
>98%
ABT-333 is an NS5B non-nucleoside polymerase inhibitor.
ABT-639
CAS:1235560-28-7
Trade Name: ABT639,ABT 639
Formula: C20H20ClF2N3O3S
DC9706
>98%
ABT-639 is a novel, peripherally acting, selective T-type Ca2+ channel blocker. ABT-639 blocks recombinant human T-type (Cav3.2) Ca2+ channels in a voltage-dependent fashion (IC50 = 2 M) and attenuates LVA currents in rat DRG neurons (IC50 = 8 M).
ABT-719
CAS:162829-90-5
Trade Name: ABT-719,ABT 719,ABT719,A-86719.1
Formula: C18H20FN3O3
DC9262
>98%
ABT-719 is a potent bacterial DNA gyrase inhibitor.
ABT-719 HCL
CAS:162763-53-3
Trade Name: ABT-719,ABT 719,ABT719,A-86719.1
Formula: C18H20FN3O3.HCl
DC9261
>98%
ABT-719 is a potent bacterial DNA gyrase inhibitor.
ABT-737
CAS:852808-04-9
Trade Name: ABT-737,ABT737,ABT 737
Formula: C42H45ClN6O5S2
DC1022
99%
ABT-737 is a BH3 mimetic inhibitor of Bcl-xL, Bcl-2 and Bcl-w with EC50 of 78.7 nM, 30.3 nM and 197.8 nM, respectively.
ABT-751(E 7010)
CAS:141430-65-1
Trade Name: ABT751; ABT 751; E7010; E-7010; E 7010
Formula: C18H17N3O4S
DC7353
>98%
ABT-751(E 7010) is a novel bioavailable tubulin-binding and antimitotic sulfonamide agent with IC50 of about 1.5 and 3.4 M in neuroblastoma and non-neuroblastoma cell lines, respectively.
ABT888 (FREE BASE)
CAS:912444-00-9
Formula: C13H16N4O
DC8899
>98%
Veliparib (ABT-888) is a potent inhibitor of PARP1 and PARP2 with Ki of 5.2 nM and 2.9 nM, respectively.
AC 55541
CAS:916170-19-9
Trade Name: AC55541, AC-55541
Formula: C25H20BrN5O3
DC7698
>98%
AC 55541 is a potent and selective protease-activated receptor 2 (PAR2) agonist (pEC50 = 6.7) that displays no activity at other PAR subtypes or at over 30 other receptors involved in nociception and inflammation.
AC260584
CAS:560083-42-3
Trade Name: AC-260584; AC 260584
Formula: C20H29FN2O2
DC10293
>98%
AC260584 is an M1 muscarinic receptor allosteric agonist with a pEC50 of 7.6.
AC264613
CAS:1051487-82-1
Trade Name: AC 264613,AC-264613
Formula: C19H18BrN3O2
DC10117
>98%
AC264613 is a potent and selective protease-activated receptor 2 (PAR2) agonist (pEC50 = 7.5). Displays no activity at other PAR subtypes and exhibits no significant activity at over 30 other receptors implicated in nociception and inflammation.
AC710
CAS:1351522-04-7
Trade Name: AC710; AC 710; AC-710
Formula: C31H42N6O4
DC7700
>98%
AC710, is a potent Globally Selective Inhibitor of Platelet-Derived Growth Factor Receptor-Family Kinases.
ACACETIN
CAS:480-44-4
Formula: C16H12O5
DC9917
>98%
Acacetin is an O-methylated flavone found in Robinia pseudoacacia (black locust), Turnera diffusa (damiana),Betula pendula (silver birch),and in the fern Asplenium normale.
ACALABRUTINIB(ACP196)
CAS:1420477-60-6
Trade Name: ACP-196; ACP196; ACP 196
Formula: C26H23N7O2
DC9660
>98%
Acalabrutinib (ACP-196) is a second-generation, selective, irreversible inhibitor of BTK.
ACALISIB
CAS:870281-34-8
Trade Name: UNII-OVW60IDW1D;Acalisib (GS-9820);
Formula: C21H16FN7O
DC8760
>98%
Acalisib (GS-9820) is a potent and selective inhibitor of PI3Kd with IC50 value of 12.7 nM.
ACARBOSE
CAS:56180-94-0
Formula: C25H43NO18
DCA-014
>98%,Standard References Grade
>98%,Standard References
ACEBILUSTAT(ZK322)
CAS:943764-99-6
Trade Name: ZK 322,ZK-322
Formula: C29H27N3O4
DC9986
>98%
Acebilustat(ZK322) is a potent and selective leukotriene A4 hydrolase inhibitor.
ACEGASTRODINE
CAS:64291-41-4
Formula: C21H26O11
DCY-178
>98%,Standard References Grade
>98%,Standard References
ACELARIN
CAS:840506-29-8
Trade Name: NUC-1031; NUC1031; NUC 1031
Formula: C25H27F2N4O8P
DC10318
>98%
Acelarin (NUC-1031) is a ProTide transformation and enhancement of the widely-used nucleoside analogue, gemcitabine.
ACEMETACIN
CAS:53164-05-9
Formula: C21H18ClNO6
DC9127
>98%
Acemetacin is a non-steroidal anti-inflammatory drug and a glycolic acid ester of indometacin that is a cyclooxygenase inhibitor.
ACESULFAME POTASSIUM
CAS:55589-62-3,124030-40-6,133249-02-2,33665-90-6(free
Trade Name: N/A
Formula: C4H5NO4S.K
DCAPI1249
>99%
ACETAMINOPHEN
CAS:103-90-2
Formula: C8H9NO2
DC9900
>98%
Acetaminophen is a COX inhibitor for COX-1 and COX-2 with IC50 of 113.7 M and 25.8 M, respectively.
ACETANILIDE (ANTIFEBRIN)
CAS:103-84-4
Trade Name: N-phenylacetamide, Acetanil, Acetamidobenzene, Acetylaniline, NSC 7636
Formula: C8H9NO
DCAPI1009
>99%
Acetanilide (Antifebrin)
ACETAZOLAMIDE
CAS:59-66-5
Formula: C4H6N4O3S2
DC8978
>98%
Acetazolamide is a potent carbonic anhydrase (CA) inhibitor; best-studied agent for the amelioration of acute mountain sickness (AMS).
ACETIC ACID OCTYL ESTER
CAS:112-14-1
Formula: C10H20O2
DCZ-149
>98%
>98%,Standard References
ACETOHYDROXAMIC ACID
CAS:546-88-3
Trade Name: Acetohydroxamic acid
Formula: C2H5NO2
DC10248
>98%
Acetohydroxamic acid is an Urease Inhibitor. In the urine, it acts as an antagonist of the bacterial enzyme urease.
ACETYL-11-KETO--BOSWELLIC ACID
CAS:67416-61-9
Formula: C32H48O5
DCT-034
>98%,Standard References Grade
>98%,Standard References
ACETYL-TRANS-RESVERATROL
CAS:42206-94-0
Formula: C20H18O6
DCY-176
>98%,Standard References Grade
>98%,Standard References
ACETYLACONITINE
CAS:77181-26-1
Formula: C36H49NO12
DCY-025
>98%,Standard References Grade
>98%,Standard References
ACETYLCHOLINE IODIDE
CAS:2260-50-6
Formula: C7H16NO2.I
DC9894
>98%
Acetylcholine iodide is a neurotransmitter found at neuromuscular junctions, autonomic ganglia, parasympathetic effector junctions, a subset of sympathetic effector junctions, and at many sites in the central nervous system.
ACETYLCORYNOLINE
CAS:18797-80-3
Formula: C23H23NO6
DCY-077
>98%,Standard References Grade
>98%,Standard References
ACETYLDIHYDROMICROMELIN A
CAS:94285-22-0
DCY-103
>98%,Standard References Grade
>98%,Standard References
ACETYLSALICYLIC ACID
CAS:50-78-2
Formula: C9H8O4
DC8956
>98%
ACETYLSPIRAMYCIN (ASPM)
CAS:24916-51-6
Formula: C45H76N2O15
DC10637
>98%
Acetylspiramycin (ASPM) is a macrolide antimicrobial agent.
ACETYTASTRAGALOSIDE
DCY-129
>98%,Standard References Grade
>98%,Standard References
ACEVALTRATE
CAS:25161-41-5
Formula: C24H32O10
DCC-048
>98%,Standard References Grade
>98%,Standard References
ACEVALTRATUM
DCY-113
>98%,Standard References Grade
>98%,Standard References
ACIPIMOX
CAS:51037-30-0,76958-97-9(sodiumsalt)
Trade Name: K-9321, Olbemox, Olbetam
Formula: C6H6N2O3
DCAPI1205
>99%
Acipimox
ACITAZANOLAST (WP-871,ZEPELIN)
CAS:114607-46-4
Trade Name: Acitazanolast, WP871, Zepelin,WP 871
Formula: C9H7N5O3
DC1092
>98%
Acitazanolast is an active metabolite of tazanolast and anti-allergic drug.
ACITRETIN
CAS:55079-83-9,925701-88-8(sodiumsalt)
Trade Name: Soriatane
Formula: C21H26O3
DCAPI1244
>99%
Acitretin
ACIVICIN
CAS:42228-92-2
Trade Name: NSC 163501,Antibiotic AT-125,U 42126
Formula: C5H7ClN2O3
DC8818
>98%
Acivicin is a glutamine analog that irreversibly inhibits glutamine-dependent amidotransferases involved in nucleotide and amino acid biosynthesis (Kis = 10 and 560 M for anthranilate synthase and glutamate synthase, respectively).
ACLIDINIUM BROMIDE
CAS:320345-99-1
Formula: C26H30BrNO4S2
DC8941
>98%
Aclidinium Bromide(LAS 34273; LAS-W 330) is a long-acting, inhaled muscarinic antagonist as a maintenance treatment for chronic obstructive pulmonary disease (COPD).
ACOLBIFENE
CAS:182167-02-8
Trade Name: EM 652; EM-652; EM652; SCH57068; SCH-57068; SCH 57068.
Formula: C29H31NO4
DC7354
>98%
acolbifene, also known as EM-652, or SCH-57068, is a selective estrogen receptor modulator (SERM). Acolbifene is currently being studied in the prevention of breast cancer in women at high risk of breast cancer. EM-652 (SCH 57068) and the prodrug EM-800 (
ACONINE
CAS:509-20-6
Formula: C25H41NO9
DCW-015
>98%,Standard References Grade
>98%,Standard References
ACONITINE
CAS:302-27-2
Formula: C34H47NO11
DCW-006
>98%,Standard References Grade
>98%,Standard References
ACOTIAMIDE
CAS:185106-16-5
Formula: C21H30N4O5S
DC8798
>98%
Acotiamide acts as an acetylcholinesterase inhibitor
ACOTIAMIDE HCL
CAS:773092-05-0
Trade Name: Ym-443,Acotiamide HCl
Formula: C21H31ClN4O5S
DC8285
>98%
ACRIVASTINE
CAS:87848-99-5
Trade Name: BW825C
Formula: C22H24N2O2
DC10279
>98%
Acrivastine (BW825C) is a short acting histamine 1 receptor antagonist for the treatment of allergic rhinitis.
ACSS2 INHIBITOR
CAS:508186-14-9
Formula: C20H18N4O2S2
DC10492
>98%
ACSS2 inhibitor is a novel ACSS2 inhibitor.
ACT058362 (PALOSURAN)
CAS:540769-28-6
Trade Name: ACT058362,ACT-058362
Formula: C25H30N4O2
DC7970
>98%
Palosuran (ACT-058362) is a new potent and specific antagonist of the human UT receptor with an IC50 of 3.60.2 nM.
ACTB-1003
CAS:939805-30-8
Trade Name: ACTB1003,ACTB 1003
Formula: C27H26F5N7O3
DC7997
>98%
ACTB-1003 is a potent inhibitor of FGFR1 with IC50 <10 nM in FGFR-1 biochemical assay; more information can be find in Patent WO/2007/064883A2, Example 12.
ACTINOMYCIN D
CAS:50-76-0
Formula: C62H86N12O16
DC4197
99%
Dactinomycin (also known generically as Actinomycin D ) is the most significant member of actinomycines, which are a class of polypeptide antibiotics isolated from soil bacteria of the genus Streptomyces.
ACUMAPIMOD
CAS:836683-15-9
Formula: C22H19N5O2
DC10417
>98%
Acumapimod (BCT197) is an orally active p38 MAP kinase inhibitor, with an IC50 of less than 1 M for p38a.
ACY-738
CAS:1375465-91-0
Trade Name: ACY738,ACY-738,ACY 738
Formula: C14H14N4O2
DC8476
>98%
ACY-738 demonstrates inhibitory activity against recombinant HDAC6 with IC50 values of 1.7 nM, with respective average selectivity over class I HDACs being 100-fold.
ACYCLOVIR(ACICLOVIR)
CAS:59277-89-3
Trade Name: Aciclovir, Acycloguanosine, Zovirax
Formula: C8H11N5O3
DCAPI1273
>99%
Acyclovir (Aciclovir)
AD80
CAS:1384071-99-1
Formula: C22H19F4N7O
DC10633
>98%
AD80, a multikinase inhibitor, shows strong activity against human RET, BRAF, S6K, and SRC but were much less active than either AD57 or AD58 against mTOR. The IC50 value for RET is 4 nM.
ADAMANTANE
CAS:281-23-2
Formula: C10H16
DCJ-016
>98%,Standard References Grade
>98%,Standard References
ADAPALENE
CAS:106685-40-9
Trade Name: Differin
Formula: C28H28O3
DCAPI1013
>99%
Adapalene
ADAROTENE
CAS:496868-77-0
Trade Name: ST 1926;ST-1926;ST1926
Formula: C25H26O3
DC9362
>98%
Adarotene (ST1926) is an effective apoptosis inducer and surprisingly produced DNA damage.ST1926 exhibites a potent antiproliferative activity on a large panel of human tumor cells._x000D_IC50 value: 0.12 uM (LNCaP cell) [1]_x000D_Target: Apoptosis inducer; Antican
ADEFOVIR DIPIVOXIL
CAS:142340-99-6
Trade Name: Bis-POM PMEA, Preveon, Hepsera
Formula: C20H32N5O8P
DC4155
99%
Adefovir Dipivoxil(Preveon, Hepsera) works by blocking reverse transcriptase, an enzyme that is crucial for the hepatitis B virus (HBV) to reproduce in the body.
ADEMETIONINE DISULFATE TOSYLATE
CAS:97540-22-2
Trade Name: Ademetionine disulfate tosylate
Formula: C22H34N6O16S4
DC10244
>98%
Ademetionine Disulfate Tosylate is the disulfate-tosylate mixed salt of a mixture of diastereoisomers of the ademetionine ions. Ademetionine possesses anti-inflammatory activity and has been used in treatment of chronic liver disease.
ADENINE
CAS:73-24-5
Formula: C5H5N5
DCX-060
>98%,Standard References Grade
>98%,Standard References
ADENOSINE (ADENOCARD)
CAS:58-61-7
Trade Name: Adenocard
Formula: C10H13N5O4
DCAPI1268
>99%
Adenosine (Adenocard)
ADIPHENINE HCL
CAS:50-42-0
Trade Name: N/A
Formula: C20H25NO2DCAPI1201
>99%
Adiphenine HCl
ADIPORON
CAS:924416-43-3
Formula: C27H28N2O3
DC7049
>98%
AdipoRon is a novel small-molecule AdipoR agonist; binds to both AdipoR1(Kd= 1.8 uM) and AdipoR2(Kd=3.1 uM).
ADJUDIN (AF-2364)
CAS:252025-52-8
Trade Name: AF-2364,AF 2364,AF2364
Formula: C15H12Cl2N4O
DC8355
>98%
AF-2364, an analogue of Lonidamine (LND), had a contraceptive effect when orally administered to adult SpragueDawley rats.
ADL5859 HCL
CAS:850173-95-4
Trade Name: ADL 5859,ADL-5859
Formula: C24H28N2O3.HCl
DC7050
>98%
ADONITO
CAS:488-81-3
Formula: C5H12O5
DCA-012
>98%,Standard References Grade
>98%,Standard References
ADOPRAZINE
CAS:222551-17-9
Trade Name: SLV 313;SLV313;SLV-313
Formula: C24H24FN3O2
DC9324
>98%
Adoprazine, a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties._x000D_
ADRAFINIL
CAS:63547-13-7
Trade Name: CRL 40028;Olmifon
Formula: C15H15NO3S
DC9549
>98%
Adrafinil (CRL-40028, Olmifon), prodrug of modafinil, is a mild central nervous system stimulant drug used to relieve excessive sleepiness and inattention, Adrafinil is believed to serve as an alpha-1 adrenoceptor agonist._x000D_
ADT-OH
CAS:18274-81-2
Trade Name: ACS1
Formula: C9H6OS3
DC10577
>98%
ADT-OH is a derivative of anethole dithiolethione (ADT) and synthetic hydrogen sulfide (H2S) donor.
ADX 47273
CAS:851881-60-2
Trade Name: ADX-47273,ADX47273
Formula: C20H17F2N3O2
DC8087
>98%
ADX-47273 is a novel, potent and selective metabotropic glutamate receptor 5 allosteric modulator with an EC50 of 170 nM.
ADX-88178
CAS:1235318-89-4
Trade Name: ADX-88178,ADX 88178,ADX88178
Formula: C12H12N6S
DC10465
>98%
ADX-88178 is a novel potent, selective, and brain-penetrant positive allosteric modulator of the mGlu4 receptor.
AEBSF-HYDROCHLORIDE
CAS:30827-99-7
Formula: C8H11ClFNO2S
DC7703
>98%
AEBSF HCl is a broad spectrum, irreversible serine protease inhibitor.
AEE-788(NVP-AEE788)
CAS:497839-62-0
Trade Name: AEE788
Formula: C27H32N6
DC5113
>98%
AEE788 is a potent inhibitor of EGFR and HER2/ErbB2 with IC50 of 2 nM and 6 nM, less potent to VEGFR2/KDR, c-Abl, c-Src, and Flt-1, does not inhibit Ins-R, IGF-1R, PKCa and CDK1. Phase 1/2.
AEGR-733(LOMITAPIDE)
CAS:182431-12-5
Trade Name: AEGR-733; BMS-201038; AEGR733; BMS201038; AEGR 733; BMS 201038,
Formula: C39H37F6N3O2
DC7900
>98%
Lomitapide (AEGR-733) is a novel proprietary MTP-inhibitor.
AESCIN IA
CAS:123748-68-5
Formula: C55H86O24
DCQ-063
>98%,Standard References Grade
>98%,Standard References
AESCULUSIDE B
CAS:26339-92-4
Formula: C48H78O22
DCQ-090
>98%,Standard References Grade
>98%,Standard References
AF-353
CAS:865305-30-2
Trade Name: CHEMBL526307,AF 353,AF353
Formula: C14H17IN4O2
DC7783
>98%
AF-353 is a novel, orally bioavailable, highly potent and selective P2X3/P2X2/3 receptor antagonist.
AFATINIB (BIBW2992)
CAS:439081-18-2
Trade Name: Afatinib, BIBW2992,BIBW-2292
Formula: C24H25ClFN5O3
DC1024
99%
BIBW2992 (Afatinib, Tomtovok, Tovok) irreversibly inhibits EGFR/HER2 including EGFRwt, EGFRL858R, EGFRL858R/T790M and HER2 with IC50 of 0.5 nM, 0.4 nM, 10 nM and 14 nM, respectively.
AFLOQUALONE
CAS:56287-74-2
Formula: C16H14FN3O
DC9026
>98%
Afloqualone is a agonist of GABA receptor .
AFN-1252(DEBIO 1452)
CAS:620175-39-5
Trade Name: API1252; Debio1452,API 1252; Debio-1452,API1252; Debio1452
Formula: C22H21N3O3
DC10513
>98%
AFN-1252(Debio 1452) is a potent inhibitor of enoyl-acyl carrier protein reductase (FabI), inhibited all clinical isolates of Staphylococcus aureus and Staphylococcus epidermidis at concentrations of =0.12 g/ml.
AFOXOLANER
CAS:1093861-60-9
Trade Name: Afoxolaner
Formula: C26H17ClF9N3O3
DC9764
>98%
Afoxolaner is an isoxazoline that inhibits insect and acarine ligand-gated chloride channels, in particular those gated by the neurotransmitter gamma-aminobutyric acid (GABA), blocking pre and post synaptic transfer of chloride ions across cell membranes.
AFURESERTIB (GSK2110183)
CAS:1047644-62-1
Formula: C18H17Cl2FN4OS
DC8411
>98%
Afuresertib (GSK2110183) is a potent, orally bioavailable Akt inhibitor with Ki of 0.08 nM, 2 nM, and 2.6 nM for Akt1, Akt2, and Akt3, respectively. Phase 2.
AFURESERTIB HCL (GSK-2110183)
CAS:1047645-82-8
Trade Name: Afuresertib,GSK 2110183,GSK2110183
Formula: C18H18Cl3FN4OS
DC7994
>98%
Afuresertib (GSK2110183) is a potent pan-AKT inhibitor that demonstrated synergy with bortezomib in preclinical models of multiple myeloma (MM).
AG 1406
CAS:71308-34-4
Trade Name: AG1406,AG-1406
Formula: C16H18N2O
DC10589
>98%
AG 1406 is a selective inhibitor of the receptor tyrosine kinase VEGF receptor 2 .
AG-024322
CAS:837364-57-5
Trade Name: AG-024322; AG24322; AG 024322.
Formula: C23H20F2N6
DC7164
>98%
AG-24322 is a second generation CDK inhibitor. AG-024322 is a potent inhibitor of CDK1, CDK2, and CDK4 that produces cell-cycle arrest and antitumor activity in preclinical models. The no-adverse-effect dose of AG-024322 was 2 mg/kg and associated with ov
AG-1024 (TYRPHOSTIN)
CAS:65678-07-1
Trade Name: AG1024; Tyrphostin AG 1024
Formula: C14H13BrN2O
DC7052
>98%
AG-1024 (Tyrphostin) inhibits IGF-1R autophosphorylation with IC50 of 7 M, less potent to IR with IC50 of 57 M.
AG-120(IVOSIDENIB)
CAS:1448347-49-6
Trade Name: AG120,AG 120
Formula: C28H22ClF3N6O3
DC8051
>98%
AG-120 is a first-in-class, orally available, selective, potent inhibitor of the mutated IDH1 protein.
AG-1478 (TYRPHOSTIN AG-1478)
CAS:153436-53-4
Trade Name: AG1478, Tyrphostin AG1478, AG 1478
Formula: C16H14ClN3O2
DC1078
>98%
AG-1478 (Tyrphostin AG-1478) is a selective EGFR inhibitor with IC50 of 3 nM.
AG-1557
CAS:189290-58-2
Trade Name: AG 1557,AG1557
Formula: C16H14IN3O2
DC8079
>98%
AG-1557 is an ultra-potent inhibitor of epidermal growth factor receptor tyrosine kinase (EGFRK).
AG-18
CAS:118409-57-7
Trade Name: RG-50810; Tyrphostin A23; AG-18; AG18; RG 50810; RG50810
Formula: C10H6N2O2
DC7051
>98%
AG-18(RG-50810; Tyrphostin A23) inhibits EGFR with IC50 of 40 M.
AG-221(ENASIDENIB)
CAS:1446502-11-9
Trade Name: AG221,AG 221
Formula: C19H17F6N7O
DC8374
>98%
AG-221 is an orally available, selective, potent inhibitor of the mutated IDH2 protein.
AG-494
CAS:133550-35-3
Trade Name: AG-494,AG 494,AG494
Formula: C16H12N2O3
DC10623
>98%
AG-494 is an inhibitor of epidermal growth factor receptor kinase with an IC50 value of 1 M in HT-22 cells.
AG-L-59687
CAS:793035-88-8
Trade Name: AGL-59687
Formula: C24H34BrN5O7S
DC2063
>98%
0
AG13958
CAS:319460-94-1
Trade Name: AG 13958,AG-13958
Formula: C26H22FN7O
DC8507
>98%
AG13958 is a VEGF inhibitor that was clinical development by Pfizer in 2006-07 for treatment of age-related macular degeneration (AMD).
AG14361
CAS:328543-09-5
Trade Name: AG14361; AG-14361; AG 14361.
Formula: C19H20N4O
DC5106
>98%
AG14361 is a potent inhibitor of PARP1 with Ki of <5 nM. It is at least 1000-fold more potent than the benzamides.
AG490
CAS:133550-30-8
Trade Name: AG-490,AG 490
Formula: C17H14N2O3
DC2096
>98%
AG-490 (Tyrphostin B42) is an inhibitor of EGFR, ErbB2 and JAK2 with IC50 of 0.1 M, 13.5 M, and ~10 M, respectively.
AG879
CAS:148741-30-4
Trade Name: AG 879,AG-879
Formula: C18H24N2OS
DC8557
>98%
Tyrphostin AG 879 is a protein tyrosine kinase inhibitor with potent effects on TrkA.
AG881
CAS:1644545-52-7
Trade Name: AG 881, AG-881
Formula: C14H12ClN6F6
DC10439
>98%
AG-881 is a potent and selective orally available inhibitor of mutated forms of both isocitrate dehydrogenase type 1 (IDH1) in the cytoplasm and type 2 (IDH2).
AGI-5198
CAS:1355326-35-0
Trade Name: IDH-C35,AGI5198,AGI 5196
Formula: C27H31FN4O2
DC5050
>98%
AGI-5198 is the first highly potent and selective inhibitor of IDH1 R132H/R132C mutants with IC50 of 0.07 M/0.16 M.
AGI-6780
CAS:1432660-47-3
Trade Name: AGI 6780; AGI6780
Formula: C21H18F3N3O3S
DC7174
>98%
AGI-6780 is the first highly potent and selective small molecule inhibitor of isocitrate dehydrogenases, which binds in an allosteric manner at the dimer interface of mutant IDH2-R140Q (IC50=23 nM).
AGK2
CAS:304896-28-4
Trade Name: AGK2,AGK-2,AGK 2
Formula: C23H13Cl2N3O2
DC8437
>98%
AGK2 is a potent, and selective SIRT2 inhibitor with IC50 of 3.5 M.
AGN 194310
CAS:229961-45-9
Trade Name: AGN194310; AGN-194310; VTP194310; VTP 194310; VTP-194310
Formula: C28H24O2S
DC7767
>98%
AGN 194310(VTP-194310) is a potent and selective pan-RARs agonist with Kd values of 3/2/5 nM for RARa//? respectively.
AGNUSIDE
CAS:11027-63-7
Formula: C22H26O11
DCM-041
>98%,Standard References Grade
>98%,Standard References
AGOMELATINE
CAS:138112-76-2
Trade Name: Valdoxan, Melitor, Thymanax
Formula: C15H17NO2
DC3171
>98%
Agomelatine is classified as a norepinephrine-dopamine disinhibitor (NDDI) due to its antagonism of the 5-HT2C receptor.
AGRIMOL B
CAS:55576-66-4
Formula: C37H46O12
DCX-015
>98%,Standard References Grade
>98%,Standard References
AHAS INHIBITOR(BTB06584)
CAS:219793-45-0
Trade Name: BTB 06584,BTB-06584,BTB06584
Formula: C19H12ClNO6S
DC7632
>98%
AHAS inhibitor is a novel acetohydroxyacid synthase(AHAS) inhibitor, a promising drug target against Mycobacterium tuberculosis (MTB).
AHU-377 HEMICALCIUM SALT
CAS:1369773-39-6
Trade Name: AHU-377,AHU 377 ,AHU377
Formula: C24H28Ca0.5NO5
DC8735
>98%
AHU-377 is an inhibitor of neprilysin with IC50 value of 5 nM.
AHU-377(SACUBITRIL)
CAS:149709-62-6
Trade Name: AHU-377,AHU 377 ,AHU377
Formula: C24H29NO5
DC8734
>98%
AHU-377 is an inhibitor of neprilysin with IC50 value of 5 nM.
AI-10-49
CAS:1256094-72-0
Trade Name: AI 1049,AI1049
Formula: C30H22F6N6O5
DC8064
>98%
AI-10-49 selectively binds to CBF-SMMHC and disrupts its binding to RUNX1.
AICAR (ACADESINE)
CAS:2627-69-2
Trade Name: AICAR (Acadesine)
Formula: C9H14N4O5
DC7047
>98%
Acadesine results in accumulation of ZMP, which mimics the stimulating effect of AMP on AMPK and AMPK kinase. Phase 3.
AILANTHONE
CAS:981-15-7
Formula: C20H24O7
DCC-047
>98%,Standard References Grade
>98%,Standard References
AIM-100
CAS:873305-35-2
Trade Name: AIM 100;AIM100
Formula: C23H21N3O2
DC9330
>98%
AIM-100 is a small molecule inhibitor of Ack1 with an IC50 of 24 nM_x000D_IC50 value: 24 nM [3]_x000D_Target: Ack1_x000D_Ack1 inhibitor AIM-100 not only inhibited Ack1 activation but also suppressed AKT tyrosine phosphorylation, leading to cell cycle arrest in the G1 ph
AJ-97166
CAS:746667-48-1
Trade Name: 6-(3-(6-Methylpyridin-2-yl)-1H-pyrazol-4-yl)
Formula: C17H13N5
DC9674
>98%
AJUGOL
CAS:52949-83-4
Formula: C15H24O9
DCZ-150
>98%
>98%,Standard References
AKEBIA SAPONIN D
CAS:39524-08-8
Formula: C47H76O18
DCC-014
>98%,Standard References Grade
>98%,Standard References
AKP-11
CAS:1220973-37-4
Trade Name: AKP-11,AKP 11,AKP11
Formula: C22H22ClN3O5
DC10525
>98%
AKP-11 is A Novel S1P1 Agonist with Favorable Safety Profile Attenuates Experimental Autoimmune Encephalomyelitis in Rat Model of Multiple Sclerosis.
AKR1C3 INHIBITOR 5F
CAS:1275482-57-9
Trade Name: AKR1C3 Inhibitor 5f
Formula: C14H13NO3
DC9843
>98%
A highly potent and selective inhibitor of the type 5 17--hydroxysteroid dehydrogenase AKR1C3.
AKT INHIBITOR IV
CAS:681281-88-9
Formula: C31H27N4SI
DC8050
>98%
Akt Inhibitor IV is n Inhibitor of Akt protein kinase
AKT INHIBITOR VIII
CAS:612847-09-3
Formula: C34H29N7O
DC8458
>98%
Akt Inhibitor VIII is a cell-permeable quinoxaline compound that has been shown to potently, selectively, allosterically, and reversibly inhibit Akt1, Akt2, and Akt3 activity (IC50 = 58 nM, 210 nM, and 2.12 M; respectively).
AKT-I-1
CAS:473382-39-7
Trade Name: Akt-I-1,AktI1
Formula: C22H30N6
DC8509
>98%
The compound (Akt-I-1) inhibits only Akt1 (IC50 4.6 M) and does not inhibit AKT2, or AKT3.
AKT-I-1,2 HCL
CAS:473382-50-2
Formula: C23H21N3.HCl
DC10055
>98%
The compound (Akt-I-1,2) inhibited both Akt1 and Akt2 with IC50 values of 2.7 and 21 M respectively.
AKT1 AND AKT2-IN-1
CAS:893422-47-4
Formula: C33H29N7O
DC8695
>98%
Akt1 and Akt2-IN-1 is an allosteric inhibitor of Akt1 (IC50 = 3.5 nM) and Akt2 (IC50 = 42 nM), with potent and balanced activity.
AL 082D06(D-06)
CAS:256925-03-8
Trade Name: AL-082D06; D06; D-06,AL082D06
Formula: C23H24ClN3O2
DC9677
>98%
AL 082D06(D-06) is the first selective, nonsteroidal glucocorticoid receptor (GR) antagonist with Ki of 210 nM, exhibits excellent selectivity against AR, PR, MR and ER(Ki > 10 uM).
ALANTOLACTONE
CAS:546-43-0
Formula: C15H20O2
DCT-023
>98%,Standard References Grade
>98%,Standard References
ALBASPIDIN AA
CAS:3570-40-9
Formula: C21H24O8
DCM-046
>98%,Standard References Grade
>98%,Standard References
ALBASPIDIN AP
CAS:59092-91-0
Formula: C22H26O8
DCM-047
>98%,Standard References Grade
>98%,Standard References
ALBENDAZOLE(ALBENZA)
CAS:54965-21-8
Trade Name: Albenza, Eskazole, Zentel, Andazol
Formula: C12H15N3O2S
DCAPI1243
>99%
Albendazole(Albenza)
ALBIFLORIN
CAS:39011-90-0
Formula: C23H28O11
DCS-011
>98%,Standard References Grade
>98%,Standard References
ALCAFTADINE
CAS:147084-10-4
Trade Name: N/A
Formula: C19H21N3O
DCAPI1467
>99%
ALCAFTADINE
ALDA-1
CAS:349438-38-6
Trade Name: ALDA1,ALDA 1
Formula: C15H11Cl2NO3
DC8723
>98%
Alda-1 is an ALDH2 agonist, cell-permeable activator of both the wild-type ALDH2*1 and the asian E487K mutant ALDH2*2 forms of mitochondrial aldehyde dehydrogenase 2 (mtALDH2).
ALDOXORUBICINHCL
CAS:1361563-03-2
Trade Name: Aldoxorubicin HCl, CHEMBL2107827, 1361563-03-2, D10384
Formula: C37H43ClN4O13
DC7355
>98%
Inhibitor of reverse transcriptase and RNA polymerase; immunosuppressive agent; intercalates in DNA.
ALENDRONATE(FOSAMAX)
CAS:121268-17-5
Trade Name: N/A
Formula: C4H13NO7P2.3H2O.Na
DCAPI1034
>99%
Alendronate (Fosamax)
ALFACALCIDOL
CAS:41294-56-8
Trade Name: N/A
Formula: C27H44O2
DCAPI1534
>99%
1a-Hydroxyvitamin D3 is a form of vitamin D that helps the body absorb calcium from food.
ALFUZOSIN
CAS:81403-80-7
Trade Name: SL 77499
Formula: C19H27N5O4
DC9334
>98%
Alfuzosin is an a1 adrenergic receptor antagonist used to treat benign prostatic hyperplasia (BPH)._x000D_
ALISKIREN HEMIFUMARATE
CAS:173334-58-2
Trade Name: N/A
Formula: 2(C30H53N3O6).C4H4O4
DCAPI1495
>99%
Aliskiren hemifumarate(CGP 60536) is a direct renin inhibitor with IC50 of 1.5 nM.
ALISMOXIDE
CAS:87701-68-6
Formula: C15H26O2
DCH-034
>98%,Standard References Grade
>98%,Standard References
ALISOL A
CAS:19885-10-0
Formula: C30H50O5
DCZ-044
>98%,Standard References Grade
>98%,Standard References
ALISOL A 24-ACETATE
CAS:18674-16-3
Formula: C32H52O6
DCZ-061
>98%,Standard References Grade
>98%,Standard References
ALISOL B
CAS:18649-93-9
Formula: C28H44O4
DCZ-045
>98%,Standard References Grade
>98%,Standard References
ALISOL B 23-ACETATE
CAS:26575-95-1
Formula: C28H44O4
DCY-036
>98%,Standard References Grade
>98%,Standard References
ALISOL C MONOACETATE
CAS:26575-93-9
Formula: C32H48O6
DCZ-062
>98%,Standard References Grade
>98%,Standard References
ALIZARIN
CAS:72-48-0
Formula: C14 H8 O4
DCT-039
>98%,Standard References Grade
>98%,Standard References
ALK INHIBITOR 1
CAS:761436-81-1
Trade Name: Benzenesulfonamide, 2-[[5-bromo-2-[[2-methoxy-4-(4-methyl-1-piperazinyl)phenyl]amino]-4-pyrimidinyl]
Formula: C23H28BrN7O3S
DC9338
>98%
ALK inhibitor 1 is a novel and selective inhibitor for the ALK kinase.
ALK INHIBITOR 2
CAS:761438-38-4
Trade Name: Benzenesulfonamide, 2-[[5-chloro-2-[[2-methoxy-4-(4-methyl-1-piperazinyl)phenyl]amino]-4-pyrimidinyl
Formula: C23H28ClN7O3S
DC9339
>98%
ALK inhibitor 2 is a novel and selective inhibitor for the ALK kinase.
ALLANTOIN
CAS:97-59-6
Formula: C4H6N4O3
DCN-015
>98%,Standard References Grade
>98%,Standard References
ALLASECURININE
CAS:N/A
Formula: C13H15NO2
DCZ-284
>98%
purity >98%,Standard References
ALLICIN
CAS:539-86-6
Formula: C6H10OS2
DCD-065
>98%,Standard References Grade
>98%,Standard References
ALLIIN
CAS:556-27-4
Formula: C6H11NO3S
DCS-053
>98%,Standard References Grade
>98%,Standard References
ALLM (CALPAIN INHIBITOR)
CAS:136632-32-1
Trade Name: ALLM (Calpain Inhibitor),Ac-LLM-CHO
Formula: C19H35N3O4S1
DC8106
>95%
ALLM (Calpain Inhibitor) is cell-permeable, peptide aldehyde inhibitor of calpains and cathepsins.
ALLO-1
CAS:37468-32-9
Formula: C17H15ClN2O2
DC8570
>98%
ALLO-1 is a SMO antagonist that inhibits both wild-type (IC50 = 50 nM) and mutant SMO, including the D473H SMO mutant (IC50s = 300-1000 nM).
ALLOCRYPTOPINE
CAS:485-91-6
Formula: C21H23NO5
DCB-059
>98%,Standard References Grade
>98%,Standard References
ALLOPREGNANOLONE
CAS:516-54-1
Trade Name: 3a,5a-THP; SAGE547; SAGE 547; SAGE-547
Formula: C21H34O2
DC10311
>98%
Allopregnanolone is a progesterone metabolite. Allopregnanolone is an allosteric modulator of the GABA receptor.
ALLOPURINOL
CAS:315-30-0
Formula: C5H4N4O
DC8945
>98%
Allopurinol (Zyloprim) is a xanthine oxidase inhibitor with an IC50 of 7.820.12 M.
ALLOPURINOL RIBOSIDE
CAS:16220-07-8
Formula: C10H12N4O5
DC10303
>98%
Allopurinol riboside, a metabolite of allopurinol, shows potent activities against parasites.
ALLOPURINOL SODIUM (ALOPRIM)
CAS:17795-21-0
Trade Name: Lopurin, Zyloprim, Aloprim
Formula: C5H4N4NaO
DCAPI1097
>99%
Allopurinol Sodium (Aloprim)
ALMOREXANT HCL (ACT-078573)
CAS:913358-93-7
Trade Name: ACT-078573; ACT 078573; ACT078573
Formula: C29H32ClF3N2O3
DC7692
>98%
Almorexant(ACT078573) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM for OX1 and OX2, respectively.
ALMOTRIPTAN
CAS:154323-57-6
Trade Name: N/A
Formula: C17H25N3O2S
DCAPI1478
>99%
Almotriptan
ALMOTRIPTAN MALATE(PNU180638)
CAS:181183-52-8
Trade Name: Axert; Almogran; PNU-180638,PNU 180638
Formula: C21H31N3O7S
DC8284
>98%
Almotriptan Malate is a 5-HT1B/1D-receptor agonist used to treat migraine.
ALNUSONE
CAS:33457-62-4
Formula: C19H18O
DCQ-061
>98%,Standard References Grade
>98%,Standard References
ALOEEMODIN
CAS:481-72-1
Formula: C15H10O5
DCL-014
>98%,Standard References Grade
>98%,Standard References
ALOGLIPTIN
CAS:850649-61-5
Trade Name: N/A
Formula: C18H21N5O2
DCAPI1579
>99%
Alogliptin
ALOGLIPTIN BENZOATE
CAS:850649-62-6
Trade Name: Nesina; SYR 322
Formula: C25H27N5O4
DC5076
>98%
Alogliptin is an orally administered, anti-diabetic drug in the DPP-4 inhibitor class. A randomized clinical trial reporting in 2011 aimed to determine the efficacy and safety of alogliptin versus placebo and voglibose among newly diagnosed Type 2 diabete
ALOSETRON HYDROCHLORIDE
CAS:122852-69-1
Trade Name: Alosetron Hydrochloride
Formula: C17H18N4O.HCl
DC10234
>98%
Alosetron Hydrochloride is the hydrochloride salt form of alosetron, a potent and selective 5-HT3 receptor antagonist.
ALPELISIB(BYL-719)
CAS:1217486-61-7
Trade Name: BYL 719; BYL719
Formula: C19H22F3N5O2S
DC7094
>98%
BYL719 is a potent and selective PI3Ka inhibitor with IC50 of 5 nM, ;liitle or no effect on PI3K/?/d.
ALPHA-BOSWELLIC ACID,3-ACETYL
DCY-089
>98%,Standard References Grade
>98%,Standard References
ALPHA-HEDERIN
CAS:27013-91-8
Formula: C42H68O12
DC9920
>98%
alpha-hederin is a water-soluble pentacyclic triterpenoid saponin, possessing several biological properties such as antispasmodic, moliscicidic, anthelmithic and inhibiting cell proliferation.
ALPHA-VINIFERIN
CAS:62218-13-7
Formula: C42H30O9
DCP-008
>98%,Standard References Grade
>98%,Standard References
ALPINETIN
CAS:36052-37-6
Formula: C16H14O4
DCS-034
>98%,Standard References Grade
>98%,Standard References
ALPROSTADIL(CAVERJECT)
CAS:745-65-3
Trade Name: Prostaglandin E1, Edex, Muse, Liprostin
Formula: C20H34O5
DCAPI1328
>99%
Alprostadil(Caverject)
ALS-22335
CAS:N/A
Trade Name: ALS-22335,ALS 22335,ALS22335
Formula: C23H31FN3O10P
DC8366
>98%
ALS-22335,ALS 22335,ALS22335
ALSERIN
CAS:50-55-5
Formula: C33H40N2O9
DCL-022
>98%,Standard References Grade
>98%,Standard References
ALSTERPAULLONE
CAS:237430-03-4
Trade Name: 9-Nitropaullone
Formula: C16H11N3O3
DC9838
>98%
Alsterpaullone is a potent ATP-competitive and cell cycle cyclin-dependent kinase inhibitor, that is reported to be the most active Paullone.
ALTIRATINIB(DCC-2701)
CAS:1345847-93-9
Trade Name: Altiratinib, DCC2701,DCC 2701
Formula: C26H21F3N4O4
DC8072
>98%
Altiratinib is a MET/TIE2/VEGFR2/TRK (A,B,C) kinase inhibitor in Phase 1 clinical development for the treatment of invasive solid tumors including glioblastoma.
ALTRETAMINE(HEXALEN)
CAS:645-05-6,2975-00-0(HCl)
Trade Name: Hexalen
Formula: C9H18N6
DCAPI1290
>99%
Altretamine (Hexalen)
ALVELESTAT (AZD9668)
CAS:848141-11-7
Trade Name: AZD9668; AZD-9668; AZD 9668
Formula: C25H25N5O4S
DC7079
>98%
Alvelestat (AZD9668) is a novel, oral inhibitor of neutrophil elastase (NE) with the pIC50 of 7.9 for Human NE.
ALVERINE CITRATE
CAS:5560-59-8
Trade Name: N/A
Formula: C20H27N.C6H8O7
DCAPI1250
>99%
Alverine citrate is a drug used for functional gastrointestinal disorders.
ALVESPIMYCIN (HYDROCHLORIDE)
CAS:467214-21-7
Trade Name: 17-DMAG; KOS-1022; NSC 707545
Formula: C32H49ClN4O8
DC9483
>98%
Alvespimycin Hcl(17-DMAG;NSC 707545) is a potent, water-soluble HSP90 inhibitor with IC50 of 62 nM._x000D_
ALVIMOPAN
CAS:156053-89-3
Formula: C25H32N2O4
DC8584
>98%
Alvimopan(LY 246736; ADL 8-2698) is a peripherally acting mu-opioid receptor (PAM-OR, IC50= 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery.
ALVIMOPAN DIHYDRATE
CAS:170098-38-1
Formula: C25H36N2O6
DC8605
>98%
Alvimopan(LY 246736; ADL 8-2698) is a peripherally acting mu-opioid receptor (PAM-OR, IC50= 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery.
ALVIMOPAN MONOHYDRATE
CAS:1383577-62-5
Formula: C25H34N2O5
DC8606
>98%
Alvimopan(LY 246736; ADL 8-2698) is a peripherally acting mu-opioid receptor (PAM-OR, IC50= 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery.
ALW-II-41-27
CAS:1186206-79-0
Trade Name: Eph receptor tyrosine kinase inhibitor
Formula: C32H32F3N5O2S
DC10209
>98%
ALW-II-41-27 is a novel Eph receptor tyrosine kinase inhibitor, used for cancer treatment.
AM 281
CAS:202463-68-1
Formula: C21H19Cl2IN4O2
DC7251
>98%
Potent, selective CB1 cannabinoid receptor antagonist/inverse agonist (Ki values are 12 and 4200 nM for CB1 and CB2 receptors respectively). Increases locomotor activity following systemic administration in vivo. Analog of SR141716A (Ki = 14 nM).
AM-2394
CAS:1442684-77-6
Trade Name: AM2394,AM 2394
Formula: C22H25N5O4
DC9830
>98%
AM-2394 is a potent and selective Glucokinase agonist (GKA), which catalyzes the phosphorylation of glucose to glucose-6-phosphate.
AM095
CAS:1345614-59-6
Trade Name: AM-095,AM095,AM 095
Formula: C27H23N2NaO5
DC8621
>98%
AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 M for recombinant human or mouse LPA1 respectively.
AM095 FREE ACID
CAS:1228690-36-5
Trade Name: AM-095,AM095,AM 095
Formula: C27H24N2O5
DC8622
>98%
AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 M for recombinant human or mouse LPA1 respectively.
AM2099
CAS:1443373-17-8
Trade Name: AM 2099,AM-2099
Formula: C19H13F3N4O3S2
DC9909
>98%
AM-2099 is a potent and selective NaV1.7 Inhibitor.
AM251
CAS:183232-66-8
Trade Name: AM-251
Formula: C22H21Cl2IN4O
DC8765
>98%
AM251 is a potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 306-fold selectivity over CB2 receptors; also potent GPR55 agonist (EC50 = 39 nM).
AM580
CAS:102121-60-8
Trade Name: AM-580,AM 580,CD336; NSC608001; Ro 40-6055
Formula: C22H25NO3
DC7054
>98%
A retinoic acid analog and selective RARa agonist
AM679
CAS:1206880-66-1
Trade Name: AM-679;AM 679
Formula: C40H44N4O5S
DC9447
>98%
AM679 is a potent and selective FLAP inhibitor with IC50s of 2.2 nM/0.6 nM/154 nM for FLAP binding/hLA/hWB respectively.
AM966
CAS:1228690-19-4
Trade Name: AM966,AM-966,AM 966
Formula: C27H23ClN2O5
DC8623
>98%
AM966 is a high affinity, selective, oral LPA1 (lysophosphatidic acid receptor, IC50=17 nM) antagonist, with selectivity for this receptor over the other LPA receptors.
AMANTADINE HCL
CAS:665-66-7
Formula: C10H18ClN
DC8958
>98%
Amantadine Hydrochloride is an antiviral and an antiparkinsonian drug.
AMBRISENTAN
CAS:177036-94-1
Trade Name: N/A
Formula: C22H22N2O4
DCAPI1496
>99%
A nonpeptide endothelin ETA receptor antagonist. Antihypertensive.
AMBROXOL HCL
CAS:23828-92-4
Formula: C13H19Br2ClN2O
DC9126
>98%
AMCASERTIB(BBI503)
CAS:1129403-56-0
Trade Name: BBI 503,BBI-503
Formula: C31H33N5O2S
DC10372
>98%
Amcasertib(BBI503) is an orally administered investigational agent designed to inhibit cancer stem cell pathways, including Nanog, by targeting stemness kinases.
AMD3465
CAS:185991-07-5
Trade Name: AMD3465,AMD-3465,AMD 3465
Formula: C24H38N6.6HBr
DC5056
>98%
AMD3465 is a Potent, selective CXCR4 antagonist; exhibits 8-fold higher affinity than AMD 3100 (Cat.No. 3299). Inhibits SDF-1a-ligand binding (Ki = 41.7 nM).
AMENAMEVIR
CAS:841301-32-4
Trade Name: ASP2151,ASP 2151,ASP-2151
Formula: C24H26N4O5S
DC10621
>98%
Amenamevir, also known as ASP2151, is a herpes virus helicase-primase inhibitor.
AMENTOFLAVONE
CAS:1617-53-4
Formula: C30H18O10
DCS-044
>98%,Standard References Grade
>98%,Standard References
AMETANTRONE
CAS:64862-96-0
Trade Name: CI-881; NSC 196473; NSC 287513; NSC-196473; NSC-287513; ametantrone diacetate.
Formula: C22H28N4O4
DC7356
>98%
Ametantrone is a new anthracenedione antineoplastic agents, produced a concentration-dependent inhibition of hepatic microsomal lipid peroxidation.
AMFENAC SODIUM
CAS:61618-27-7
Formula: C15H12NNaO3.H2O
DC9036
>98%
AMG 837 (CALCIUM HYDRATE)
CAS:1259389-38-2
Trade Name: AMG-837 calcium hydrate;AMG837 calcium hydrate
Formula: C26H22F3O4-
DC9457
>98%
AMG 837 calcium hydrate is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents._x000D_
AMG 853(AMG853;VIDUPIPRANT)
CAS:1169483-24-2
Trade Name: AMG-853, AMG853, Vidupiprant
Formula: C28H27Cl2FN2O6S
DC6310
>98%
AMG 853 is novel a CRTH2 and DP Dual Antagonist.
AMG 900
CAS:945595-80-2
Trade Name: AMG-900;AMG900
Formula: C28H21N7OS
DC9366
>98%
AMG 900 is a potent and highly selective pan-Aurora kinases inhibitor for Aurora A/B/C with IC50 of 5 nM/4 nM /1 nM; >10-fold selective for Aurora kinases than p38a, Tyk2, JNK2, Met and Tie2.
AMG 925
CAS:1401033-86-0
Trade Name: AMG 925,AMG925,AMG-925
Formula: C26H29N7O2
DC8397
>98%
AMG 925 is a potent and selective dual inhibtor of CDK4/FLT3 with IC50s of 1.5 nM and 2.4 nM for CDK4 and FLT3, respectively; with IC50 of 19 nM in MOLM-13 cell.
AMG-1
CAS:913376-84-8
Trade Name: AMG1,AMG 1
Formula: C31H29FN4O5
DC8514
>98%
AMG-1 is a potent inhibitor of human c-Met and RON with IC50 values of 4 and 9 nmol/L respectively.
AMG-208
CAS:1002304-34-8
Trade Name: AMG208; AMG 208
Formula: C22H17N5O2
DC7056
>98%
AMG-208 is a potent small molecular c-Met inhibitor with an IC50 of 9.3 nM.
AMG-25
CAS:1003311-62-3
Trade Name: AMG25,AMG 25
Formula: C23H17N5O2
DC10051
>95%
AMG-25 exhibits potent inhibition of c-Kit with greater than 200-fold selectivity over KDR, p38, Lck and Src.
AMG-319
CAS:1608125-21-8
Trade Name: AMG-319,AMG 319,AMG319
Formula: C21H16FN7
DC8618
>98%
AMG 319 is an investigational, highly selective, small molecule inhibitor of PI3Kd that blocks B cell proliferation following BCR stimulation both in vitro and in vivo, inhibits basal AKT phosphorylation, and inhibits proliferation in lymphoid tumor cells
AMG-3969
CAS:1361224-53-4
Trade Name: AMG3969,AMG 3969
Formula: C21H20F6N4O3S
DC10101
>98%
AMG-3969 is a potent glucokinase-glucokinase regulatory protein interaction (GK-GKRP) disruptor with an IC50 of 4 nM.
AMG-47A
CAS:882663-88-9
Trade Name: AMG 47,AMG-47,AMG47
Formula: C29H28F3N5O2
DC7001
>98%
AMG-47a is a potent inhibitor of Lck and T cell proliferation; exhibits anti-inflammatory activity (ED50 = 11 mg/kg) in the anti-CD3 induced production of IL-2 in mice.
AMG-837
CAS:865231-46-5
Trade Name: AMG-837; AMG837
Formula: C26H21F3O3
DC7867
>98%
AMG 837 is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents.
AMG-TIE2-1
CAS:870223-96-4
Trade Name: 870223-96-4; AMG-Tie2; AMG-Tie2-1; 4-methyl-3-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-yloxy)-N-(
Formula: C25H20F3N5O2
DC8503
>98%
AMG-Tie2-1 is a highly potent, non-selective inhibitor of Tie-2 (IC50 <1 nM).
AMG232
CAS:1352066-68-2
Trade Name: AMG-232,AMG 232
Formula: C28H35Cl2NO5S
DC9793
>98%
AMG232 is a potent, selective and orally bioavailable inhibitor of MDM2-p53 interaction with IC50 value of 9.1 nM in EdU cells .
AMG337
CAS:1173699-31-4
Trade Name: AMG 337,AMG-337
Formula: C23H22FN7O3
DC8845
>98%
AMG-337 is a potent and highly selective small molecule ATP-competitive MET kinase inhibitor. AMG 337 inhibits MET kinase activity with an IC50 of < 5nM in enzymatic assays.
AMG517
CAS:659730-32-2
Trade Name: AMG517; AMG-517
Formula: C20H13F3N4O2S
DC7055
>98%
AMG 517 is a potent and selective TRPV1 antagonist, antagonizes capsaicin, proton, and heat activation of TRPV1 with IC50 of 0.76 nM, 0.62 nM and 1.3 nM.
AMG9810
CAS:545395-94-6
Trade Name: AMG 9810,AMG-9810
Formula: C24H24ClFN2O
DC10132
>98%
AMG9810 is a potent and selective, competitive vanilloid TRPV1 receptor antagonist (IC50 = 17 nM).
AMI-1
CAS:20324-87-2
Trade Name: AMI-1,AMI 1,AMI1
Formula: C21H12N2O9S24Na
DC8292
>98%
AMI-1 is a PRMT and HIV-1 RT polymerase inhibitor.
AMICARBAZONE
CAS:129909-90-6
Trade Name: BAY314666; BAY-MKH 3586;BAY 314666; BAY-MKH3586
Formula: C10H19N5O2
DC9548
>98%
Amicarbazone(BAY-MKH3586; BAY314666) is a potent inhibitor of photosynthetic electron transport via binding to the Qb domain of photosystem II (PSII); herbicide with a broad spectrum of weed control._x000D_
AMIDOPYRINE
CAS:58-15-1
Trade Name: N/A
Formula: C13H17N3O
DCAPI1263
>99%
Amidopyrine is white crystalline substance used as an analgesic and antipyretic.
AMIFOSTINE
CAS:112901-68-5
Formula: C5H15N2O3PS
DC9022
>98%
AMIKACIN HYDRATE
CAS:1257517-67-1,37517-28-5(freebase)
Trade Name: N/A
Formula: C22H43N5O13.xH2O
DCAPI1043
>99%
Amikacin is an aminoglycoside antibiotic used to treat different types of bacterial infections.
AMILORIDE HYDROCHLORIDE
CAS:17440-83-4
Formula: C6H8ClN7O.HCl.2H2O
DC9042
>98%
AMINEPTINE
CAS:57574-09-1
Trade Name: Survector
Formula: C22H27NO2
DC9427
>98%
Amineptine(Survector) is a tricyclic antidepressant drug selectively blocking dopamine uptake, on 3H-imipramine binding, which was investigated in platelets of major depressed patients in conjunction with changes in clinical state._x000D_
AMINOCAPROIC ACID (AMICAR)
CAS:60-32-2
Trade Name: Amicar, ε-amino caproic acid, ε-Ahx, 6-aminohexanoic acid
Formula: C6H13NO2
DCAPI1279
>99%
Aminocaproic acid (Amicar)
AMINOGLUTETHIMIDE
CAS:125-84-8
Formula: C13H16N2O2
DC8984
>98%
Aminoglutethimide is an aromatase inhibitor with IC50 of 10 M.
AMIODARONE HCL
CAS:19774-82-4
Formula: C25H30ClI2NO3
DC9189
>98%
Amiodarone is an antiarrhythmic drug for inhibition of ATP-sensitive potassium channel with IC50 of 19.1 M.
AMLODIPINE BESYLATE
CAS:111470-99-6
Formula: C26H31ClN2O8S
DC9181
>98%
Amlodipine besylate is a long-acting calcium channel blocker.
AMMONIUM GLYCYRRHIZINATE (AMGZ)
CAS:1407-03-0
Trade Name: AMGZ
Formula: C42H62O16.NH3
DCAPI1067
>99%
Ammonium Glycyrrhizinate (AMGZ)
AMMOTHAMNINE
CAS:16837-52-8
Formula: C15H24N2O2
DCY-013
>98%,Standard References Grade
>98%,Standard References
AMOROLFINE HCL
CAS:78613-38-4
Trade Name: Amorolfin, Curanail, Loceryl, Locetar, Odenil
Formula: C21H35NO.HCl
DCAPI1343
>99%
Amorolfine HCl
AMOXICILLIN SODIUM(AMOX)
CAS:34642-77-8
Trade Name: Amoxycillin
Formula: C16H18N3O5S.Na
DCAPI1158
>99%
Amoxicillin sodium (Amox)
AMPICILLIN SODIUM
CAS:69-52-3,24863-47-6,57748-55-7,69-53-4(freebase)
Trade Name: N/A
Formula: C16H18N3NaO4S
DCAPI1309
>99%
Ampicillin is a beta-lactam antibiotic that is part of the aminopenicillin family.
AMPIROXICAM
CAS:99464-64-9
Trade Name: CP65703;Flucam;Nasil;CP 65703;CP-65703
Formula: C20H21N3O7S
DC9406
>98%
Ampiroxicam(CP65703) is a nonselective cyclooxygenase inhibitor uesd as anti-inflammatory drug._x000D_
AMPRENAVIR
CAS:161814-49-9
Trade Name: Agenerase
Formula: C25H35N3O6S
DC7058
>98%
Amprenavir (Agenerase) is a HIV protease inhibitor(Ki=0.6 nM) used to treat HIV infection.
AMRINONE
CAS:60719-84-8
Formula: C10H9N3O
DC8957
>98%
AMRUBICIN(SM-5887)
CAS:110267-81-7
Trade Name: Calsed; AMR
Formula: C25H25NO9
DC7002
>98%
Amrubicin(SM-5887) is a novel anthracycline derivative for treatment of bladder carcinoma.
AMSACRINE
CAS:51264-14-3
Trade Name: AMSA;m-AMSA;CI-880;SN-11841;acridinyl anisidide
Formula: C21H19N3O3S
DC9634
>98%
Amsacrine (mAMSA) an antineoplastic agent which can intercalate into the DNA of tumor cells.
AMUVATINIB (MP-470)
CAS:850879-09-3
Trade Name: MP-470; MP 470; MP470; HPK 56
Formula: C23H21N5O3S
DC7324
>98%
Amuvatinib (MP-470) is a potent and multi-targeted inhibitor of c-Kit, PDGFRa and Flt3 with IC50 of 10 nM, 40 nM and 81 nM, respectively.
AMYGDALIN
CAS:29883-15-6
Formula: C20H27NO11
DCK-001
>98%,Standard References Grade
>98%,Standard References
AN-2690(TAVABOROLE)
CAS:174671-46-6
Trade Name: Tavaborole; AN2690; AN 2690
Formula: C7H6BFO2
DC7061
>98%
AN-2690(Tavaborole), an antifungal agent with activity against Trichophyton species, in a topical solution formulation, for the potential treatment of onychomycosis.
AN3365(EPETRABOROLE)
CAS:1234563-16-6
Trade Name: AN 3365,AN-3365,GSK2251052,GSK 2251052,GSK-2251052
Formula: C11H16BNO4.HCl
DC9827
>98%
AN3365 is a first-in-class antibiotic that demonstrates potent activity across a wide spectrum of Gram-negative bacteria, including those resistant to many other antibiotics.
ANA-12
CAS:219766-25-3
Trade Name: ANA 12,ANA12
Formula: C22H21N3O3S
DC8029
>98%
ANA-12 is a potent and selective TrkB antagonist with anxiolytic and antidepressant activity in mice.
ANACARDIC ACID
CAS:16611-84-0
Formula: C22H36O3
DC8322
>98%
Anacardic acid inhibits the histone acetyltransferase (HAT) activity of the transcription co-activators p300 and p300/CREB-binding protein-associated factor (pCAF) with IC50 values of 8.5 and 5 M, respectively.
ANACETRAPIB(MK0859)
CAS:875446-37-0
Trade Name: MK-0859, MK 0859, MK0859
Formula: C30H25F10NO3
DC7804
>98%
Anacetrapib (MK0859) is a potent, selective, reversible rhCETP and mutant CETP(C13S) inhibitor with IC50 of 7.9 nM and 11.8 nM, increases HDL-C and decreases LDL-C, does not increase aldosterone or blood pressure. Phase 3.
ANAGLIPTIN
CAS:739366-20-2
Trade Name: Suiny;SK-0403
Formula: C19H25N7O2
DC9429
>98%
Anagliptin is a potent and selective DPP-4 inhibitor(IC50= 3.8 nM); > 10 fold less potent for DPP-8 and DPP-9._x000D_
ANAGRELIDE (HYDROCHLORIDE)
CAS:58579-51-4
Trade Name: Agrylin hydrochloride;Xagrid hydrochloride;BL4162A
Formula: C10H8Cl3N3O
DC9580
>98%
Anagrelide Hydrochloride(BL4162A) is a drug used for the treatment of essential thrombocytosis._x000D_
ANAMORELIN
CAS:249921-19-5
Trade Name: RC-1291; ONO-7643; RC1291; ONO7643; RC 1291; ONO 7643
Formula: C31H42N6O3
DC7357
>98%
Anamorelin(RC1291; ONO-7643) is a synthetic orally active ghrelin receptor agonist which is under development for the management of non-small lung cancer associated cachexia/anorexia.
ANASTROZOLE
CAS:120511-73-1
Trade Name: N/A
Formula: C17H19N5
DCAPI1425
>99%
Anastrozole is known to inhibit the CYP19 enzyme (aromatase, IC50 = 15 nM) that converts androgens to estrogens. Anastrozole has been seen to reversibly bind to the CYP19 enzyme through competitive inhibition.
ANAVEX 2-73
CAS:195615-84-0
Formula: C19H23NO.HCl
DC10615
>98%
Anavex 2-73 hydrochloride is a Sigma-1 Receptor agonist with an IC50 of 860 nM.
ANDARINE(GTX-007,S-4)
CAS:401900-40-1
Trade Name: GTX 007,GTX007
Formula: C19H18F3N3O6
DC8122
>98%
Andarine (S-4) is an investigational selective androgen receptor modulator (SARM) and an active partial agonist.
ANDROGRAPHOLIDE
CAS:5508-58-7
Formula: C20H30O5
DCC-010
>98%,Standard References Grade
>98%,Standard References
ANEMARSAPONIN B
CAS:139051-27-7
Formula: C45H74O18
DCZ-036
>98%,Standard References Grade
>98%,Standard References
ANEMARSAPONIN E
Formula: C46H78O19
DCZ-035
>98%,Standard References Grade
>98%,Standard References
ANEMONIN
CAS:90921-11-2
Formula: C10H8O4
DCB-069
>98%,Standard References Grade
>98%,Standard References
ANEMOSIDE B4
CAS:129741-57-7
Formula: C59H96O26
DCB-029
>98%,Standard References Grade
>98%,Standard References
ANETHOLE TRITHIONE
CAS:532-11-6
Formula: C10H8OS3
DCD-028
>98%,Standard References Grade
>98%,Standard References
ANGELOYLISOGOMISIN O
CAS:83864-70-4
Formula: C28H34O8
DCD-063
>98%,Standard References Grade
>98%,Standard References
ANGIOTENSIN II HUMAN
CAS:4474-91-3
Trade Name: Angiotensin II;Hypertensin II;Ang II;DRVYIHPF
Formula: C50H71N13O12
DC9348
>98%
Angiotensin II human is a peptide hormone that causes vasoconstriction and a subsequent increase in blood pressure._x000D_
ANGOROSIDE C
CAS:115909-22-3
Formula: C36H48O19
DCA-016
>98%,Standard References Grade
>98%,Standard References
ANIDULAFUNGIN
CAS:166663-25-8
Trade Name: N/A
Formula: C58H73N7O17
DCAPI1490
>99%
Anidulafungin
ANIRACETAM
CAS:72432-10-1
Formula: C12H13NO3
DC8976
>98%
Aniracetam(Ro 13-5057) is a nootropics and neuroprotective drug, which is selectively modulates the AMPA receptor and nAChR.
ANISIC ALDEHYDE
CAS:123-11-5
Formula: C8H8O2
DCD-024
>98%,Standard References Grade
>98%,Standard References
ANLE138B
CAS:882697-00-9
Trade Name: Anle-138b; Anle 138b
Formula: C16H11BrN2O2
DC10168
>98%
Anle138b is a novel oligomer modulator.
Anlotinib
CAS:1058156-90-3
Formula: C23H22FN3O3
DC10371
>98%
Anlotinib is a EGFR inhibitor extracted from patent 2015185012 A1, compound 1,which can be used to treat non-small cell lung cancer.
ANSAMITOCIN P-3
CAS:66547-09-9
Trade Name: Antibiotic C 15003P3; Maytansinol butyrate; C15003P3
Formula: C32H43ClN2O9
DC8241
>98%
Ansamitocin P-3, a potent anti-tumor maytansinoid found in Actinosynnema pretiosum, is a maytansine analog which displays potent cytotoxicity against the human solid tumor cell lines A-549 and HT-29.
ANTICONVULSANT 7903
CAS:82351-05-1
Trade Name: Lvguidingan,3,4-dichlorophenyl propenylisobutylamide
Formula: C13H15Cl2NO
DC9728
>98%
ANTIPYRINE
CAS:60-80-0
Formula: C11H12N2O
DC8959
>98%
Antipyrine is an analgesic and antipyretic agent
ANWULIGAN
CAS:107534-93-0
Formula: C20H24O4
DCA-015
>98%,Standard References Grade
>98%,Standard References
AP-III-A4(ENOBLOCK) HYDROCHLORIDE
CAS:1177827-73-4(freebase)
Formula: C31H44ClFN8O3
DC9247
>96.7%
ENOblock Hcl(AP-III-a4 Hcl) is a novel small molecule which is the first, nonsubstrate analogue that directly binds to enolase and inhibits its activity (IC50=0.576 uM); inhibit cancer cell metastasis in vivo.
AP219
CAS:779282-36-9
Formula: C28H34O2P
DC8581
>98%
AP219 is a control compound for AP39, containing the triphenylphosphonium scaffold but lacking the H2S-releasing portion.
APALUTAMIDE(ARN509)
CAS:956104-40-8
Trade Name: ARN 509; ARN-509
Formula: C21H15F4N5O2S
DC7064
>98%
ARN-509 is a selective and competitive androgen receptor inhibitor with IC50 of 16 nM, useful for prostate cancer treatment.
APATINIB (FREE BASE)
CAS:811803-05-1
Trade Name: Apatinib; YN968D1
Formula: C24H23N5O
DC8465
>98%
Apatinib is an orally bioavailable, small-molecule receptor tyrosine kinase inhibitor with potential antiangiogenic and antineoplastic activities.
APATINIB MESYLATE
CAS:1218779-75-9
Trade Name: N/A
Formula: C25H27N5O4S
DC4101
99%
Apatinib (YN968D1) is an orally bioavailable, selective VEGFR2 inhibitor with IC50 of 1 nM.
APD597(JNJ-38431055)
CAS:897732-93-3
Trade Name: JNJ-38431055; APD-597; APD 597; JNJ38431055; JNJ 38431055
Formula: C21H29N5O6S
DC8804
>98%
APD597(JNJ-38431055) is a GPR119 agonist intended for the treatment of type 2 diabetes, with EC50 of 46 nM for hGPR119.
APD668
CAS:832714-46-2
Trade Name: APD 668; APD-668
Formula: C21H24FN5O5S
DC7655
>98%
APD668 is a potent GPR119 agonist with EC50 of 2.7 nM and 33 nM for hGPR119 and ratGPR119 respectively.
APIGENIN
CAS:520-36-5
Formula: C15H10O5
DC5895
>98%,Standard References Grade
A plant flavonoid that has been found to inhibit cell proliferation by arresting the cell cycle at the G2/M phase.
APIGENIN 7-O-(2G-RHAMNOSYL)GENTIOBIOSIDE
CAS:174284-20-9
Formula: C33H40O19
DCQ-092
>98%,Standard References Grade
>98%,Standard References
APIGENIN-7-GLUCOSIDE,APIGENIN-7-O-SS-D-GLUCOPYRANOSIDE
CAS:578-74-5
Formula: C21H20O10
DCQ-073
>98%,Standard References Grade
>98%,Standard References
APIGENIN-7-O-GLUCURONIDE
CAS:29741-09-1
Formula: C21H18O11
DCQ-072
>98%,Standard References Grade
>98%,Standard References
APIIN
CAS:26544-34-3
Formula: C26H28O14
DCQ-077
>98%,Standard References Grade
>98%,Standard References
APILIMOD
CAS:541550-19-0
Trade Name: STA 5326; STA5326; STA-5326
Formula: C23H26N6O2
DC8275
>98%
Apilimod(STA 5326) is a potent IL-12/IL-23 inhibitor, IL-12 production in cultures of IFN-r/LPSstimulated human PBMCs is strongly inhibited by STA-5326 with an IC50 of 10 nM.
APILIMOD MESYLATE
CAS:870087-36-8
Trade Name: STA 5326 mesylate; STA5326 mesylate; STA-5326 mesylate
Formula: C25H34N6O8S2
DC8276
>98%
Apilimod(STA 5326) mesylate is a potent IL-12/IL-23 inhibitor, IL-12 production in cultures of IFN-r/LPSstimulated human PBMCs is strongly inhibited by STA-5326 with an IC50 of 10 nM.
APITOLISIB(GDC-0980)
CAS:1032754-93-0
Trade Name: GDC-0980; RG7422; RG-7422; GDC 0980; GNE 390.
Formula: C23H30N8O3S
DC5081
>98%
GDC-0980 (RG7422) is a potent, class I PI3K inhibitor for PI3Ka//d/? with IC50 of 5 nM/27 nM/7 nM/14 nM, respectively. Also a mTOR inhibitor with Ki of 17 nM, and highly selective versus others PIKK family kinases.
APIXABAN (BMS 562247-01)
CAS:503612-47-3
Formula: C25H25N5O4
DC5114
>98%
Apixaban is a highly selective, reversible inhibitor of Factor Xa with Ki of 0.08 nM and 0.17 nM in human and rabbit, respectively.
APOPTOSIS ACTIVATOR 2
CAS:79183-19-0
Formula: C15H9Cl2NO2
DC2066
>98%
Apoptosis Activator 2 activates caspases in a cytochrome c-dependent manner and induces apoptosis in tumor cells.
APOPTOZOLE
CAS:1054543-47-3
Formula: C33H25F6N3O3
DC10122
>98%
Apoptozole is an inhibitor of heat shock protein 70 (Hsp70; 65% inhibition at 200 M) that acts by blocking its ATPase activity.
APREMILAST
CAS:608141-41-9
Trade Name: CC 10004; CC10004; CC-10004
Formula: C22H24N2O7S
DC7063
>98%
Apremilast(CC10004) is a novel small molecule inhibitor of PDE4 with an IC50 value of 74 nM.
APREPITANT (MK-0869, L-754030)
CAS:170729-80-3
Trade Name: MK0869
Formula: C23H21F7N4O3
DC6906
>98%
Substance P antagonists (SPA).
APRICITABINE
CAS:160707-69-7
Formula: C8H11N3O3S
DC7003
>98%
Apricitabine is a novel nucleoside reverse transcriptase inhibitor for the treatment of HIV infection that is refractory to existing drugs
APROTININ
CAS:9087-70-1
Formula: C284H432N84O79S7
DC10207
>98%
Aprotinin is a serine protease inhibitor isolated from bovine lung which inhibits trypsin and chymotrypsin with Ki values of 0.06 pM and 9 nM, respectively.
APS-2-79
CAS:2002381-25-9
Trade Name: APS 2 79,APS279,APS-279
Formula: C23H21N3O3
DC10048
>98%
APS-2-79 is a novel modulator of KSR-dependent MAPK signalling,KSR2,IC50=120 nM
APS-2-79 HYDROCHLORIDE
CAS:2002381-31-7
Trade Name: APS 2 79,APS279,APS-279
Formula: C23H21N3O3.HCl
DC9808
>98%
APS-2-79 is a novel modulator of KSR-dependent MAPK signalling,KSR2,IC50=120 nM
APS-3-77 HCL
CAS:N/A
Trade Name: APS 3 77,APS377,APS-377
Formula: C24H23N3O3.HCl
DC9809
>98%
APS-3-77 is the negative binder of KSR2.
APTO-253
CAS:916151-99-0
Trade Name: LOR-253; LT-253
Formula: C22H14FN5
DC8664
>98%
APTO-253 is a novel small molecule with potent anti-tumor activity in cancer cells via induction of the gene that expresses the Krppel-like factor 4 (KLF4) master transcription factor, leading to cell cycle inhibition and programmed cell death.
APY0201
CAS:1232221-74-7
Trade Name: APY 0201 ,APY-0201 ,APY0201
Formula: C23H23N7O
DC7922
>98%
APY0201 is a potent, highly selective PIKfyve kinase inhibitor.
APY29
CAS:1216665-49-4
Trade Name: APY 29; APY-29
Formula: C17H16N8
DC7358
>98%
APY29 is an allosteric modulator of IRE1a; inhibits IRE1a autophosphorylation (IC50 = 280 nM) and activates IRE1a RNase activity.
AR 231453
CAS:733750-99-7
Trade Name: AR231453; AR-231453
Formula: C21H24FN7O5S
DC8764
>98%
AR231453 is a potent and selective small molecule agonist of GPR119 that enhances glucose-dependent insulin secretion and glucagon-like peptide 1 (GLP-1) release; Antidiabetic agent.
AR-7
CAS:80306-38-3
Trade Name: AR7,AR 7
Formula: C15H12ClNO
DC10135
>98%
AR7 is a retinoic acid receptor a (RARa) antagonist.
AR-A014418(GSK3SS,INHIBITOR,VIII)
CAS:487021-52-3
Trade Name: AR-AO 14418; AR 0133418; AR 014418; GSK 3 inhibitor
Formula: C12H12N4O4S
DC7004
>98%
AR-A014418 is a selective and effective GSK3 inhibitor with an IC 50 value of 104 +/- 27 nM; no significant inhibition on 26 other kinases.
ARA-G
CAS:38819-10-2
Formula: C10H13N5O5
DC8888
>98%
Ara-G (9--D-Arabinofuranosyl guanine) is an inducer of apoptosis, inhibitor of DNA synthesis, an antimetabolite, and antineoplastic.
ARABINOFURANOSYLCYTOSINE
CAS:147-94-4
Trade Name: N/A
Formula: C9H13N3O5
DCAPI1471
>99%
1--D-Arabinofuranosylcytosine, a cytosine analogue, inhibits DNA polymerases a, d, and e, and RNA polymerases resulting in suppression of DNA synthesis and repair. 1--D-Arabinofuranosylcytosine acts as an antimetabolic agent which is responsible for dam
ARALOSIDE V
CAS:340963-86-2
Formula: C54H88O23
DCL-029
>98%,Standard References Grade
>98%,Standard References
ARALOSIDE VII
CAS:340982-22-1
Formula: C54H88O24
DCL-030
>98%,Standard References Grade
>98%,Standard References
ARALOSIDE X
CAS:344911-90-6
Formula: C60H98O28
DCL-028
>98%,Standard References Grade
>98%,Standard References
ARBIDOL HCL
CAS:131707-23-8
Trade Name: N/A
Formula: C22H25BrN2DCAPI1051
>99%
Arbidol HCl
ARBUTIN
CAS:497-76-7
Formula: C12H16O7
DCX-007
>98%,Standard References Grade
>98%,Standard References
ARCTIGENIN
CAS:7770-78-7
Formula: C21H24O6
DCN-013
>98%,Standard References Grade
>98%,Standard References
ARCTIIN(NSC 315527)
CAS:20362-31-6
Trade Name: Arctii; NSC 315527; Arctigenin-4-glucoside
Formula: C27H34O11
DC9659
>99%
Arctiin, a plant lignan that can be extracted from the Arctium lappa (burdock) seeds, is a possible environmental endocrine disruptor compounds and have been shown to influence sex hormone metabolism as well as protein synthesis, steroid biosynthesis.
ARECAIDINE
CAS:499-04-7
Formula: C7H11NO2
DCB-084
>98%,Standard References Grade
>98%,Standard References
ARECOLINE HYDROBROMIDE
CAS:300-08-3
Formula: C8H14BrNO2
DCB-061
>98%,Standard References Grade
>98%,Standard References
ARG-GLY-ASP-SER
CAS:91037-65-9
Trade Name: RGDS peptide;Fibronectin Inhibitor
Formula: C15H27N7O8
DC9487
>98%
Arg-Gly-Asp-Ser(RGDS peptide) is an integrin binding sequence that inhibits integrin receptor function; decreases systemic inflammation via inhibition of collagen-triggered activation of leukocytes and attenuates expression of inflammatory cytokines, iNOS
ARGATROBAN
CAS:74863-84-6
Trade Name: N/A
Formula: C23H36N6DCAPI1329
>99%
Argatroban
ARGATROBAN MONOHYDRATE
CAS:141396-28-3
Trade Name: Argipidine monohydrate; Acova monohydrate
Formula: C23H38N6O6S
DC8841
>98%
Argatroban monohydrate is a direct, selective thrombin inhibitor.
ARIPIPRAZOLE
CAS:129722-12-9
Formula: C23H27Cl2N3O2
DC9147
>98%
Aripiprazole(Abilify) is a human 5-HT1A receptor partial agonist with a Ki of 4.2 nM.
ARISTOLACTAM I
CAS:13395-02-3
Formula: C17H11NO4
DCM-060
>98%,Standard References Grade
>98%,Standard References
ARISTOLOCHIC ACID
CAS:313-67-7
Formula: C17H11NO7
DCM-050
>98%,Standard References Grade
>98%,Standard References
ARISTOLOCHIC ACID B
CAS:475-80-9
Formula: C16H9NO6
DCM-071
>98%,Standard References Grade
>98%,Standard References
ARISTOLOCHIC ACID C
CAS:4849-90-5
Formula: C16H9NO7
DCM-029
>98%,Standard References Grade
>98%,Standard References
ARISTOLONE
CAS:25274-27-5
Formula: C15H22O
DCZ-268
>98%
>98%,Standard References
ARM390 HYDROCHLORIDE
CAS:209808-47-9
Trade Name: ARM 390,ARM-390,ARM390
Formula: C23H29ClN2O
DC10110
>98%
ARM390 is a non-peptidic, low-internalizing d-selective opioid receptor agonist.
ARMODAFINIL
CAS:112111-43-0
Trade Name: R-Modafinil; Nuvigil; R-(-)-Modafinil; CEP 10952; CRL 40982
Formula: C15H15NO2S
DC9421
>98%
Armodafinil(CRL 40982; CEP 10952) is an enantiopure drug consisting of just the active (-)-(R)-enantiomer of the racemic drug modafinil (Provigil).
ARN2966(2-PMAP)
CAS:102212-26-0
Trade Name: ARN-2966;ARN 2966
Formula: C12H12N2O
DC9345
>98%
ARN2966 is a potent post-transcriptional modulator of APP expression; reduces expression of APP with resultant lower production of A.
ARQ 621
CAS:1095253-39-6
Trade Name: ARQ-621,ARQ621
Formula: C28H24Cl2FN5O2
DC7820
>98%
ARQ 621 is an allosteric, and selective Eg5 mitotic motor protein inhibitor. Phase 1.
ARQ-092
CAS:1313881-70-7
Trade Name: ARQ092,ARQ 092
Formula: C27H24N6
DC9972
>98%
ARQ 092 is an oral activie, potent and selective AKT inhibitor with IC50 values: 5.0 nM (AKT1); 4.5 nM (AKT2); 16 nM (AKT3).
ARRY-380
CAS:937265-83-3
Trade Name: ARRY380; ARRY 380
Formula: C29H27N7O4S
DC8763
>98%
ARRY-380 is a potent and selective HER2 inhibitor with IC50 of 8 nM, equipotent against truncated p95-HER2, 500-fold more selective for HER2 versus EGFR.
ARRY-520 (R ENANTIOMER)
CAS:885060-08-2
Trade Name: 1,3,4-Thiadiazole-3(2H)-carboxamide, 2-(3-aminopropyl)-5-(2,5-difluorophenyl)-N-methoxy-N-methyl-2-p
Formula: C20H22F2N4O2S
DC9495
>98%
ARRY-520 R enantiomer is the R form of ARRY-520, which is a synthetic, small molecule kinesin spindle protein (KSP) inhibitor with IC50 of 6 nM._x000D_
ARS-853
CAS:1629268-00-3
Trade Name: ARS853,ARS 853
Formula: C22H29ClN4O3
DC8816
>98%
ARS-853 is a selective, covalent inhibitor of KRAS-G12C that inhibits mutant KRAS driven signaling by binding to the GDP bound oncoprotein and preventing activation.
ARS-853 INTERMEDIATE
CAS:N/A
Formula: C19H27ClN4O2
DC8854
>98%
The intermediate of ARS-853.ARS-853 is a selective, covalent inhibitor of KRAS-G12C that inhibits mutant KRAS driven signaling by binding to the GDP bound oncoprotein and preventing activation.
ARTEANNUIN
CAS:50906-56-4
Formula: C15H20O3
DCQ-085
>98%,Standard References Grade
>98%,Standard References
ARTEMETHER
CAS:71963-77-4
Formula: C16H26O5
DCH-010
>98%,Standard References Grade
>98%,Standard References
ARTEMISETIN
CAS:479-90-3
Formula: C21H22O11
DCA-011
>98%,Standard References Grade
>98%,Standard References
ARTEMISINIC ACID
CAS:80286-58-4
Formula: C15H22O2
DCQ-054
>98%,Standard References Grade
>98%,Standard References
ARTEMISININ
CAS:63968-64-9
Formula: C15H22O5
DCQ-005
>98%,Standard References Grade
>98%,Standard References
ARTESUNATE
CAS:88495-63-0
Formula: C19H28O8
DCQ-039
>98%,Standard References Grade
>98%,Standard References
ARTICAINE HCL
CAS:23964-57-0
Trade Name: N/A
Formula: C13H20N2O3S.HCl
DCAPI1125
>99%
Articaine is a dental local anesthetic which contains an additional ester group that is metabolized by estearases in blood and tissue.
ARV-771
CAS:1949837-12-0
Trade Name: ARV 771; ARV771
Formula: C49H60ClN9O7S2
DC10334
>98%
ARV-771 is a potent bromodomain and extra-terminal (BET) proteins degrader with Kd values of 4.7, 7.6, 7.6 nM against bromodomain 2, 3 and 4, respectively.
AS 602801(BENTAMAPIMOD)
CAS:848344-36-5
Trade Name: AS-602801,Bentamapimod,AS602801
Formula: C25H23N5O2S
DC8256
>98%
AS 602801(Bentamapimod) is a novel, orally active inhibitor of JNK.
AS-1413(AMONAFIDE)
CAS:69408-81-7
Formula: C16H17N3O2
DC8923
>98%
Amonafide(AS1413) produces protein-associated DNA-strand breaks through a topoisomerase II-mediated reaction, but does not produce topoisomerase I-mediated DNA cleavage.
AS-252424
CAS:900515-16-4
Trade Name: AS252424,AS 252424
Formula: C14H8FNO4S
DC3112
>98%
AS-252424 is a novel, potent and selective inhibitor of PI3K? with IC50 of 33 nM.
AS-8351
CAS:796-42-9
Trade Name: AS8351,AS 8351,NSC51355,NSC 51355,NSC-51355
Formula: C17H13N3O2
DC9840
>98%
AS 8351 induces reprogramming of human fetal lung fibroblasts into functional cardiomyocytes, in combination with CHIR 99021, A83-01, BIX 01294, SC1, Y-27632, OAC2, SU 16f and JNJ 10198409.
AS1842856
CAS:836620-48-5
Trade Name: AS 1842856,AS-1842856
Formula: C18H22FN3O3
DC10086
>98%
AS1842856 is a potent and cell-permeable Foxo1 inhibitor with an IC50 of 30 nM.
AS2034178,
CAS:1030846-42-4
Trade Name: AS-2034178,AS 2034178
Formula: C27H29FN2O3
DC8204
>98%
AS605240
CAS:648450-29-7
Trade Name: AS-605240; AS 605240
Formula: C12H7N3O2S
DC7068
>98%
AS-605240 is a potent and selective inhibitor of PI 3-kinase ? (PI3K?) (IC50 = 8 nM). AS-605240 displays 30-fold selectivity over PI3Kd and PI3K and 7.5-fold selectivity over PI3Ka.
AS703026
CAS:1236699-92-5
Trade Name: Pimasertib; MSC1936369B; AS-703026; AS 703026, Pimasertib; MSC1936369B; AS-703026; AS 703026
Formula: C15H15FIN3O3
DC7868
>98%
AS703026(Pimasertib) is a highly selective, potent, ATP non-competitive allosteric inhibitor of MEK1/2 with IC50 of 5 nM-2 M in MM cell lines.
ASC-J9
CAS:917813-54-8
Trade Name: ASC J9
Formula: C23H24O6
DC4169
99%
ASC-J9, is antitumor agent. ASC-J9 suppresses castration-resistant prostate cancer growth via degradation of full-length and splice variant androgen receptors.
ASCOMYCIN (IMMUNOMYCIN,FK-520)
CAS:11011-38-4
Trade Name: FK520,FK 520
Formula: C43H69NO12
DC1049
99%
Ascomycin is an analog of tacrolimus with immunosuppressive, neurotrophic and antifungal activities.
ASENAPINE MALEATE
CAS:85650-56-2
Trade Name: Saphris maleate; Org 5222 maleate; Org-5222 maleate; Org5222 maleate
Formula: C17H16ClNO.C4H4O4
DC8583
>98%
Novel psychopharmacologic agent. Displays antagonist activity at 5-HT, dopamine, noradrenalin and histamine receptor subtypes (pKi values are 8.60, 8.40, 10.15, 9.75, 10.46, 8.84, 9.60, 9.94, 8.85, 8.90, 8.84, 9.38, 8.95, 8.93, 8.9, 9.49, 8.91, 9.00 and 8
ASIATIC ACID
CAS:464-92-6
Formula: C30H48O5
DCJ-009
>98%,Standard References Grade
>98%,Standard References
ASIATICOSIDE
CAS:16830-15-2
Formula: C48H78O19
DCJ-001
>98%,Standard References Grade
>98%,Standard References
ASL 601(ACECAINIDE)
CAS:34118-92-8
Trade Name: Acecainide; N-acetylprocainamide, ASL 601; ASL-601; ASL601
Formula: C15H24ClN3O2
DC10592
>98%
Acecainide, also known as N-acetylprocainamide and ASL 601, is the N-acetylated metabolite of procainamide.
ASP 7663
CAS:1190217-35-6
Trade Name: ASP 7663,ASP-7663,ASP7663
Formula: C14H14FNO3
DC10558
>98%
ASP 7663 is a selective TRPA1 activator (EC50 values are ~0.5 M in human, mouse and rat).
ASP-9521
CAS:1126084-37-4
Trade Name: ASP9521; ASP-9521; ASP 9521. AKR1C3 inhibitor ; 17HSD5 inhibitor
Formula: C19H26N2O3
DC10588
>98%
ASP-9521 is a potent, selective and orally available AKR1C3 inhibitor with an IC50 of 11 nM for human AKR1C3.
ASP3026
CAS:1097917-15-1
Trade Name: ASP 3026; ASP-3026
Formula: C29H40N8O3S
DC7359
>98%
ASP3026 is a novel and selective inhibitor for ALK with IC50 of 3.5 nM.
ASPARTAME
CAS:22839-47-0
Trade Name: Nutrasweet
Formula: C14H18N2DCAPI1120
>99%
Aspartame
ASPERULOSIDE
CAS:14259-45-1
Formula: C18H22O11
DCC-077
>98%,Standard References Grade
>98%,Standard References
AST-1306
CAS:1050500-29-2
Trade Name: AST1306; AST 1306
Formula: C24H18ClFN4O2,C7H8O3S
DC7360
>98%
AST-1306 is a novel irreversible inhibitor of EGFR and ErbB2 with IC50 of 0.5 nM and 3 nM, also effective in mutation EGFR T790M/L858R, more potent to ErbB2-overexpressing cells, 3000-fold selective for ErbB family than other kinases.
ASTILBIN
CAS:29838-67-3
Formula: C21H22O11
DCL-002
>98%,Standard References Grade
>98%,Standard References
ASTRAGALIN
CAS:480-10-4
Formula: C21H20O11
DCZ-020
>98%,Standard References Grade
>98%,Standard References
ASTRAGALOSIDE
CAS:84687-42-3
Formula: C41H68O14
DCH-036
>98%,Standard References Grade
>98%,Standard References
ASTRAGALOSIDE
CAS:84676-89-1
Formula: C41H66O15
DCH-037
>98%,Standard References Grade
>98%,Standard References
ASTRAGALOSIDE A
CAS:83207-58-3
Formula: C41H65O14
DC8641
>98%
Astragaloside A, also known as astragaloside IV, is known to have diverse protective effects for the cardiovascular, immune, digestive, and nervous systems.
ASTRAGALOSIDE IV
CAS:84687-43-4
Formula: C41H68O14
DCH-013
>98%,Standard References Grade
>98%,Standard References
ASUNAPREVIR
CAS:630420-16-5
Trade Name: BMS-650032; BMS 650032; BMS650032
Formula: C35H46ClN5O9S
DC7361
>98%
Asunaprevir (BMS-650032) is a potent hepatitis C virus (HCV) NS3 protease inhibitor.
AT-101 (AT101)
CAS:866541-93-7
Trade Name: AT 101, AT101
Formula: C32H34O10
DC2015
>98%
AT-101 is a BH3 mimetic known to be a potent inhibitor of antiapoptotic Bcl-2 family members.
AT-406
CAS:1071992-99-8
Trade Name: CHEMBL2158051, AT406, AT 406, SureCN2724374, QCR-136, SM406, SM 406, AT406 (SM-406)
Formula: C32H43N5O4
DC7363
>98%
AT-406 (formerly known as SM-406) is an orally bioavailable potent IAP (inhibitor of apoptosis protein) of XIAP, cIAP1, and cIAP2 with Ki of 66.4 nM, 1.9 nM, and 5.1 nM, respectively.
AT-56
CAS:162640-98-4
Trade Name: AT 56,AT56
Formula: C25H27N5
DC7364
>98%
AT-56 is a selective, competitive, and highly bioavailable inhibitor of lipocalin-type prostaglandin D synthase (L-PGDS) with a Ki value of 75 M.
AT13148
CAS:1056901-62-2
Trade Name: AT-13148,AT 13148
Formula: C17H16ClN3O
DC7362
>98%
AT13148 is a novel, oral multi-AGC kinase inhibitor with potent pharmacodynamic and antitumor activity; AKT, p70S6K, PKA, ROCK, and SGK inhibitor.
AT7519
CAS:844442-38-2
Trade Name: AT 7519; AT-7519
Formula: C16H17Cl2N5O2
DC9676
>98%
AT7519 is a multi-CDK inhibitor for CDK1, 2, 4, 6 and 9 with IC50 of 10-210 nM; less potent to CDK3 and little active to CDK7.
AT7519 (TRIFLUOROACETATE)
CAS:1431697-85-6
Trade Name: AT 7519 trifluoroacetate;AT-7519 trifluoroacetate
Formula: C18H18Cl2F3N5O4
DC9395
>98%
AT7519 trifluoroacetate is a multi-CDK inhibitor for CDK1, 2, 4, 6 and 9 with IC50 of 10-210 nM; less potent to CDK3 and little active to CDK7.
AT7519 HCL
CAS:902135-91-5
Trade Name: AT7519, AT-7519
Formula: C16H17Cl2N5O2
DC1025
99%
AT7519 is a novel multi-CDK inhibitor for CDK1/cyclin B, CDK2/Cyclin A, CDK3/Cyclin E, CDK4/Cyclin D1, CDK5/p35 and CDK6/Cyclin D3 with IC50 of 210 nM, 47 nM, 360 nM, 100 nM, 13 nM and 170 nM, respectively.
AT7867
CAS:857531-00-1
Trade Name: AT-7867;AT 7867
Formula: C20H20ClN3
DC9335
>98%
AT7867 is a potent ATP-competitive inhibitor of Akt1/2/3 and p70S6K/PKA with IC50 of 32 nM/17 nM/47 nM and 85 nM/20 nM, respectively; little activity outside the AGC kinase family._x000D_
AT7867 (DIHYDROCHLORIDE)
CAS:1431697-86-7
Trade Name: AT-7867 dihydrochloride;AT 7867 dihydrochloride
Formula: C20H22Cl3N3
DC9336
>98%
AT7867 Hcl is a potent ATP-competitive inhibitor of Akt1/2/3 and p70S6K/PKA with IC50 of 32 nM/17 nM/47 nM and 85 nM/20 nM, respectively; little activity outside the AGC kinase family._x000D_
AT9283
CAS:896466-04-9
Trade Name: AT-9283; AT 9283
Formula: C19H23N7O2
DC7070
>98%
AT9283 is a small molecule a multi-targeted inhibitor with of 4, 1.2, 1.1 and approximate 3 nM for Bcr-Abl(T3151), Jak2 and Jak3, aurora A and B, respectively.
ATAZANAVIR
CAS:198904-31-3
Trade Name: BMS-232632-05, Reyataz,BMS23263205
Formula: C38H52N6O7.H2SO4
DC3150
>98%
Atazanavir is a HIV protease inhibitor with Ki of 2.66 nM.
ATAZANAVIR (SULFATE)
CAS:229975-97-7
Trade Name: BMS 232632 sulfate;BMS-232632 sulfate;BMS232632 sulfate
Formula: C38H54N6O11S
DC9480
>98%
Atazanavir sulfate is a sulfate salt form of atazanavir that is an highly potent HIV-1 protease inhibitor._x000D_
ATB-346
CAS:1226895-20-0
Trade Name: ATB346;ATB 346
Formula: C21H19NO3S
DC7365
>98%
ATB-346 is a novel hydrogen sulphide-releasing derivative of naproxen with markedly reduced toxicity.
ATENOLOL
CAS:29122-68-7
Formula: C14H22N2O3
DC9020
>98%
Atenolol is a selective 1 receptor antagonist.
ATGLISTATIN
CAS:1469924-27-3
Formula: C17H21N3O
DC7366
>98%
Atglistatin is a highly potent, selective and competitive inhibitor of adipose triglyceride lipase (ATGL) with an IC50 of ~0.7 M for inhibition of lipolysis in vitro, but no toxicity up to a concentration of 50 M.
ATI-2341
CAS:1337878-62-2
Formula: C104H178N26O25S2
DC9878
>98%
ATI-2341, pepducin targeting the C-X-C chemokine receptor type 4 (CXCR4), is an allosteric agonist activating the inhibitory heterotrimeric G protein (Gi) to promote inhibition of cAMP production and induce calcium mobilization.
ATIPAMEZOLE
CAS:104054-27-5
Formula: C14H16N2
DC8925
>98%
Atipamezole(MPV1248) is an alpha-adrenoceptor antagonist with high affinity and selectivity for the alpha 2-receptor.
ATIPAMEZOLE HCL
CAS:104075-48-1
Formula: C14H17ClN2
DC8998
>98%
Atipamezole Hcl(MPV1248 Hcl) is an alpha-adrenoceptor antagonist with high affinity and selectivity for the alpha 2-receptor.
ATN-161
CAS:262438-43-7
Trade Name: ATN161; ATN 161
Formula: C23H35N9O8S
DC7709
>98%
ATN-161 (Ac-PHSCN-NH2) is a five -amino-acid peptide derived from the synergy region of fibronectin; a beta integrin antagonist with antitumor activity.
ATOCALCITOL
CAS:302904-82-1
Trade Name: N/A
Formula: C32H46O4
DCAPI1522
>99%
Atocalcitol
ATOMOXETINE HCL
CAS:82248-59-7
Formula: C17H22ClNO
DC9034
>98%
Atomoxetine Hcl(LY 139603; Tomoxetine Hcl) is a potent and selective noradrenalin re-uptake inhibitor (Ki values are 5, 77 and 1451 nM for inhibition of radioligand binding to human NET, SERT and DAT respectively).
ATOPAXAR(E5555)
CAS:751475-53-3
Formula: C29H38FN3O5
DC9198
>98%
ATORVASTATIN CALCIUM
CAS:134523-03-8
Trade Name: N/A
Formula: C33H34FN2O50.5 Ca1.5 H2O
DCAPI1442
>99%
Atorvastatin Calcium
ATOVAQUONE(ATAVAQUONE)
CAS:95233-18-4
Trade Name: N/A
Formula: C22H19ClO3
DCAPI1390
>99%
Atovaquone is a medication used to treat or prevent for pneumocystis pneumonia, toxoplasmosis, malaria, and babesia.
ATP (ADENOSINE-TRIPHOSPHATE)
CAS:987-65-5
Trade Name: N/A
Formula: C10H14N5DCAPI1401
>99%
ATP (Adenosine-Triphosphate)
ATRACTYLENOLIDE 1
CAS:73069-13-3
Formula: C15H18O2
DCB-033
>98%,Standard References Grade
>98%,Standard References
ATRACTYLENOLIDE II
CAS:73069-14-4
Formula: C15H20O2
DCB-034
>98%,Standard References Grade
>98%,Standard References
ATRACTYLENOLIDE III
CAS:73030-71-4
Formula: C15H20O3
DCB-035
>98%,Standard References Grade
>98%,Standard References
ATRACTYLODIN
CAS:55290-63-6
Formula: C13H10O
DCC-022
>98%,Standard References Grade
>98%,Standard References
ATRACTYLON
CAS:6989-21-5
Formula: C15H20O
DCZ-188
>98%
>98%,Standard References
ATRACTYLOSIDE A
CAS:126054-77-1
Formula: C21H36O10
DCC-052
>98%,Standard References Grade
>98%,Standard References
ATRACURIUM BESYLATE
CAS:64228-81-5
Trade Name: N/A
Formula: C53H72N2DCAPI1288
>99%
Atracurium besylate
ATRASENTAN HYDROCHLORIDE
CAS:195733-43-8
Trade Name: ABT-627; ABT627; ABT 627; Abbott 147627
Formula: C29H39ClN2O5
DC10018
>98%
Atrasentan Hcl(A-147627) is an endothelin antagonist receptor (IC50=0.0551 nM, ETA) being developed for the treatment of prostate cancer.
ATROPINE SULFATE MONOHYDRATE
CAS:5908-99-6
Formula: C34H50N2O11S
DCZ-260
>98%
>98%,Standard References
AU1235
CAS:1338780-86-1
Trade Name: AU1235,AU-1235,AU 1235
Formula: C17H19F3N2O
DC10552
>98%
AU1235 is an adamantyl urea inhibitor of Mycobacterium tuberculosis.
AUCUBIN
CAS:479-98-1
Formula: C15H22O9
DCT-016
>98%,Standard References Grade
>98%,Standard References
AURANTIO-OBTUSIN
CAS:67979-25-3
Formula: C17H14O7
DCC-007
>98%,Standard References Grade
>98%,Standard References
AURISTATIN E
CAS:160800-57-7
Trade Name: Auristatin E
Formula: C40H69N6O7
DC10138
>98%
Auristatin E is a cytotoxic tubulin modifier with potent and selective antitumor activity; MMAE analog and cytotoxin in Antibody-drug conjugates.
AURORA A INHIBITOR I
CAS:1158838-45-9
Formula: C31H31ClFN7O2
DC7964
>98%
Aurora A inhibitor I is a selective Aurora A inhibitor (Aurora A: IC50=0.0034 M; Aurora B IC50=3.4 M), (B/A ratio=1000).
AUTEN-99
CAS:1049780-58-6
Trade Name: Auten-99,Auten 99,Auten99
Formula: C17H15BrN2S
DC10548
>98%
Auten-99 is a novel inhibitor of the myotubularin phosphatase Jumpy (also called MTMR14), acrossing the blood-brain barrier and exerting potent neuroprotective effects.
AUTOPHINIB
CAS:1644443-47-9
Formula: C14H11ClN6O3
DC10461
>98%
Autophinib is a novel potent autophagy inhibitor, inhibiting autophagy induced by starvation or Rapamycin by targeting the lipid kinase VPS34.
AV-412(MP-412)
CAS:451492-95-8
Trade Name: AV-412,MP-412,AV 412,MP 412,AV412,MP412
Formula: C27H28ClFN6O
DC8253
>98%
AV-412(MP-412) is a potent dual inhibitor of EGFR and ErbB2(IC50=19 nM) tyrosine kinases, including the mutant EGFR(L858R IC50=0.51 nM, T790M IC50=0.79 nM); inhibits autophosphorylation of EGFR and ErbB2 with IC(50) of 43 and 282 nM, respectively.
AVAGACESTAT (BMS-708163)
CAS:1146699-66-2
Trade Name: BMS708163,BMS 708163
Formula: C20H17ClF4N4O4S
DC3114
>98%
BMS-708163 is a potent, selective ?-secretase inhibitor of A40 and A42 with IC50 of 0.3 nM and 0.27 nM, respectively.
AVANAFIL(TA-1790)
CAS:330784-47-9
Formula: C23H26ClN7O3
DC8799
>98%
Avanafil(TA-1790) is a potent and highly selective phosphodiesterase-5(PDE-5) inhibitor(IC50=5.2 nM) for erectile dysfunction; lower selectivity against PDE1, PDE6, and PDE11.
AVASIMIBE (CI-1011)
CAS:166518-60-1
Trade Name: CI1011
Formula: C29H43NO4S
DC1094
>98%
Avasimibe inhibits ACAT and CYP2C9 with IC50 of 3.3 M and 2.9 M, respectively.
AVIBACTAM SODIUM
CAS:1192491-61-4
Trade Name: NXL-104,NXL 104,NXL104
Formula: C7H10N3NaO6S
DC8351
>98%
Avibactam sodium(NXL-104) is a non--lactam -lactamase inhibitor antibiotic.
AVIBACTAM SODIUM HYDRATE
Formula: C7H12N3NaO7S
DC8709
>98%
Avibactam sodium hydrate is a non--lactam -lactamase inhibitor antibiotic.
AVICULARIN(GUAJAVARIN)
CAS:572-30-5;22255-13-6
Formula: C20H18O11
DCB-049
>98%,Standard References Grade
>98%,Standard References
AVIPTADIL
CAS:40077-57-4
Trade Name: Vasoactive Intestinal Peptide (human, rat, mouse, rabbit, canine, porcine)
Formula: C147H238N44O42S
DC10325
>98%
Aviptadil (INN) is an analog of vasoactive intestinal polypeptide (VIP) for the treatment of erectile dysfunction.
AVITINIB FREE BASE
CAS:1557267-42-1
Trade Name: AC0010MA; AC-0010MA; AC 0010MA; AC0010; AC-0010; AC 0010.
Formula: C26H28FN7O2
DC10009
>98%
Avitinib is an orally available, irreversible, epidermal growth factor receptor (EGFR) mutant-selective inhibitor, with potential antineoplastic activity.
AVITINIB MALEATE
CAS:1557268-88-8
Trade Name: AC0010MA; AC-0010MA; AC 0010MA; AC0010; AC-0010; AC 0010.
Formula: C30H30FN7O6
DC10008
>98%
Avitinib is an orally available, irreversible, epidermal growth factor receptor (EGFR) mutant-selective inhibitor, with potential antineoplastic activity.
AVL-292
CAS:1202757-89-8
Trade Name: CC-292; AVL292; AVL-292; AVL 292
Formula: C22H22FN5O3
DC5014
>98%
AVL-292 is a covalent, highly selective, orally active small molecule inhibitor of Btk currently being evaluated in a Phase 1b clinical trial in relapsed.
AVN 944
CAS:297730-17-7
Trade Name: AVN-944,AVN 944,AVN944,VX 944,VX944
Formula: C25H27N5O5
DC8843
>98%
AVN-944(VX-944) is a selective, noncompetitive inhibitor of the enzyme directed against human IMPDH with Ki of 6-10 nM for IMPDH1/IMPDH2.
AVN944
CAS:501345-02-4
Trade Name: VX 944, AVN-944;
Formula: C24H25N5O5
DC8565
>98%
AVN-944(VX-944) is a selective, noncompetitive inhibitor of the enzyme directed against human IMPDH with Ki of 6-10 nM for IMPDH1/IMPDH2.
AVOBENZONE(PARSOL 1789)
CAS:70356-09-1
Trade Name: Eusolex 9020, Escalol 517, Parsol 1789
Formula: C20H22O3
DCAPI1313
>99%
Avobenzone(Parsol 1789)
AVOSENTAN
CAS:290815-26-8
Trade Name: Ro 67-0565; SPP-301
Formula: C23H21N5O5S
DC9436
>98%
Avosentan(Ro 67-0565; SPP-301) is a potent, selective endothelin receptor(ETA receptor) antagonist._x000D_
AWD 131-138(IMEPITOIN)
CAS:188116-07-6
Trade Name: Imepitoin; AWD131-138
Formula: C13H14ClN3O2
DC7071
>98%
AWD 131-138(Imepitoin) is a new low-affinity partial benzodiazepine receptor agonist with potent anticonvulsant and anxiolytic properties in rodent models.
AX-024
CAS:1704801-24-0
Trade Name: AX-024,AX024,AX 024
Formula: C21H23FNO2Cl
DC10545
>98%
AX-024 is the first-in-class inhibitor of T cell receptor (TCR); AX-024 is an orally available inhibitor of the TCR-Nck interaction that selectively inhibits TCR-triggered T cell activation (IC50 value 1 nM).
AX15836
CAS:N/A
Trade Name: AX15836; AX 15836; AX-15836
Formula: C32H40N8O5S
DC10649
>98%
AX15836 is a highly potent and selective ERK5 inhibitor.
AX20017
CAS:329221-38-7
Trade Name: AX-20017; AX 20017
Formula: C13H16N2O2S
DC10412
>98%
AX20017 is a small-molecule protein kinase G (PknG) inhibitor with an IC50 of 0.39 M.
AXITINIB
CAS:319460-85-0
Trade Name: AG-013736,AG 013736,AG013736
Formula: C43H69NO12
DCAPI1524
>99%
Axitinib is a non-selective receptor kinase inhibitor of Flt and Flk proteins. This compound also inhibits VEGFR-1, VEGFR-2, VEGFR-3, PDGFR- and c-KIT with IC50 of 0.1 nM, 0.2 nM, 0.1-0.3 nM, 1.6 nM and 1.7 nM, respectively. Axitinib is studied as an ant
AZ-33(AZ33)
CAS:1370290-34-8
Trade Name: AZ-33,AZ33,AZ 33
Formula: C25H27N3O6S
DC9667
>98%
AZ-33 is a inhibitor of LDH-A with an IC50 of 0.5 M.
AZ-6102
CAS:1645286-75-4
Trade Name: AZ-6102,AZ6102,AZ 6102
Formula: C25H28N6O
DC7926
>98%
AZ6102 is a potent TNKS1/2 inhibitor that has 100-fold selectivity against other PARP family enzymes and shows 5 nM Wnt pathway inhibition in DLD-1 cells.
AZ-628
CAS:878739-06-1
Trade Name: AZ-628,cas 878739-06-1,AZ 628,AZ628
Formula: C27H25N5O2
DC7370
>98%
AZ-7371(DPRE1-IN-1)
CAS:1494675-86-3
Trade Name: AZ7371,AZ 7371
Formula: C18H21N5O3
DC8842
>98%
AZ-7371(DprE1-IN-1) is a novel non-covalent DprE1 inhibitor.
AZ-960
CAS:905586-69-8
Trade Name: AZ960,AZ 960
Formula: C18H16F2N6
DC7367
>98%
AZ 960 is a novel ATP competitive JAK2 inhibitor with IC50 and Ki of <3 nM and 0.45 nM, 3-fold selectivity of AZ960 for JAK2 over JAK3.
AZ191
CAS:1594092-37-1
Trade Name: AZ-191,AZ 191
Formula: C24H27N7O
DC7746
>98%
AZ191 is a potent and selective DYRK1B inhibitor with IC50 of 17 nM, about 5- and 110-fold selectivity over DYRK1A and DYRK2, respectively.
AZ20
CAS:1233339-22-4
Trade Name: AZ-20; AZ 20,
Formula: C21H24N4O3S
DC7906
>98%
AZ20 is a novel potent and selective inhibitor of ATR kinase with IC50 of 5 nM, 8-fold selectivity over mTOR.
AZ3146
CAS:1124329-14-1
Trade Name: AZ 3146; AZ-3146
Formula: C24H32N6O3
DC7072
>98%
AZ3146 is a potent and selective monopolar spindle 1 (Mps1) kinase inhibitor (IC50 = 35 nM); less potent to FAK, JNK1, JNK2, and Kit.
AZ505
CAS:1035227-43-0
Trade Name: AZ-505,AZ 505
Formula: C29H38Cl2N4O4
DC8537
>98%
AZ505 is a potent and highly selective inhibitor of the oncogenic protein SMYD2(IC50=0.12 uM) with potential anticancer activity, >600 fold than SMYD3(IC50>83.3 uM); DOT1L(IC50>83.3 uM);EZH2(IC50>83.3 uM).
AZ5104
CAS:1421373-98-9
Trade Name: AZ-5104,AZ 5104
Formula: C27H31N7O2
DC8052
>98%
AZ5104 is an active circulating metabolite of AZD9291.
AZ9482
CAS:1825345-33-2
Trade Name: AZ 9482,AZ-9482
Formula: C26H22N6O2
DC10056
>98%
AZ9482, a potent and selective PARP inhibitor featuring an amide linkage to a 2-piperazinyl-3-cyano-pyridine.
AZAPERONE
CAS:1649-18-9
Trade Name: Fluoperidol
Formula: C19H22FN3O
DC8713
>98%
Azaperone acts as a dopamine antagonist but also has some antihistaminic and anticholinergic properties. Azaperone is a pyridinylpiperazine and butyrophenone neuroleptic drugwith sedative and antiemetic effects, which is used mainly as a tranquilizer in
AZAPHEN (DIHYDROCHLORIDE MONOHYDRATE)
CAS:63302-99-8
Trade Name: Azafen dihydrochloride monohydrate;Pipofezin dihydrochloride monohydrate;Pipofezine dihydrochloride
Formula: C16H23Cl2N5O2
DC9629
>98%
Pipofezine(Azafen or Azaphen) is a potent inhibitor of the reuptake of serotonin.
AZASETRON HCL
CAS:123040-16-4
Trade Name: N/A
Formula: C17H21Cl2N3O3
DCAPI1427
>99%
Azasetron Hydrochloride is a 5-HT3 receptor antagonist which is used as an anti-emetic.
AZATADINE (DIMALEATE)
CAS:3978-86-7
Trade Name: Azatadine maleate;Optimine;Zadine
Formula: C28H30N2O8
DC9469
>98%
Azatadine dimaleate is an histamine and cholinergic inhibitor with IC50 of 6.5 nM and 10 nM, respectively._x000D_
AZATHIOPRINE (AZASAN, IMURAN)
CAS:446-86-6
Trade Name: Azasan, Imuran, Azamun, BW-57-322, NSC-39084
Formula: C9H7N7O2S
DCAPI1182
>99%
Azathioprine (Azasan, Imuran)
AZD 7762
CAS:860352-01-8
Trade Name: AZD7762; AZD-7762
Formula: C17H19FN4O2S.HCl
DC7076
>98%
AZD7762 is a potent and selective inhibitor of Chk1 with IC50 of 5 nM; equally potent against Chk2 and less potent against CAM, Yes, Fyn, Lyn, Hck and Lck.
AZD-0156
CAS:1821428-35-6
Trade Name: AZ0156,AZ 0156
Formula: C26H31N5O3
DC9309
>98%
AZD-0156 is an orally bioavailable ataxia telangiectasia mutated (ATM) kinase inhibitor, with potential chemo-/radio-sensitizing and antineoplastic activities.
AZD-2281 (OLAPARIB)
CAS:763113-22-0
Trade Name: AZD2281; KU-0059436; KU0059436; AZD-2281; KU0059436; AZD 2281
Formula: C24H23FN4O3
DC4110
>99%
Olaparib (AZD2281, KU0059436) is a selective inhibitor of PARP1 and PARP2 with IC50 of 5 nM and 1 nM, respectively.
AZD-26
CAS:1357158-81-6
Trade Name: AZD-26,AZD 26,AZD26
Formula: C22H21N3O
DC7748
>98%
AZD-26 is an inhibitor of AKT. AZD-26 inhibits the phosphorylation of Thr308 on AKT in BT474 cells with an IC50 of 422 nM.
AZD-3463
CAS:1356962-20-3
Trade Name: AZD3463; AZD 3463; ALK/IGF1R inhibitor
Formula: C24H25ClN6O
DC7074
>98%
AZD-3463 is an ALK/IGF1R inhibitor which overcomes multiple mechanisms of acquired resistance to crizotinib.
AZD-3759
CAS:1626387-80-1
Trade Name: AZD-3759,AZD 3759,,AZD3759
Formula: C22H23ClFN5O3
DC8472
>98%
AZD3759 is an orally available inhibitor of the epidermal growth factor receptor (EGFR), with potential antineoplastic activity.
AZD-3965
CAS:1448671-31-5
Trade Name: AZD-3965,AZD3965,AZD 3965
Formula: C21H24F3N5O5S
DC9263
>98%
AZD3965 is a selective inhibitor of monocarboxylate transporter 1 (MCT1) with a binding affinity of 1.6 nM, is 6 fold selective over MCT2 and does not inhibit MCT4 at 10 M.
AZD-3988
CAS:892489-52-0
Trade Name: AZD-3988, AZD3988, AZD 3988
Formula: C23H22F2N4O4
DC8060
>98%
AZD-3988 is a potent and selective diacylglycerol acyltransferase (DGAT-1) inhibitor (IC50 = 0.6 nM).
AZD-5597
CAS:924641-59-8
Trade Name: AZD5597,AZD 5597,AZD-5597
Formula: C23H28FN7O
DC7075
>98%
AZD-5597 is potent CDK inhibitor with in vitro anti-proliferative effects against a range of cancer cell lines.
AZD-6738
CAS:1352226-88-0
Trade Name: AZD-6738,AZD 6738,AZD6738
Formula: C20H24N6O2S
DC8468
>98%
AZD6738 is an orally active, and selective ATR kinase inhibitor with IC50 of 1 nM. Phase 1/2.
AZD-7547
CAS:252017-04-2
Trade Name: AZD 7547,AZD7547
Formula: C19H18ClF3N2O5S
DC8837
>98%
AZD7545 is a novel, selective small-molecule inhibitor of PDHK2 (PDH kinase2) with an IC50 of 36.8 nM and 6.4 nM for PDHK1 and PDHK2 respectively.
AZD-8055
CAS:1009298-09-2
Trade Name: AZD-8055; AZD8055; AZD 8055.
Formula: C25H31N5O4
DC5084
>98%
AZD-8055 is a potent, selective, and orally bioavailable ATP-competitive mTOR kinase inhibitor with an IC50 of 0.8 nM.
AZD-8931(SAPITINIB)
CAS:848942-61-0
Trade Name: AZD-8931,AZD8931,AZD 8931
Formula: C23H25ClFN5O3
DC7078
>98%
Sapitinib(AZD8931) is a reversible, ATP competitive inhibitor of EGFR, ErbB2 and ErbB3 with IC50 of 4 nM, 3 nM and 4 nM respectively.
AZD-9291 MESYLATE (OSIMERTINIB,MERELETINIB)
CAS:1421373-66-1
Trade Name: Mereletinib mesylate; EGFR inhibitor; AZD9291 mesylate; AZD 9291 mesylate,Tagrisso
Formula: C29H37N7O5S
DC8462
>99%
AZD-9291 is a potent and selective mutated forms EGFR inhibitor(Exon 19 deletion EGFR IC50=12.92 nM, L858R/T790M EGFR IC50= 11.44 nM, wild type EGFR IC50= 493.8 nM).
AZD0865(LINAPRAZAN)
CAS:847574-05-4
Trade Name: AZD0865,AZD-0865,AZD 0865
Formula: C21H26N4O2
DC10534
>98%
AZD0865 is a potent agent that inhibits gastric H(+),K(+)-ATPase activity and acid formation in vitro, with a fast onset of effect.
AZD1080
CAS:612487-72-6
Trade Name: AZD 1080,AZD-1080
Formula: C19H18N4O2
DC5054
>98%
AZD1080 is a selective, orally active, brain permeable GSK3 inhibitor, inhibits human GSK3a and GSK3 with Ki of 6.9 nM and 31 nM, respectively, shows >14-fold selectivity against CDK2, CDK5, CDK1 and Erk2.
AZD1152 (BARASERTIB)
CAS:722543-31-9
Trade Name: Barasertib; AZD-1152; AZD 1152
Formula: C26H31FN7O6P
DC7060
>98%
AZD1152 (barasertib), pro-drug of barasertib-hQPA, is a selective Aurora B kinase inhibitor, AZD1152 inhibited the proliferation various types of human leukemia cells with an IC50 ranging from 3 nM to 40 nM.
AZD1208
CAS:1204144-28-4
Trade Name: AZD-1208;, AZD1208;, AZD 1208.
Formula: C21H21N3O2S
DC5012
>98%
AZD1208 is orally available, small molecule inhibitor of PIM kinases with potential antineoplastic activity.
AZD1283
CAS:919351-41-0
Trade Name: AZD-1283,AZD 1283
Formula: C23H26N4O5S
DC9731
>98%
AZD1283 is a potent antagonist of the P2Y12 receptor with EC50 of 3.0 ug/kg/min, TI >10; with binding IC50 of 11 nM.
AZD1480
CAS:935666-88-9
Trade Name: AZD 1480,AZD-1480
Formula: C14H14ClFN8
DC5032
>98%
AZD1480 is a novel ATP-competitive JAK2 inhibitor with IC50 of 0.26 nM, selectivity against JAK3 and Tyk2, and to a smaller extent against JAK1. Phase 1/2.
AZD1981
CAS:802904-66-1
Formula: C19H17ClN2O3S
DC7572
>98%
AZD1981 is a potent, selective CRTh2 (DP2) receptor antagonist with IC50 of 4 nM, showing >1000-fold selectivity over more than 340 other enzymes and receptors, including DP1
AZD2014
CAS:1009298-59-2
Trade Name: AZD 2014; AZD-2014
Formula: C25H30N6O3
DC7073
>98%
AZD2014 is a novel mTOR inhibitor with IC50 of 2.8 nM; highly selective against multiple PI3K isoforms (a//?/d).
AZD2461
CAS:1174043-16-3
Trade Name: AZD-2461
Formula: C22H22FN3O3
DC1037
>98%
AZD2461 is a novel PARP inhibitor with potential to bypass Pgp-mediated resistance to Olaparib.
AZD2858
CAS:486424-20-8
Trade Name: AZD-2858,AZD 2858
Formula: C21H23N7O3S
DC6302
99%
AZD2858 is a selective GSK-3 inhibitor with an IC50 of 68 nM, activating Wnt signaling, increases bone mass in rats.
AZD2932
CAS:883986-34-3
Trade Name: AZD 2932, AZD-2932, AGN-PC-00AQ5T,AZD2932
Formula: C24H25N5O4
DC7799
>98%
AZD-2932 is a high affinity inhibitor of VEFGR-2 and PDGFR.
AZD3264
CAS:1609281-86-8
Trade Name: AZD-3264; AZD 3264
Formula: C21H23N5O4S
DC8658
>98%
AZD 3264 is an IkB-kinase IKK2 Inhibitor, IKK2 has been identified as one of the novel pathways to treat inflammatory conditions such as asthma, chronic pulmonary obstructive disorder (COPD) and rheumatoid arthritis.
AZD3514
CAS:1240299-33-5
Trade Name: AZD 3514, AZD-3514
Formula: C25H32F3N7O2
DC5013
>98%
AZD3514 is a potent and oral androgen receptor with Ki of 2.2 M and has ability of reducing AR protein expression.
AZD3839
CAS:1227163-84-9
Trade Name: AZD3839,AZD-3839,AZD 3839
Formula: C24H16F3N5
DC8400
>98%
AZD3839 is a potent and selective BACE1 inhibitor with Ki of 26.1 nM, about 14-fold selectivity over BACE2. Phase 1.
AZD4547
CAS:1035270-39-3
Trade Name: AZD-4547, AZD 4547
Formula: C26H33N5O3
DC1075
>98%
AZD4547 is a novel selective FGFR inhibitor targeting FGFR1, FGFR2, and FGFR3 with IC50 of of 0.2 nM, 2.5 nM, and 1.8 nM, respectively.
AZD5153 6-HYDROXY-2-NAPHTHOIC ACID
CAS:1869912-40-2
Trade Name: AZD 5153 6-Hydroxy-2-naphthoic acid; AZD-5153 6-Hydroxy-2-naphthoic acid
Formula: C36H41N7O6
DC10288
>98%
AZD5153 6-Hydroxy-2-naphthoic acid is the 6-Hydroxy-2-naphthoic acid of AZD5153. AZD5153 is a potent, selective, and orally available BET/BRD4 bromodomain inhibitor; disrupts BRD4 with an IC50 of 1.7 nM.
AZD5363
CAS:1143532-39-1
Trade Name: AZD-5363; AZD 5363
Formula: C21H25ClN6O2
DC7368
>98%
AZD5363, a novel pyrrolopyrimidine-derived compound, inhibits all AKT isoforms (IC50 <10 nM).
AZD5438
CAS:602306-29-6
Trade Name: AZD 5438; AZD5438
Formula: C18H21N5O2S
DC7369
>98%
AZD5438 is a potent inhibitor of CDK1/2/9 with IC50 of 16 nM/6 nM/20 nM. It is less potent to CDK5/6.
AZD5582
CAS:1258392-53-8
Trade Name: AZD5582,AZD-5582,AZD 5582
Formula: C58H78N8O8
DC8232
>98%
AZD5582 is a novel class of dimeric Smac mimetics as potent IAP antagonist; binds potently to the BIR3 domains of cIAP1, cIAP2, and XIAP (IC50 = 15, 21, and 15 nM, respectively).
AZD6244 (SELUMETINIB,ARRY-142886)
CAS:606143-52-6
Trade Name: ARRY-142886, Selumetinib,AZD-6244,ARRY142886
Formula: C17H15BrClFN4O3
DC1069
>98%
AZD6244 (Selumetinib, ARRY-142886) is highly potent to inhibit MEK1 with IC50 of 14 nM.
AZD6482
CAS:1173900-33-8
Trade Name: AZD-6482, AZD 6482
Formula: C22H24N4O4
DC8004
>98%
AZD6482 is a PI3K inhibitor with IC50 of 10 nM, 8-, 87- and 109-fold more selective to PI3K than PI3Kd, PI3Ka and PI3K?.
AZD8186
CAS:1627494-13-6
Trade Name: AZD8186,AZD-8186,AZD 8186
Formula: C24H25F2N3O4
DC8380
>98%
AZD8186 is an inhibitor of the beta isoform of phosphoinositide-3 kinase (PI3K), with potential antineoplastic activity.
AZD8330(ARRY-424704; ARRY-704)
CAS:869357-68-6
Trade Name: ARRY-424704; ARRY-704; AZD-8330; ARRY424704; ARRY704; AZD 8330
Formula: C16H17FIN3O4
DC7077
>98%
AZD8330(ARRY-424704; ARRY-704) is a novel, selective, non-ATP competitive MEK 1/2 inhibitor with IC50 of 7 nM.
AZD8797
CAS:911715-90-7
Trade Name: AZD 8797; AZD-8797
Formula: C19H25N5OS2
DC10202
>98%
AZD8797 is an allosteric non-competitive modulator of the human CX3CR1 receptor; antagonizes CX3CL1 with IC50 values of 6 and 300 nM in B-lymphocyte cell line and human whole blood, respectively.
AZD8835
CAS:1620576-64-8
Formula: C22H31N9O3
DC9879
>98%
AZD8835 ia a novel mixed inhibitor of PI3Ka and PI3Kd with IC50 of 6.2 nM and 5.7 nM, respectively, also with selectivity against PI3K (IC50=431 nM) and PI3K? (IC50=90 nM).
AZD9056 HYDROCHLORIDE
CAS:345303-91-5
Trade Name: AZD-9056 hydrochloride; AZD 9056 hydrochloride
Formula: C24H36Cl2N2O2
DC10425
>98%
AZD9056 is a selective orally active inhibitor of P2X7 which plays a significant role in inflammation and pain-causing diseases.
AZD9362
CAS:1905412-80-7
Trade Name: AZD 9362;AZD-9362
Formula: C24H27ClN8O2
DC10112
>98%
AZD-9362 is dual IGF-IR/InsR inhibitor.
AZD9496
CAS:1639042-08-2
Trade Name: AZD-9496,AZD 9496
Formula: C25H25F3N2O2
DC9268
>98%
AZD9496 is a potent and orally bioavailable selective estrogen receptor downregulator(Ki=0.7 nM) and antagonist.
AZELAIC ACID
CAS:123-99-9
Trade Name: Azelaic acid
Formula: C9H16O4
DC10245
>98%
Azelaic acid is an organic compound produced by the ozonolysis of oleic acid and possesses antibacterial, keratolytic, comedolytic, and anti-oxidant activity.
AZELASTINE HCL
CAS:79307-93-0
Formula: C22H25Cl2N3O
DC9130
>98%
Azelastine HCl is a potent, second-generation, selective, histamine antagonist.
AZELIRAGON(PF-04494700,TTP488)
CAS:603148-36-3
Trade Name: PF04494700,TTP-488,PF 04494700,TTP 488,PF-04494700,TTP488
Formula: C32H38ClN3O2
DC8338
>98%
Azeliragon is an oral, small-molecule inhibitor of RAGE.
AZELNIDIPINE
CAS:123524-52-7
Formula: C33H34N4O6
DCAPI1590
>98%
Azelnidipine is an L-type calcium channel protein inhibitor
AZIDOTHYMIDINE (AZT)
CAS:30516-87-1
Formula: C10H13N5O4
DC9864
>98%
Selective reverse transcriptase inhibitor. Exhibits 100-fold selectivity for HIV reverse transcriptase over DNA polymerase a.
AZILSARTAN
CAS:147403-03-0
Trade Name: N/A
Formula: C25H20N4O5
DCAPI1469
>99%
Azilsartan(TAK-536) is a specific and potent angiotensin II type 1 receptor antagonist with IC50 of 2.6 nM.
AZILSARTAN KAMEDOXOMIL
CAS:863031-24-7
Formula: C30H23N4O8.K
DC4210
>98%
Azilsartan medoxomil is an angiotensin II receptor antagonist indicated for the treatment of mild to moderate essential hypertension.
AZILSARTAN MEDOXOMIL
CAS:863031-21-4
Formula: C30H24N4O8
DC8901
>98%
Azilsartan medoxomil(TAK 491) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension.
AZIMILIDE (DIHYDROCHLORIDE)
CAS:149888-94-8
Trade Name: NE-10064 Dihydrochloride
Formula: C23H30Cl3N5O3
DC9596
>98%
Azimilide 2Hcl(NE-10064 2Hcl) is a class III antiarrhythmic compound, inhibits I(Ks) and I(Kr) in guinea-pig cardiac myocytes and I(Ks) (minK) channels expressed in Xenopus oocytes._x000D_
AZITHROMYCIN(ZITHROMAX)
CAS:83905-01-5
Trade Name: N/A
Formula: C38H72N2DCAPI1362
>99%
Azithromycin (Zithromax)
AZM475271
CAS:476159-98-5
Trade Name: AZM-475271;M475271;M-475271
Formula: C23H27ClN4O3
DC9627
>98%
AZM475271 is a potent and selective Src kinase inhibitor with IC50 of 5 nM; no inhibitory activity on Flt3, KDR, Tie-2._x000D_
AZOCOSTEROL 2HCL
CAS:1249-84-9
Formula: C25H44N2O.2ClH
DC4141
99%
Azocosterol is a potential avian reproductive inhibitor.
AZOMYCIN (2-NITROIMIDAZOLE)
CAS:527-73-1
Trade Name: 2-Nitroimidazole
Formula: C3H3N3O2
DCAPI1225
>99%
Azomycin (2-Nitroimidazole)
AZORAMIDE
CAS:932986-18-0
Formula: C15H17ClN2OS
DC9818
>98%
Azoramide is a small-molecule modulator of the unfolded protein response with antidiabetic activity.
AZTREONAM (AZACTAM, CAYSTON)
CAS:78110-38-0
Trade Name: Monobactam, SQ 26776, Squibb 26776
Formula: C13H17N5O8S2
DCAPI1341
>99%
Aztreonam (Azactam, Cayston)
B-AP15(NSC687852)
CAS:1009817-63-3
Trade Name: NSC687852,NSC-687852,NSC 687852
Formula: C22H17N3O6
DC8203
>98%
b-AP15(NSC687852) is a specific inhibitor of the deubiquitinating enzymes UCHL5 and Usp14 of the 26S proteasome. It blocks the deubiquitinating activity of the 26S proteasome.
B-HT 920
CAS:36085-73-1
Trade Name: Domin; Talipexole dihydrochloride
Formula: C10H17Cl2N3S
DC9426
>98%
B-HT 920(Talipexole 2Hcl) is a dopamine D2 receptor agonist, a2-adrenoceptor agonist and 5-HT3 receptor antagonist, which displays antiParkinsonian activity._x000D_
B-RAF IN 1
CAS:950736-05-7
Formula: C29H24F3N5O
DC7718
>98%
B-Raf IN 1 is a highlt potent and selective B-Raf inhibitor with IC50 of 24 nM; equipotent against c-Raf (IC50= 25 nM).
B-RAF INHIBITOR (BENZAMIDE)
CAS:1315330-11-0
Trade Name: 1315330-11-0, SureCN14689441, AKOS016012030, B-Raf inhibitor|1315330-11-0, CS-1099, AK122840, HY-772
Formula: C29H31F3N6O2
DC7537
>98%
A B-Raf inhibitor, pyrazine and pyrrolo[2,3-b]pyridine derivatives, useful in the treatment of cancer and proliferative diseases.
B-RAF INHIBITOR 1
CAS:1093100-40-3
Formula: C26H19ClN8
DC8921
>98%
B-Raf inhibitor 1 is a potent and selective B-Raf inhibitor with cell IC50s of 0.31 uM and 2 nM for A375 proliferation and A375 p-ERK respectively.
B02
CAS:1290541-46-6
Formula: C22H17N3O
DC10026
>98%
B02 is a cell-permeable pyridinylvinyl-quinazolinone compound that is shown to specifically inhibit human RAD51 (IC50 = 27.4 M).
BACCATINE III
CAS:27548-93-2
Formula: C31H38O11
DCZ-169
>98%
>98%,Standard References
BACITRACIN ZINC
CAS:1405-89-6
Trade Name: N/A
Formula: C66H101N17O16SZn
DCAPI1066
>99%
Bacitracin zinc
BACLOFEN
CAS:1134-47-0
Formula: C10H12ClNO2
DC8971
>98%
Baclofen is a gamma-amino-butyric acid (GABA) derivative used as a skeletal muscle relaxant.
BAF312 (SIPONIMOD)
CAS:1230487-00-9
Trade Name: Siponimod; Siponimod [INN]; BAF-312, BAF 312
Formula: C29H35F3N2O3
DC7694
>98%
BAF312 is a potent and selective agonist of S1P with EC50 value of 0.39nM for S1P1 receptors and 0.98nM for S1P5 receptors, respectively
BAFETINIB (INNO-406)
CAS:859212-16-1
Trade Name: NS-187, Bafetinib, INNO406
Formula: C30H31F3N8O
DC2013
>98%
Bafetinib (INNO-406) is a potent and selective dual Bcr-Abl/Lyn inhibitor with IC50 of 5.8 nM and 19 nM, respectively.
BAFILOMYCIN A1(BAF-A1)
CAS:88899-55-2
Formula: C35H58O9
DC8858
>98%
Bafilomycin A1 is a vacuolar H+-ATPase inhibitor with IC50 of 0.44 nM.
BAICALEIN
CAS:491-67-8
Formula: C15H10O5
DCH-018
>98%,Standard References Grade
>98%,Standard References
BAICALIN
CAS:21967-41-9
Formula: C21H18O11
DCH-016
>98%,Standard References Grade
>98%,Standard References
BAKKENOLIDE A
CAS:19906-72-0
Formula: C15H22O2
DCF-024
>98%,Standard References Grade
>98%,Standard References
BAKUCHIOL
CAS:10309-37-2
Formula: C18H24O
DCB-040
>98%,Standard References Grade
>98%,Standard References
BALAGLITAZONE
CAS:199113-98-9
Trade Name: DRF-2593;NN-2344;DRF2593;NN2344;DRF 2593;NN 2344
Formula: C20H17N3O4S
DC9602
>98%
Balaglitazone (DRF-2593; NN-2344) is a novel partial agonist of PPAR-?._x000D_
BALAPIRAVIR
CAS:690270-29-2
Trade Name: R-1626; R 1626; Ro 4588161; R1626; Ro4588161; Ro-4588161
Formula: C21H30N6O8
DC7541
>98%
Balapiravir (R1626, Ro 4588161) is the prodrug of a nucleoside analogue inhibitor of the hepatitis C virus (HCV) RNA-dependent RNA polymerase (R1479, RG1479).
BALICATIB
CAS:354813-19-7
Trade Name: AAE581; AAE 581; AAE-581
Formula: C23H33N5O2
DC7371
>98%
Balicatib(AAE-581) is a potent and selective inhibitor of cathepsin K; 10-100-fold more potent in cell-based enzyme occupancy assays than against cathepsin B, L, and S.
BALOFLOXACIN
CAS:127294-70-6
Trade Name: N/A
Formula: C20H24FN3DCAPI1046
>99%
Balofloxacin
BALSALAZIDE
CAS:80573-04-2
Trade Name: Colazal;Giazo
Formula: C17H15N3O6
DC9562
>98%
Balsalazide is an anti-inflammatory compound used in the treatment of Inflammatory Bowel Disease._x000D_
BAM 7
CAS:331244-89-4
Trade Name: BAM7; BAM-7
Formula: C21H19N5O2S
DC7080
>98%
BAM 7 is a direct and selective activator of proapoptotic Bax with EC50 of 3.3 M.
BAMAQUIMAST
CAS:135779-82-7
Formula: C16H21N3O3
DC9869
>98%
Bamaquimast is an inhibitor of proton pump extracted from patent US2005165041, example 138.
BAMBUTEROL HCL
CAS:81732-46-9
Formula: C18H30ClN3O5
DC9117
>98%
Bambuterol Hcl is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma; it also is a prodrug of terbutaline.
BAN ORL 24
CAS:1401463-54-4
Trade Name: BANORL 24,BAN ORL24,BANORL24,BAN ORL-24
Formula: C27H35N3O2.2HCl
DC8298
>98%
BAN ORL 24 is a potent, selective, competitive ORL1 non-peptide agonist. Displays 1000-fold selectivity over classical opioid receptors.
BAOHUOSIDE I
CAS:113558-15-9
Formula: C27H30O10
DCB-063
>98%,Standard References Grade
>98%,Standard References
BAPTA/AM(BAPTA-AM)
CAS:126150-97-8
Trade Name: BAPTA/AM,BAPTAAM,BAPTA AM,BAPTA-AM
Formula: C34H40N2O18
DC10502
>98%
BAPTA/AM is a membrane permeable form of BAPTA, a selective chelator of Ca2+.
BAR 502
CAS:1612191-86-2
Trade Name: BAR 502,BAR-502,BAR502
Formula: C25H44O3
DC10564
>98%
BAR502 is a dual FXR and GPBAR1 agonist with IC50 values of 2 M and 0.4 M, respectively.
BAR501
CAS:1632118-69-4
Trade Name: BAR 501; BAR-501
Formula: C26H46O3
DC10385
>98%
BAR501 is a potent and selective agonist of GPBAR1 with an EC50 of 1 M.
BARASERTIB (AZD1152-HQPA)
CAS:722544-51-6
Trade Name: AZD1152, AZD-1152
Formula: C26H30FN7O3
DC1029
>98%
AZD1152-HQPA (Barasertib) is a highly selective Aurora B inhibitor with IC50 of 0.37 nM.
BARBALOIN
CAS:1415-73-2
Formula: C21H22O9
DCL-008
>98%,Standard References Grade
>98%,Standard References
BARDOXOLONE METHYL
CAS:218600-53-4
Formula: C32H43NO4
DC4135
99%
Bardoxolone methyl (also known as RTA 402 and CDDO-methyl ester) is an orally-available first-in-class synthetic triterpenoid belonging to the antioxidant inflammation modulator (AIM) class.
BARICITINIB (INCB28050, LY3009104)
CAS:1187594-09-7
Trade Name: Baricitinib, INCB28050, LY3009104.
Formula: C16H17N7O2S
DC5064
>98%
Baricitinib is a selective JAK1 and JAK2 inhibitor with IC50 of 5.9 nM and 5.7 nM, ~70 and ~10-fold selective versus JAK3 and Tyk2, no inhibition to c-Met and Chk2. Phase 3.
BARICITINIB PHOSPHATE
CAS:1187595-84-1
Trade Name: INCB-028050,LY-3009104,INCB 028050,LY 3009104,INCB028050,LY3009104
Formula: C16H20N7O6PS
DC8258
>98%
Baricitinib phosphate(INCB 028050; LY 3009104) is a selective JAK1 and JAK2 inhibitor with IC50 of 5.9 nM and 5.7 nM, ~70 and ~10-fold selective versus JAK3 and Tyk2, no inhibition to c-Met and Chk2.
BASMISANIL(RG1662)
CAS:1159600-41-5
Trade Name: RG 1662; RG-1662; RG1662; RO5186582; RO-5186582; RO 5186582; Basmisanil
Formula: C21H20FN3O5S
DC9935
>98%
Basmisanil is a highly selective inverse agonist/negative allosteric modulator of a5 subunit-containing GABAA receptors which is under development by Roche for the treatment of cognitive impairment associated with Down syndrome.
BATEFENTEROL(GSK961081)
CAS:743461-65-6
Trade Name: GSK961081; GSK-961081; GSK 961081; TD-5959; TD 5959; TD5959; Batefenterol
Formula: C40H42ClN5O7
DC10021
>98%
Batefenterol(GSK961081,TD-5959)is a Muscarinic Antagonist and 2-Agonist possessing both muscarinic antagonist (MA) and 2-adrenoceptor agonist (BA) properties (MABA).
BATIMASTAT(BB-94)
CAS:130370-60-4
Trade Name: BB94,BB 94
Formula: C23H31N3O4S2
DC8133
>98%
Batimastat was used to study the role of MMP in proteolytic release of EGF in human follicular thyroid carcinoma cell line FTC-133.
BAVACHININ A
CAS:19879-30-2
Formula: C21H22O4
DCB-076
>98%,Standard References Grade
>98%,Standard References
BAY 1082439
CAS:1375469-38-7
Trade Name: BAY10-82439; BAY 10-82439; BAY-10-82439; BAY1082439; BAY 1082439; BAY-1082439
Formula: C25H30N6O5
DC9939
>98%
BAY 1082439 is a highly selective and balanced PI3Ka/ inhibitor demonstrated potent activity in tumors with activated PI3Ka and loss-of-function of PTEN.
BAY 11-7085
CAS:196309-76-9
Trade Name: Bay117085,Bay11-7085
Formula: C13H15NO2S
DC8038
>98%
BAY 11-7085 is an irreversible inhibitor of TNFa-induced I?Ba phosphorylation with an IC50 value of 10 M.
BAY 41-2272
CAS:256376-24-6
Trade Name: BAY 41-2272, 256376-24-6, UNII-34A162J6WB, IN1523, BAY-41-2272, 3-(4-Amino-5-cyclopropylpyrimidin-2-
Formula: C20H17FN6
DC7782
>98%
BAY 41-2272 is a soluble guanylate cyclase agonist, activates human mononuclear phagocytes
BAY 41-4109
CAS:298708-81-3
Trade Name: Bay41-4109; Bay-41-4109; Bayer 41-4109
Formula: C18H13ClF3N3O2
DC10294
>98%
BAY 41-4109 is a potent inhibitor of human hepatitis B virus (HBV) with an IC50 of 53 nM.
BAY 41-4109 (RACEMATE)
CAS:298708-79-9
Trade Name: Bay41-4109 racemate; Bay-41-4109 racemate
Formula: C18H13ClF3N3O2
DC10085
>98%
BAY 41-4109 racemate is a potent inhibitor of human hepatitis B virus (HBV) with an IC50 of 53 nM.
BAY 41-4109 LESS ACTIVE ENANTIOMER
CAS:476617-51-3
Trade Name: Bay41-4109 less active enantiomer; Bay-41-4109 less active enantiomer; Bayer 41-4109 less active ena
Formula: C18H13ClF3N3O2
DC10291
>98%
Bay 41-4109 less active enantiomer shows less activity than Bay 41-4109. BAY 41-4109 is a potent inhibitor of human hepatitis B virus (HBV) with an IC50 of 53 nM.
BAY 59-3074
CAS:406205-74-1
Trade Name: BAY-59-3074; BAY 59-3074; BAY59-3074
Formula: C18H13F6NO4S
DC9783
>98%
Bay 59-3074 is a novel CB1/CB2 receptor partial agonist (Ki values are 48.3 and 45.5 nM at human CB1 and CB2 receptors respectively).
BAY 59-7939(RIVAROXABAN)
CAS:366789-02-8
Formula: C19H18ClN3O5S
DC5108
>98%
Rivaroxaban (Xarelto; BAY 59-7939) is a novel, oral, direct Factor Xa (FXa) inhibitor in late-stage development for the prevention and treatment of thromboembolic disorders.
BAY 60-7550
CAS:439083-90-6
Trade Name: BAY 607550;Bay60-7550;Bay-60-7550
Formula: C27H32N4O4
DC9578
>98%
Bay 60-7550 is a potent PDE2 inhibitor with IC50 values of 2.0 nM (bovine) and 4.7 nM (human); 50-fold more selective for PDE2 compared to PDE1 and greater than 100-fold selective compared to PDE5, PDE3B, PDE4B, PDE7B, PDE8A, PDE9A, PDE10A, and PDE11A._x000D_
BAY 61-3606 (DIHYDROCHLORIDE)
CAS:648903-57-5
Trade Name: BAY61-3606 dihydrochloride;BAY 61-3606
Formula: C20H20Cl2N6O3
DC9632
>98%
BAY 61-3606 2Hcl is a potent, ATP-competitive, reversible, and highly selective inhibitor of Syk tyrosine kinase activity (Ki= 7.5 nM) with no inhibitory effect against Btk, Fyn, Itk, Lyn, and Src._x000D_
BAY 80-6946
CAS:1032568-63-0
Trade Name: BAY80-6946; Copanlisib
Formula: C23H28N8O4
DC9591
>98%
BAY 80-6946(Copanlisib) is a potent and highly selective reversible PI3K inhibitor for PI3Ka/ with IC50 of 0.469 nM/3.72 nM._x000D_
BAY 87-2243
CAS:1227158-85-1
Trade Name: BAY87 2243,BAY 87 2243,BAY87-2243
Formula: C26H26F3N7O2
DC7996
>98%
BAY 87-2243 is a highly potent and selective inhibitor of hypoxia-induced HIF-1 activation.
BAY-1143572
CAS:1414943-88-6
Trade Name: BAY1143572; BAY 114357
Formula: C18H18FN5O2S
DC10376
>98%
BAY 1143572 is a highly selective, potent and orally available inhibitor of PTEFb/CDK9; inhibits the proliferation of AML cell lines with a median IC50 of 385 nM.
BAY-1895344
CAS:1876467-74-1
Trade Name: BAY1895344,BAY 1895344,BAY-1895344
Formula: C20H22ClN7O
DC10526
>98%
BAY-1895344 is a potent and selective ATM inhibitor. BAY 1895344 shows potent anti-tumor efficacy in monotherapy and strong combination potential with the targeted alpha therapy Radium-223 dichloride.
BAY-876
CAS:1799753-84-6
Trade Name: BAY876,BAY 876
Formula: C24H16F4N6O2
DC10107
>98%
BAY-876 is the first highly selective GLUT1 inhibitor with IC50 of 0.002 uM. show good metabolic stability in vitro and high oral bioavailability in vivo.
BAY11-7082
CAS:19542-67-7
Trade Name: BAY 11-7821
Formula: C10H9NO2S
DC7869
>98%
BAY 11-7082 is a NF-?B inhibitor, inhibits TNFa-induced I?Ba phosphorylation with IC50 of 10 M. Also inhibiting components of the ubiquitin system.
BAY1125976
CAS:1402608-02-9
Trade Name: BAY-1125976; BAY 1125976
Formula: C23H21N5O
DC10408
>98%
BAY1125976 is a selective allosteric Akt1/2 inhibitor; inhibits Akt1 and Akt2 activity with IC50 values of 5.2 nM and 18 nM at 10 M ATP, respectively.
BAY1217389
CAS:1554458-53-5
Trade Name: BAY1217389; BAY-1217389; BAY 1217389
Formula: C27H24F5N5O3
DC9679
>98%
BAY1217389 is an orally bioavailable, selective inhibitor of the serine/threonine kinase monopolar spindle 1 (Mps1, TTK), with potential antineoplastic activity.
BAYER-18
CAS:1251752-12-1
Trade Name: Bayer18,Bayer 18
Formula: C19H27FN6O2
DC10057
>98%
Bayer-18 is a selective TYK2 inhibitor, with an IC50 of 18.7nM on TYK2 as measured by TYK2 HTRF assays.
BAYOGENIN
CAS:6989-24-8
Formula: C30H48O5
DCB-053
>98%,Standard References Grade
>98%,Standard References
BAZ2-ICR
CAS:1665195-94-7
Trade Name: BAZ2ICR
Formula: C20H19N7
DC7854
>98%
BAZ2-ICR is a selective BAZ2 bromodomain inhibitor (Kd values are 109 and 170 nM for BAZ2A and BAZ2B respectively).
BAZEDOXIFENE
CAS:198481-32-2
Formula: C30H34N2O3
DC8922
>98%
Bazedoxifene is a selective estrogen receptor modulator (SERM) currently in development for osteoporosis prevention and treatment.
BAZEDOXIFENE (ACETATE)
CAS:198481-33-3
Trade Name: TSE 424;Viviant;WAY-TES 424
Formula: C32H38N2O5
DC9439
>98%
Bazedoxifene acetate (TSE 424; WAY-TES 424), a novel selective estrogen receptor modulator (SERM), has been developed to have favorable effects on bone and the lipid profile while minimizing stimulation of uterine or breast tissues.
BAZEDOXIFENE-ACETATE
CAS:198480-56-7
Trade Name: TSE 424; Viviant; WAY-TES 424
Formula: C32H38N2O5
DC7372
>98%
Bazedoxifene acetate (TSE 424; WAY-TES 424), a novel selective estrogen receptor modulator (SERM), has been developed to have favorable effects on bone and the lipid profile while minimizing stimulation of uterine or breast tissues.
BBS-4
CAS:402934-09-2
Trade Name: bbs4
Formula: C22H24N6O3
DC7870
>98%
BBT594
CAS:882405-89-2
Trade Name: BBT 594,BBT 594
Formula: C28H30F3N7O3
DC10058
>98%
BBT594 (NVP-BBT594), is potent and selective inhibitor of RET and JAK2.
BCL6 INHIBITOR(CID5721353)
CAS:301356-95-6
Trade Name: CID 5721353,CID-5721353,CID 5721353
Formula: C15H9BrN2O6S2
DC9955
>98%
CID5721353 is a B-Cell Lymphoma 6 Inhibitor (BCL6 inhibitor).
BCTC
CAS:393514-24-4
Formula: C20H25ClN4O
DC9826
>98%
BCTC is a potent and specific inhibitor of transient receptor potential cation channel subfamily M member 8 (TRPM8) in prostate cancer (PCa) DU145 cells.
BD1047.2HBR
CAS:138356-21-5
Trade Name: BD-1047,BD 1047
Formula: C13H20Cl2N2.2HBr
DC8313
>98%
BD 1047 dihydrobromide is a selective antagonist of s receptors.
BD1063 DHYDROCHLORIDE
CAS:206996-13-6
Trade Name: BD-1063 dhydrochloride; BD 1063 dhydrochloride
Formula: C13H20Cl4N2
DC10280
>98%
BD1063 dhydrochloride is a potent and selective sigma 1 receptor antagonist.
BDA-366
CAS:1821496-27-8
Trade Name: BDA-366,BDA 366,BDA366
Formula: C24H29N3O4
DC9709
>98%
BDA-366 is a Small-Molecule Bcl2 BH4 Antagonist for Lung Cancer Therapy.
BDP-12(AMPALEX)
CAS:154235-83-3
Trade Name: CX516; BDP 12; Ampakine CX516
Formula: C14H15N3O
DC5075
>98%
Ampalex (Ampakine CX516) is an ampakine and nootropic that acts as an AMPA receptor positive allosteric modulator as a treatment for Alzheimer's disease, schizophrenia and mild cognitive impairment (MCI).
BEBT-908(CUDC-908)
CAS:1235449-52-1
Trade Name: BEBT908,CUDC908,BEBT 908,CUDC 908
Formula: C23H25N9O3S
DC9718
>98%
BEBT-908(CUDC-908)is a novel PI3K/HDAC inhibitor.
BEC HYDROCHLORIDE
CAS:222638-67-7
Formula: C5H13BClNO4S
DC9964
>98%
BEC is a boronic acid-based arginine analog that acts as a slow-binding, competitive transition state inhibitor of arginase I and II (Ki = 310 nM for human recombinant type II arginase, pH 7.5).
BECLABUVIR(BMS-791325)
CAS:958002-33-0
Trade Name: BMS-791325
Formula: C36H45N5O5S
DC8178
>98%
non-nucleoside inhibitor of the NS5B
BECLOMETHASONE DIPROPIONATE
CAS:5534-09-8
Formula: C28H37ClO7
DC9172
>98%
Beclometasone dipropionate is a potent glucocorticoid agonist; it is a prodrug of the free form, beclometasone.
BEDAQUILINE (TMC207)
CAS:843663-66-1
Trade Name: Bedaquiline, TMC-207
Formula: C32H31BrN2O2
DC2012
>99.5%
TMC207 is a first-in-class diarylquinoline compound with a novel mechanism of action, the inhibition of bacterial ATP synthase, and potent activity against drug-sensitive and drug-resistant TB.
BEDAQUILINE FUMARATE
CAS:845533-86-0
Trade Name: TMC-207,TMC207,TMC 207
Formula: C36H35BrN2O6
DC8809
>99%
Bedaquiline fumarate(TMC207; R207910) is an anti-tuberculosis drug which selectively inhibit the mycobacterial energy metabolism i.e. ATP synthesis and found to be effective against all states of Mycobacterium tuberculosis.
BELINOSTAT(PXD101)
CAS:414864-00-9
Trade Name: PXD101; PX105684; PXD-101; PXD 101; PX-105684
Formula: C15H14N2O4S
DC7082
>98%
Belinostat (PXD101) is a novel pan-HDAC inhibitor with IC50 of 27 nM, with activity demonstrated in cisplatin-resistant tumors.
BELIZATINIB(TSR-011)
CAS:1357920-84-3
Trade Name: TSR011; TSR011; TSR 011; Belizatinib
Formula: C33H44FN5O3
DC10448
>98%
Belizatinib(TSR-011) is an orally available inhibitor of both the receptor tyrosine kinase anaplastic lymphoma kinase (ALK) and the tropomyosin-related kinases (TRK) TRKA, TRKB, and TRKC, with potential antineoplastic activity.
BELLIDIFOLIN
CAS:2798-25-6
Formula: C14H10O6
DCL-066
>98%,Standard References Grade
>98%,Standard References
BELNACASAN(VX-765)
CAS:273404-37-8
Trade Name: VX 765; VX-765; VX765. Belnacasan
Formula: C24H33ClN4O6
DC5080
>98%
VX-765 is a novel Caspase-1 inhibitor with an IC 50 of 0.8nM being investigated for the treatment of epilepsy, currently being developed by Vertex.
BEMPEDOIC ACID(ETC-1002;ESP-55016)
CAS:738606-46-7
Trade Name: ETC1002; ESP55016
Formula: C19H36O5
DC8182
>98%
ETC-1002(ESP-55016) is a novel, first-in-class, orally available, once-daily LDL-C lowering small molecule; activator of hepatic AMP-activated protein kinase (AMPK); also has potent inhibitory activity against hepatic ATP-citrate lyase(IC50=29 uM).
BENAZEPRIL HYDROCHLORIDE
CAS:86541-74-4
Formula: C24H29ClN2O5
DC9152
>98%
Benazepril hydrochloride, an angiotensin converting enzyme inhibitor, which is a medication used to treat high blood pressure.
BENDAMUSTINE HCL(SDX-105,CYTOSTASANE)
CAS:3543-75-7
Trade Name: Treanda,Bendamustinum;Bendamustina;DD6304600;SDX-105 Ribomustin.
Formula: C16H22Cl3N3O2
DC6908
>98%
Bendamustine HCL (Ribomustin, Treanda, SDX-105) is a DNA-damaging agent with IC50 of 50 M.
BENGENIN
CAS:477-90-7
Formula: C14H16O9
DCY-015
>98%,Standard References Grade
>98%,Standard References
BENSERAZIDE
CAS:14919-77-8
Trade Name: Serazide
Formula: C10H15N3O5.HCl
DCAPI1606
99%
Benserazide is a peripherally-acting aromatic L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.
BENZALDEHYDE
CAS:100-52-7
Formula: C7H6O
DCB-083
>98%,Standard References Grade
>98%,Standard References
BENZBROMARON
CAS:3562-84-3
Formula: C17H12Br2O3
DC8895
>98%
Benzbromarone is a highly effective and well tolerated non-competitive inhibitor of xanthine oxidase, used as an uricosuric agent, used in the treatment of gout.
BENZENESULFONAMIDE
CAS:98-10-2
Formula: C6H7NO2S
DC9885
>98%
Benzenesulfonamide ia an inhibitor of carbonic anhydrases
BENZOCAINE HYDROCHLORIDE
CAS:23239-88-5
Trade Name: Benzocaine hydrochloride
Formula: C9H11NO2.HCl
DC10223
>98%
Benzocaine hydrochloride is a surface anesthetic that acts by preventing transmission of impulses along nerve fibers and at nerve endings.
BENZOIC ACID
CAS:65-85-0
Formula: C7H6O2
DCB-013
>98%,Standard References Grade
>98%,Standard References
BENZOYLACONINE
CAS:466-24-0
Formula: C32H45NO10
DCB-010
>98%,Standard References Grade
>98%,Standard References
BENZOYLHYPACOITINE
CAS:63238-66-4
Formula: C31H43NO9
DCB-016
>98%,Standard References Grade
>98%,Standard References
BENZOYLMESACONINE
CAS:63238-67-5
Formula: C31H43NO10
DCB-009
>98%,Standard References Grade
>98%,Standard References
BENZOYLPAEONIFLORIN
CAS:38642-49-8
Formula: C30H32O12
DCB-024
>98%,Standard References Grade
>98%,Standard References
BENZYL BENZOATE
CAS:120-51-4
Formula: C14H12O2
DCZ-172
>98%
>98%,Standard References
BEPOTASTINE
CAS:190786-43-7
Formula: C21H25ClN2O3
DC8898
>98%
Bepotastine is a non-sedating, selective antagonist of the histamine 1 (H1) receptor.
BEPOTASTINE BESILATE
CAS:190786-44-8
Trade Name: N/A
Formula: C27H31ClN2O6S
DCAPI1500
>99%
1--D-Arabinofuranosylcytosine, a cytosine analogue, inhibits DNA polymerases a, d, and e, and RNA polymerases resulting in suppression of DNA synthesis and repair. 1--D-Arabinofuranosylcytosine acts as an antimetabolic agent which is responsible for dam
BERBAMINE DIHYDROCHLORIDE
CAS:6078-17-7
Formula: C37H42Cl2N2O5
DCY-001
>98%,Standard References Grade
>98%,Standard References
BERBERINE HYDROCHLORIDE
CAS:633-65-8
Formula: C20H18ClNO4
DCY-035
>98%,Standard References Grade
>98%,Standard References
BERBERRUBINE
CAS:15401-69-1
Formula: C19H15NO4
DCX-061
>98%,Standard References Grade
>98%,Standard References
BERGAMOTTIN
CAS:7380-40-7
Trade Name: Bergamotine; Bergaptin
Formula: C21H22O4
DC8027
>98%
Bergamottin is a natural furanocoumarin found principally in grapefruit juice.
BERGAPTEN
CAS:484-20-8
Formula: C12H8O4
DCF-008
>98%,Standard References Grade
>98%,Standard References
BESIFLOXACIN HCL
CAS:405165-61-9
Trade Name: N/A
Formula: C19H21ClFN3O3.HCl
DC4143
99%
Besifloxacin HCl is a fourth-generation fluoroquinolone antibiotic.
BET BROMODOMAIN INHIBITOR,CAS 1505453-59-7
CAS:1505453-59-7
Formula: C24H20ClN5O2
DC7565
>98%
A new compound which is similar with +JQ-1,BET bromodomain inhibitor
BET-BAY 002
CAS:1588521-78-1
Formula: C22H18ClN5O
DC8556
>98%
BET-BAY 002 is a potent BET inhibitor; shows efficacy in a multiple myeloma model.
BETA-BOSWELLIC ACID,11-KETO
CAS:17019-92-0
Formula: C30H46O4
DCT-017
>98%,Standard References Grade
>98%,Standard References
BETA-BOSWELLIC ACID,3-ACETYL,11-KETO
DCY-090
>98%,Standard References Grade
>98%,Standard References
BETA-D-FRUCTOPYRANOSE
CAS:7660-25-5,57-48-7
Formula: C6H12O6
DCG-029
>98%,Standard References Grade
>98%,Standard References
BETA-LAPACHONE (ARQ-501, CO-501)
CAS:4707-32-8
Trade Name: ARQ-501; NSC-26326; NSC-629749; SL-11001; beta-lapachone, -Lapachone, ARQ-501
Formula: C15H14O3
DC7905
>98%
Beta-Lapachone is a selective DNA topoisomerase I inhibitor, exhibiting no inhibitory activities against DNA topoisomerase II or ligase. Phase 2.
BETA-PINENE
CAS:127-91-3
Formula: C10H16
DCP-014
>98%,Standard References Grade
>98%,Standard References
BETA-ROSASTEROL
DCF-009
>98%,Standard References Grade
>98%,Standard References
BETAHISTINE
CAS:5638-76-6
Formula: C8H12N2
DC8830
>98%
Betahistine is a strong affinity histamine H3 receptor antagonist and weak affinity agonist of histamine H1 receptors.
BETAHISTINE DIHYDROCHLORIDE
CAS:5579-84-0
Formula: C8H14Cl2N2
DC8967
>98%
Betahistine Dihydrochloride is a histamine H3 receptors inhibitor used as an antivertigo drug.
BETAHISTINE EP IMPURITY C
CAS:5452-87-9
Formula: C15H19N3
DC8829
>98%
N-Methyl-N,N-bis(2-pyridylethyl)amine is used as a reagent in the preparation of copper pyridylmethylethylenediamine dicyanamido polymeric complexes.
BETAINE
CAS:107-43-7
Formula: C5H11NO2
DCT-010
>98%,Standard References Grade
>98%,Standard References
BETAINE HYDROCHLORIDE
CAS:590-46-5
Formula: C5H12ClNO2
DCY-098
>98%,Standard References Grade
>98%,Standard References
BETAMETHASONE (CELESTONE)
CAS:378-44-9,956901-32-9(XHCl)
Trade Name: Celestone, Betadexamethasone, Flubenisolone, Sch-4831, NCS-39470
Formula: C22H29FO5
DCAPI1169
>99%
Betamethasone (Celestone)
BETAMETHASONE VALERATE(BETNOVATE)
CAS:2152-44-5
Trade Name: Betnovate, Celestone, Betaderm, Luxiq
Formula: C27H37FO6
DCAPI1114
>99%
BETAPAR(MEPREDNISONE)
CAS:1247-42-3
Trade Name: Betanisona
Formula: C22H28O5
DCAPI1040
>99%
Betapar(Meprednisone)
BETRIXABAN
CAS:330942-05-7
Trade Name: Betrixaban;MK-4448; PRT-021; PRT-054021; MLN-1021
Formula: C23H22ClN5O3
DC7373
>98%
Betrixaban (PRT-054021) is a highly potent, selective, and orally efficacious factor Xa inhibitor with IC50 of 1.2 nM(inhibition of Factor 10a).
BETULIN
CAS:473-98-3
Formula: C30H50O2
DCB-026
>98%,Standard References Grade
>98%,Standard References
BETULINIC ACID
CAS:472-15-1
Formula: C30H48O3
DC9832
>98%
Betulinic acid, a pentacyclic triterpene, selectively induces apoptosis in tumor cells, also is a inhibitor of HIV-1 with EC50 of 1.4 M.
BETULINICALDEHYDE
CAS:13159-28-9
Formula: C30H48O2
DCB-068
>98%,Standard References Grade
>98%,Standard References
BEVIRIMAT(PA-457)
CAS:174022-42-5
Trade Name: PA-457; MPC-4326; FH11327; YK FH312
Formula: C36H56O6
DC9643
>98%
Bevirimat(YK FH312; FH11327; MPC-4326) is an anti-HIV drug derived from a betulinic acid-like compound; is believed to inhibit HIV by a novel mechanism, so-called maturation inhibition.
BEXAGLIFLOZIN(THR1442,EGT1442)|
CAS:1118567-05-7
Trade Name: EGT1442; THR1442; EGT0001442; EGT-1442; THR-1442; EGT-0001442; EGT 1442; THR 1442; EGT 0001442
Formula: C24H29ClO7
DC8186
>98%
Bexagliflozin is a potent and selective SGLT2 inhibitor with IC50 value of 5.6 M /2 nM in SGLT1 /SGLT2 respectively.
BEXAROTENE
CAS:153559-49-0
Trade Name: N/A
Formula: C24H28O2DCAPI1078
>99%
Bexarotene
BEZAFIBRATE
CAS:41859-67-0
Formula: C19H20ClNO4
DC9088
>98%
Bezafibrate(BM15075) is the first clinically tested dual and pan-PPAR co-agonism.
BFH772
CAS:890128-81-1
Trade Name: BFH-772; BFH 772
Formula: C23H15F3N3O3
DC9956
>98%
BFH772 is a potent oral VEGFR2 inhibitor, which is highly effective at targeting VEGFR2 kinase with an IC50 value of 3 nM.
BG-45
CAS:926259-99-6
Trade Name: BG45,BG 45
Formula: C11H10N4O
DC8310
>98%
BG45 is an HDAC class I inhibitor with selectivity for HDAC3 (IC50= 289 nM). It inhibits HDAC1, HDAC2, and HDAC6 with greatly reduced potency (IC50s = 2, 2.2, and >20 M, respectively).
BGB-3111
CAS:1633350-06-7
Trade Name: BGB3111; BGB 3111
Formula: C27H29N5O3
DC10335
>98%
BGB-3111 is a potent, selective and orally available Bruton's tyrosine kinase (Btk) inhibitor.
BGB283
CAS:1446090-77-2
Trade Name: BGB-283,BGB 283
Formula: C25H17F3N4O3
DC10099
>98%
BGB-283 is a Novel potent and selective RAF Kinase and EGFR inhibitor.
BGG463
CAS:890129-26-7
Trade Name: BGG 463,BGG-463
Formula: C30H29F3N6O3
DC10059
>98%
BGG463 can inhibit c-ABL-T334I, BCR-ABL and BCR-ABL-T315I variants with a 50% inhibitory concentration (IC50) of 0.25 M, 0.09 M and 0.590 M, respectively.
BGP-15
CAS:66611-37-8
Trade Name: BGP 15,BGP15
Formula: C14H22N4O2.2HCl
DC8571
>98%
BGP-15 is a PARP inhibitor and insulin sensitizer.
BH3I-1
CAS:300817-68-9
Trade Name: BH3I 1 ,BH3I1
Formula: C15H14BrNO3S2
DC9695
>98%
BH3I-1 is a cell permeable BH3 mimetic that binds to Bcl-xL. BH3I-1 is an inhibitor of Bcl-xL.
BI 2536
CAS:755038-02-9
Trade Name: BI-2536; BI2536
Formula: C28H39N7O3
DC7083
>98%
BI2536 is a potent Plk1 inhibitor with IC50 of 0.83 nM, BI2536 shows 4- and 11-fold greater selectivity against Plk2 and Plk3; BI2536 also is a BRD4 inhibitor(IC50= 25 nM).
BI-7273
CAS:1883429-21-9
Trade Name: BI 7273,BI7273
Formula: C20H23N3O3
DC9724
>98%
BI-7273 is a potent, selective, and cell-permeable BRD9 BD Inhibitor.
BI-78D3
CAS:883065-90-5
Formula: C13H9N5O5S2
DC7107
>98%
BI-78D3 is a competitive c-Jun N-terminal kinase (JNK) inhibitor (IC50 = 280 nM) that displays > 100 fold selectivity over p38a and no activity at mTOR and PI-3K.
BI-847325
CAS:1207293-36-4
Trade Name: BI-847325,BI 847325,BI847325
Formula: C29H28N4O2
DC8401
>98%
BI-847325 is an orally bioavailable, and selective dual MEK/Aurora kinase inhibitor with IC50 of 3 nM, 25 nM, 15 nM, 25 nM, and 4 nM for Xenopus laevis Aurora B, human Aurora A and Aurora C, as well as human MEK1 and MEK2, respectively. Phase 1.
BI-9564
CAS:1883429-22-8
Trade Name: BI9564,BI 9564
Formula: C20H23N3O3
DC9888
>98%
BI-9564 is a selective, and cell-permeable BRD9 BD inhibitor, with Kd of 5.9 nM for BRD9, and IC50 of > 100 M for BET family.
BI-D1870
CAS:501437-28-1
Trade Name: BID1870
Formula: C19H23F2N5O2
DC7098
>98%
BI-D1870 is a small molecule, specific inhibitor of p90 RSK (ribosomal S6 kinase) isoforms RSK1, RSK2, RSK3 and RSK4, both in vitro and in vivo, with IC50s are 31 nM, 24 nM, 18 nM, 15 nM, respectively.
BIA 10-2474
CAS:1233855-46-3
Trade Name: BIA10-2474; BIA-10-2474
Formula: C16H20N4O2
DC10404
>98%
BIA 10-2474 is an inhibitor of fatty acid amide hydrolase (FAAH) with IC50 values of 50 to 70mg/kg in various rat brain regions.
BIAPENEM
CAS:120410-24-4
Trade Name: L-627, LJC 10627
Formula: C15H18N4O4S
DC4206
99%
Biapenem is a carbapenem antibiotic.
BIBF 1120 ESYLATE
CAS:656247-18-6
Trade Name: Nintedanib; BIBF1120; Vargatef; BIBF-1120
Formula: C33H39N5O7S
DC8608
>98%
Nintedanib (BIBF 1120) is a potent triple angiokinase inhibitor for VEGFR1/2/3, FGFR1/2/3 and PDGFRa/ with IC50 of 34 nM/13 nM/13 nM, 69 nM/37 nM/108 nM and 59 nM/65 nM.
BIBR 953(DABIGATRAN)
CAS:211914-51-1
Trade Name: BIBR953,BIBR 953,BIBR-953
Formula: C25H25N7O3
DCAPI1112
>99%
BIBR 953 (Dabigatran, Pradaxa) is a highly selective, reversible, and potent thrombin inhibitor and is orally available as the prodrug, dabigatran etexilate.
BIBR-1048(DABIGATRAN,ETEXILATE)
CAS:211915-06-9
Trade Name: BIBR 1048, Dabigatran etexilate,BIBR1048
Formula: C34H41N7O5
DC1010
99%
BIBR-1048 (Dabigatran) is an anticoagulant from the class of the direct thrombin inhibitors.
BIBR-1532
CAS:321674-73-1
Trade Name: BIBR1532; BIBR-1532
Formula: C21H17NO3
DC7085
>98%
BIBR 1532 is a potent, selective, non-competitive telomerase inhibitor with IC50 of 100 nM.
BIBS39
CAS:133085-33-3
Trade Name: BIBS 39; BIBS-39
Formula: C32H36N4O3
DC9670
>98%
BIBS 39 is a new nonpeptide angiotensin II (AII) receptor antagonist.
BIBW2992-MA2 (AFATINIB DIMALEATE)
CAS:850140-73-7
Formula: C24H25ClFN5O32C4H4O4
DC3164
>98%
Afatinib is an irreversible EGFR/HER2 inhibitor with an IC50 of 14 nM for in vitro potency against HER2.
BIBX1382
CAS:196612-93-8
Trade Name: Falnidamol; BIBX-1382; BIBX 1382
Formula: C18H19ClFN7
DC7622
>98%
BIBX 1382 is a potent, selective inhibitor of EGFR tyrosine kinase (IC50 = 3 nM); displays > 1000-fold lower potency against ErbB2 (IC50 = 3.4 M) and a range of other related tyrosine kinases (IC50 > 10 M).
BICYCLOMYCIN BENZOATE
CAS:37134-40-0
Trade Name: FR2054
Formula: C19H22N2O8
DC10393
>98%
Bicyclomycin benzoate is an antibiotic exhibiting activity against a broad spectrum of Gram-negative bacteria and against the Gram-positive bacterium.
BIFEPRUNOX
CAS:350992-10-8
Formula: C24H23N3O2
DC8729
>98%
BIIB021(CNF2024)
CAS:848695-25-0
Trade Name: CNF2024; BIIB-021; BIIB 021; CNF 2024; CNF-2024
Formula: C14H15ClN6O
DC7086
>98%
BIIB021(CNF2024) is an orally available, fully synthetic small-molecule inhibitor of HSP90 with Ki and EC50 of 1.7 nM and 38 nM, respectively.
BIKININ
CAS:188011-69-0
Formula: C9H9BrN2O3
DC8263
>98%
Bikinin is a strong activator of brassinosteroid (BR) signaling.
BILASTINE
CAS:202189-78-4
Formula: C28H37N3O3
DC7995
>98%
Bilastine is a selective histamine H1 receptor antagonist used for treatment of allergic rhinoconjunctivitis and urticaria.
BILIRUBIN
CAS:635-65-4
Formula: C33H36N4O6
DCD-043
>98%,Standard References Grade
>98%,Standard References
BILOBALIDE
CAS:33570-04-6
Trade Name: N/A
Formula: C15H18O8
DCAPI1153
>99%
Bilobalide
BILOBETIN
CAS:521-32-4
Formula: C31H20O10
DCZ-164
>98%
>98%,Standard References
BIMATOPROST
CAS:155206-00-1
Trade Name: Lumigan
Formula: C25H37NO4
DCAPI1079
>99%
Bimatoprost is a prostaglandin analog used topically (as eye drops) to control the progression of glaucoma and in the management of ocular hypertension.
BINDARIT
CAS:130641-38-2
Trade Name: N/A
Formula: C19H20N2O3
DC6801
>99%
Bindarit exhibits selective inhibition against monocyte chemotactic proteins MCP-1/CCL2, MCP-3/CCL7 and MCP-2/CCL8.
BIO
CAS:667463-62-9
Trade Name: GSK-3 Inhibitor IX, 6-bromoindirubin-3-oxime
Formula: C16H10BrN3O2
DC7663
>98%
BIO (6-bromoindirubin-3'-oxime) is a specific inhibitor of GSK-3 with IC50 of 5 nM for GSK-3a/, shows >16-fold selectivity over CDK5, also a pan-JAKinhibitor.
BIO-32546
CAS:1548743-66-3
Trade Name: BIO 32546,BIO32546
Formula: C28H31F6NO3
DC8046
>98%
BIO-ACETOXIME(GSK-3,INHIBITOR,X)
CAS:667463-85-6
Trade Name: GSK3 Inhibitor X6-Bromoindirubin-3'-acetoxime
Formula: C18H12BrN3O3
DC8368
>98%
BIO-Acetoxime is an analog of the GSK3 inhibitor 6-bromoindirubin-3-oxime, or BIO
BIOCHANIN A
CAS:491-80-5
Formula: C16H12O5
DCY-009
>98%,Standard References Grade
>98%,Standard References
BIOYMIFI
CAS:1420071-30-2
Trade Name: (DR5 Activator)
Formula: C22H12BrN3O4S
DC7603
>98%
Bioymifi(DR5 Activator) is the first novel and potent small-molecule activatior of the TRAIL receptor DR5 in human cancer cells.
BIRCH-ME
CAS:119-36-8
Formula: C8H8O3
DCS-018
>98%,Standard References Grade
>98%,Standard References
BIRINAPANT (TL32711)
CAS:1260251-31-7
Trade Name: TL-32711; TL32711; TL 32711. Birinapant
Formula: C42H56F2N8O6
DC5023
>98%
Birinapant (TL32711) is a SMAC mimetic antagonist, mostly to cIAP1 with Kd of <1 nM, less potent to XIAP.
BIS(4-HYDROXYCINNAMOYL) METHANE
CAS:24939-16-0
Formula: C19H16O4
DCZ-101
>98%
>98%,Standard References
BISANTRENE
CAS:78186-34-2
Trade Name: CL216942
Formula: C22H22N8
DC10434
>98%
Bisantrene is a highly effective antitumor drug, targets eukaryotic type II topoisomerases.
BISF-3
CAS:118511-97-0
Trade Name: BISF3,BISF 3
Formula: C8H8ClN3
DC10504
>98%
BISF CAS 118511-97-0
BISINDOLYLMALEIMIDE X HCL
CAS:145317-11-9
Trade Name: BIM X,Ro 31-8425Ro 31-8425
Formula: C26H24N4O2.HCl
DC8504
>98%
Bisindolylmaleimide X is a cell-permeable, reversible, ATP-competitive protein kinase C (PKC) inhibitor (IC50 = 15 nM, rat brain PKC).
BISINDOLYLMALEIMIDE X(RO 31-8425)
CAS:1241725-89-2
Trade Name: BIM X,Ro 31-8425Ro 31-8425
Formula: C26H24N4O2
DC10052
>98%
Bisindolylmaleimide X is a cell-permeable, reversible, ATP-competitive protein kinase C (PKC) inhibitor (IC50 = 15 nM, rat brain PKC).
BISOPROLOL FUMARATE
CAS:104344-23-2
Trade Name: N/A
Formula: C40H55N2O12
DCAPI1411
>99%
()-Bisoprolol hemifumarate is a selective 1-AR adrenergic antagonist. Possesses 1/2 selectivity of approximately 100-fold and a Kd of 2-3 nM at the 1-AR (1 receptor).
BITOPERTIN
CAS:845614-11-1
Formula: C21H20F7N3O4S
DC8882
>98%
Bitopertin, also known as RG1678, is a potent and selective inhibitor of GlyT1 with an EC50 of 30nM.
BIX 02565
CAS:1311367-27-7
Trade Name: BIX-02565;BIX02565
Formula: C26H30N6O2
DC9616
>98%
BIX 02565 is a novel ribosomal S6 kinase 2 (RSK2) inhibitor with an IC50 of 1.1 nM._x000D_
BIX01294
CAS:935693-62-2
Trade Name: BIX 01294; BIX01294,BIX-01294
Formula: C28H38N6O2
DC7374
>98%
BIX01294 is an inhibitor of G9a histone methyltransferase with IC50 of 2.7 M.
BIX02188(BIX,02188)
CAS:334949-59-6
Trade Name: BIX 02188; BIX02188; BIX-02188
Formula: C26H26N4O2
DC5002
>98%
BIX02188 is a selective inhibitor of MEK5 with IC50 of 4.3 nM, also inhibits ERK5 catalytic activity with IC50 of 810 nM, and does not inhibit closely related kinases MEK1, MEK2, ERK2, and JNK2.
BIX02189(BIX,02189)
CAS:1265916-41-3
Trade Name: BIX 02189,BIX02189
Formula: C27H28N4O2
DC5003
>98%
BIX02189 is a selective inhibitor of MEK5 with IC50 of 1.5 nM, also inhibits ERK5 catalytic activity with IC50 of 810 nM, and does not inhibit closely related kinases MEK1, MEK2, ERK2, and JNK2.
BKM120(NVP-BKM120,BUPARLISIB)
CAS:944396-07-0
Trade Name: NVP-BKM-120, BKM-120; Buparlisib
Formula: C18H21F3N6O2
DC5154
>98%
BKM120 is a selective PI3K inhibitor of p110a//d/? with IC50 of 52 nM/166 nM/116 nM/262 nM, respectively. Reduced potency against VPS34, mTOR, DNAPK, with little activity to PI4K.
BKT140
CAS:664334-36-5
Trade Name: BL-8040; TF14016; 4F-Benzoyl-TN14003
Formula: C97H144FN33O19S2
DC10423
>98%
BKT140 is a novel CXCR4 antagonist with an IC50 vakue of ~1 nM.
BLEOMYCIN SULFATE
CAS:9041-93-4
Trade Name: Blenoxane
Formula: C55H85N17O25S4
DC4196
99%
Bleomycin sulfate (Blenoxane) is a glycopeptide antibiotic and an anticancer agent for squamous cell carcinomas (SCC) with IC50 of 4 nM in UT-SCC-19A cells.
BLININ
CAS:125675-09-4
Formula: C22H32O6
DCK-010
>98%,Standard References Grade
>98%,Standard References
BLONANSERIN(AD-5423)
CAS:132810-10-7
Trade Name: Lonasen; AD-5423; AD5423; AD 5423
Formula: C23H30FN3
DC7087
>98%
Blonanserin(AD-5423) is a D2/5-HT2 receptor antagonist, atypical antipsychotic.
BLU-285(AVAPRITINIB)
CAS:1703793-34-3
Trade Name: BLU-285,BLU 285,BLU285
Formula: C26H27FN10
DC10530
>98%
BLU-285 is a potent and selective exon 17 mutant KIT kinase inhibitor with IC50 of 0.27 nM for KIT D816V.
BLU-9931
CAS:1538604-68-0
Trade Name: BLU-9931,BLU 9931,BLU9931
Formula: C26H22Cl2N4O3
DC8280
>98%
BLU9931 is the first selective small molecule inhibitor of FGFR4 with IC50 of 3 nM; less potent for FGFR1/2/3(IC50> 150 nM).
BLU554
CAS:1707289-21-1
Trade Name: BLU-554,BLU 554
Formula: C24H24Cl2N4O4
DC10092
>98%
BLU-554 is a potent fibroblast growth factor receptor 4 (FGFR4) inhibitor.
BLZ945
CAS:953769-46-5
Trade Name: BLZ-945,BLZ 945
Formula: C20H22N4O3S
DC8103
>98%
BLZ945 is a highly selective and brain-penetrant inhibitor of CSF1R with IC50 of 1 nM; >3200-fold higher than its affinity for other kinases.
BM212
CAS:146204-42-4
Trade Name: BM 212,BM-212
Formula: C23H25Cl2N3
DC9853
>98%
BM-212 is a potent antimycobacterial agent and MmpL3 inhibitor.
BMH-21
CAS:896705-16-1
Trade Name: BMH 21,BMH21
Formula: C21H20N4O2
DC7959
>98%
BMH-21 is a small molecule DNA intercalator that binds ribosomal DNA and inhibits RNA polymerase I transcription; does not cause phosphorylation of H2AX.
BML-190
CAS:2854-32-2
Trade Name: BML-190,BML 190,BML190
Formula: C23H23ClN2O4
DC7840
>98%
BML-190 is an indomethacin morpholinylamide which functions as a selective inverse agonist of the human cannabinoid CB2 receptor.
BML-210(CAY10433)
CAS:537034-17-6
Trade Name: BML210; BML 210,CAY10433,CAY-10433,CAY 10433
Formula: C20H25N3O2
DC8660
>98%
BML-210 is the novel HDAC inhibitor, and its mechanism of action has not been characterized.
BML-277
CAS:516480-79-8
Trade Name: Chk2 Inhibitor II; C 3742; BML277; BML 277
Formula: C20H14ClN3O2
DC8270
>98%
BML-277 (C 3742) is a selective Chk2 (checkpoint kinase 2) inhibitor with an IC50 of 15 nM.
BMN-673 8R,9S
CAS:1207456-00-5
Trade Name: Talazoparib (8R,9S); (8R,9S)-BMN-673; BMN673 (8R,9S); BMN 673 (8R,9S)
Formula: C19H14F2N6O
DC8452
>95%,ee>92%
BMN-673 (8R,9S) is the (8R,9S) enantiomer of BMN-673. BMN 673 is a novel PARP inhibitor with IC50 of 0.58 nM(PARP1). It does not inhibit PARG and is highly sensitive to PTEN mutation.
BMS-2
CAS:888719-03-7
Trade Name: BMS2,BMS 2
Formula: C25H16F2N4O3
DC8515
>98%
BMS-2 is a potent MET kinase inhibitor with an IC50 value of 1.8nM. It also possesses potent inhibitory activity against Flt-3 and VEGFR-2 kinases, IC50 values of 4nM and 27nM respectively.
BMS-207147/RAVUCONAZOLE
CAS:182760-06-1
Formula: C22H17F2N5OS
DC9207
>98%
BMS-214662
CAS:195987-41-8
Trade Name: BMS214662; BMS 214662
Formula: C25H23N5O2S2
DC10200
>98%
BMS-214662 is a potent and selective farnesyl transferase inhibitor with potent antitumor activity with an IC50 of 1.35 nM.
BMS-265246
CAS:582315-72-8
Trade Name: BMS265246; BMS 265246
Formula: C18H17F2N3O2
DC8762
>98%
BMS-265246 is a potent and selective CDK1/2 inhibitor for CDK1/cyclin B and CDK2/cyclin E with IC50 of 6 nM and 9 nM, respectively.
BMS-3
CAS:1338247-30-5
Trade Name: BMS3;BMS 3,BMS-3
Formula: C17H12Cl2F2N4OS
DC8513
>98%
BMS-3 is a potent inhibitor of the LIM kinase. It has IC50's of 5nM and 6 nM for LIMK1 and LIMK2 respectively.
BMS-303141
CAS:943962-47-8
Trade Name: BMS303141; BMS 303141
Formula: C19H15Cl2NO4S
DC7375
>98%
BMS-303141 is a potent ATP-citrate lyase (ACL) inhibitor with IC50 value of 0.13 uM (human recombinant ACL).
BMS-309403
CAS:300657-03-8
Trade Name: BMS 309403,BMS309403
Formula: C31H26N2O3
DC8457
>98%
BMS309403 is orally active, reducing atherosclerosis in mice lacking apoplipoprotein E.
BMS-345541
CAS:547757-23-3
Trade Name: BMS345541 hydrochloride; BMS-345541 hydrochloride; BMS 345541 hydrochloride
Formula: C14H18ClN5
DC8761
>98%
BMS-345541 is a highly selective inhibitor of the catalytic subunits of IKK-2 and IKK-1 with IC50 of 0.3 M and 4 M, respectively.
BMS-5
CAS:1338247-35-0
Trade Name: BMS 5;BMS5
Formula: C17H14Cl2F2N4OS
DC8516
>98%
BMS-5 is a potent inhibitor of the LIM kinase. It has IC50 values of 7nM and 8 nM for LIMK1 and LIMK2 respectively.
BMS-536924
CAS:468740-43-4
Trade Name: BMS 536924,BMS536924
Formula: C25H26ClN5O3
DC5037
>98%
BMS-536924 is an ATP-competitive IGF-1R inhibitor with IC50 of 100 nM, modest activity for Mek, Fak, and Lck with very little activity for Akt1, MAPK1/2.
BMS-538203
CAS:543730-41-2
Trade Name: BMS538203; BMS 538203
Formula: C12H12FNO5
DC7007
>98%
BMS-538203 is a highly efficient HIV integrase inhibitor and antiviral agent.
BMS-582949 HCL
CAS:623152-17-0
Trade Name: BMS 582949, BMS582949
Formula: C22H26N6O2.HCl
DC7897
>98%
BMS-582949 is a dual action p38 Kinase Inhibitor.
BMS-599626 (AC480)
CAS:714971-09-2
Trade Name: BMS599626,AC-480, BMS 599626 (AC480)
Formula: C27H27FN8O3.HCL
DC3105
>98%
BMS-599626 (AC480) is a selective and efficacious inhibitor of HER1 and HER2 with IC50 of 20 nM and 30 nM, respectively.